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المؤلفون: Victor Moreno, Noelia Nebot, Emmanuel Bouillaud, Dung-Yang Lee, Eva Muñoz-Couselo, Christina S. Won, Eduard Gasal
المساهمون: Institut Català de la Salut, [Nebot N, Lee DY, Gasal E] Novartis Pharmaceuticals Corporation, East Hanover, New Jersey, USA. [Won CS] Novartis Institutes for BioMedical Research, East Hanover, New Jersey, USA. [Moreno V] START Madrid-FJD, Hospital Universitario Fundación Jiménez Díaz, Madrid, Spain. [Muñoz-Couselo E] Vall d’Hebron Institute of Oncology (VHIO), Barcelona, Spain. Vall d’Hebron Hospital Universitari, Barcelona, Spain. [Bouillaud E] Novartis Pharma AG, Basel, Switzerland, Vall d'Hebron Barcelona Hospital Campus
المصدر: Clinical Pharmacology in Drug Development
Scientiaمصطلحات موضوعية: Male, CYP3A4, CYP3A, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, fenómenos fisiológicos::fenómenos farmacológicos y toxicológicos::fenómenos farmacológicos::interacciones farmacológicas [FENÓMENOS Y PROCESOS], 0302 clinical medicine, Oximes, Medicine, fenómenos fisiológicos::fenómenos farmacológicos y toxicológicos::farmacocinética [FENÓMENOS Y PROCESOS], Cytochrome P-450 CYP3A, Pharmacology (medical), Drug Interactions, Rosuvastatin Calcium, OATP, Liver-Specific Organic Anion Transporter 1, Imidazoles, Articles, Middle Aged, Other subheadings::/pharmacology [Other subheadings], Physiological Phenomena::Pharmacological and Toxicological Phenomena::Pharmacokinetics [PHENOMENA AND PROCESSES], 030220 oncology & carcinogenesis, Area Under Curve, Female, pharmacokinetics, medicine.drug, Adult, Midazolam, Cmax, Original Manuscript, transporters, Chemical Actions and Uses::Pharmacologic Actions::Molecular Mechanisms of Pharmacological Action::Enzyme Inhibitors::Protein Kinase Inhibitors [CHEMICALS AND DRUGS], 03 medical and health sciences, Solute Carrier Organic Anion Transporter Family Member 1B3, Pharmacokinetics, Humans, Rosuvastatin, dabrafenib, Protein Kinase Inhibitors, drug interaction, Farmacocinètica, business.industry, acciones y usos químicos::acciones farmacológicas::mecanismos moleculares de acción farmacológica::inhibidores enzimáticos::inhibidores de proteínas cinasas [COMPUESTOS QUÍMICOS Y DROGAS], Dabrafenib, Drug interaction, Medicaments - Interacció, Proteïnes quinases - Inhibidors, Physiological Phenomena::Pharmacological and Toxicological Phenomena::Pharmacological Phenomena::Drug Interactions [PHENOMENA AND PROCESSES], Otros calificadores::/farmacología [Otros calificadores], business
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7adef14bde6abca56c9d91bfe2b8074dTest
http://europepmc.org/articles/PMC8453865Test -
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المؤلفون: Christina S. Won, Lai Wang, Jocelyn Zhou, Sam Rebello, Heidi J. Einolf
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(4)
مصطلحات موضوعية: Drug, Adult, Male, Physiologically based pharmacokinetic modelling, Time Factors, CYP3A, Metabolic Clearance Rate, Pyridines, media_common.quotation_subject, Cmax, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, Sonidegib, 03 medical and health sciences, chemistry.chemical_compound, Young Adult, 0302 clinical medicine, Pharmacokinetics, Neoplasms, Medicine, Cytochrome P-450 CYP3A, Humans, Computer Simulation, Drug Interactions, Dosing, media_common, business.industry, Biphenyl Compounds, Cytochrome P-450 CYP3A Inducers, Middle Aged, Smoothened Receptor, Healthy Volunteers, Ketoconazole, chemistry, 030220 oncology & carcinogenesis, Cytochrome P-450 CYP3A Inhibitors, Female, Rifampin, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19413d02d53b18c1ea6a8a9c3fe17ae9Test
https://pubmed.ncbi.nlm.nih.gov/28122787Test -
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المؤلفون: Xuemin, Jiang, Catherine, Dutreix, Venkateswar, Jarugula, Sam, Rebello, Christina S, Won, Haiying, Sun
المصدر: Clinical pharmacology in drug development. 6(1)
مصطلحات موضوعية: Adult, Male, Young Adult, Cytochrome P-450 CYP3A Inducers, Humans, Drug Interactions, Female, Middle Aged, Models, Theoretical, Rifampin, Healthy Volunteers, Hydroxycholesterols
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::bba78f433852d3f98a1b368751963000Test
https://pubmed.ncbi.nlm.nih.gov/27138546Test -
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المؤلفون: Christina S, Won, Tian, Lan, Karen M, Vandermolen, Paul A, Dawson, Nicholas H, Oberlies, Wilbur W, Widmer, Yolanda V, Scarlett, Mary F, Paine
المصدر: Journal of clinical pharmacology. 53(9)
مصطلحات موضوعية: Adult, Flavonoids, Male, Cross-Over Studies, Estrone, food and beverages, Organic Anion Transporters, Middle Aged, Article, Beverages, Food-Drug Interactions, Young Adult, HEK293 Cells, Coumarins, Fruit, Anti-Allergic Agents, COS Cells, Chlorocebus aethiops, Animals, Humans, Female, Terfenadine, Citrus paradisi
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::d82da768f1288bbddc92756b034f2689Test
https://pubmed.ncbi.nlm.nih.gov/23878024Test