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المؤلفون: Sanket J, Mishra, Weiya, Liu, Kristin, Beebe, Monimoy, Banerjee, Caitlin N, Kent, Vitumbiko, Munthali, John, Koren, John A, Taylor, Leonard M, Neckers, Jeffrey, Holzbeierlein, Brian S J, Blagg
المصدر: J Med Chem
مصطلحات موضوعية: Models, Molecular, Protein Folding, Molecular Conformation, Antineoplastic Agents, Heterocyclic Compounds, 4 or More Rings, Article, Substrate Specificity, Small Molecule Libraries, Structure-Activity Relationship, Urinary Bladder Neoplasms, Cell Line, Tumor, Neoplasms, polycyclic compounds, Humans, Gene Silencing, HSP90 Heat-Shock Proteins, Cell Proliferation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::fea484f03b8f837f82dd59c679412e46Test
https://pubmed.ncbi.nlm.nih.gov/33428418Test -
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المؤلفون: Daniel T. Gewirth, Nanette L.S. Que, Adam S. Duerfeldt, Brian S. J. Blagg, Jinbo Zhao, Caitlin N. Kent, Vincent M. Crowley
المصدر: Journal of medicinal chemistry. 61(7)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Stereochemistry, Substituent, Molecular Conformation, Crystallography, X-Ray, Insert (molecular biology), Article, 03 medical and health sciences, Residue (chemistry), chemistry.chemical_compound, Structure-Activity Relationship, 0302 clinical medicine, Adenosine Triphosphate, Dogs, Drug Discovery, Imidazole, Animals, Humans, HSP70 Heat-Shock Proteins, HSP90 Heat-Shock Proteins, biology, Chemistry, Membrane Proteins, Ligand (biochemistry), Hsp90, 030104 developmental biology, Cytoplasm, 030220 oncology & carcinogenesis, Drug Design, biology.protein, Molecular Medicine, Structure based, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ccca754a8ee05065988cd16059cab867Test
https://pubmed.ncbi.nlm.nih.gov/29528635Test