التفاصيل البيبلوغرافية
العنوان: |
Discovery of Pyridopyrimidinones that Selectively Inhibit the H1047R PI3Kα Mutant Protein |
المؤلفون: |
Ketcham, John M., Harwood, Stephen J., Aranda, Ruth, Aloiau, Athenea N., Bobek, Briana M., Briere, David M., Burns, Aaron C., Caddell Haatveit, Kersti, Calinisan, Andrew, Clarine, Jeffery, Elliott, Adam, Engstrom, Lars D., Gunn, Robin J., Ivetac, Anthony, Jones, Benjamin, Kuehler, Jon, Lawson, J. David, Nguyen, Natalie, Parker, Cody, Pearson, Kelly E., Rahbaek, Lisa, Saechao, Barbara, Wang, Xiaolun, Waters, Anna, Waters, Laura, Watkins, Ashlee H., Olson, Peter, Smith, Christopher R., Christensen, James G., Marx, Matthew A. |
المساهمون: |
Mirati Therapeutics |
المصدر: |
Journal of Medicinal Chemistry ; volume 67, issue 6, page 4936-4949 ; ISSN 0022-2623 1520-4804 |
بيانات النشر: |
American Chemical Society (ACS) |
سنة النشر: |
2024 |
مصطلحات موضوعية: |
Drug Discovery, Molecular Medicine |
نوع الوثيقة: |
article in journal/newspaper |
اللغة: |
English |
DOI: |
10.1021/acs.jmedchem.4c00078 |
الإتاحة: |
https://doi.org/10.1021/acs.jmedchem.4c00078Test |
حقوق: |
https://creativecommons.org/licenses/by-nc-nd/4.0Test/ |
رقم الانضمام: |
edsbas.45ED2E98 |
قاعدة البيانات: |
BASE |