نتائج البحث - "Katzenellenbogen, John A"

1

دورية أكاديمية

Asymmetric allostery in estrogen receptor-a homodimers drives responses to the ensemble of estrogens in the hormonal milieu.

المؤلفون: Min, Charles K., Nwachukwu, Jerome C., Yingwei Hou, Russo, Robin J., Papa, Alexandra, Jian Min, Rouming Peng, Sung Hoon Kim, Yvonne Ziegler, Rangarajan, Erumbi S., Izard, Tina, Katzenellenbogen, Benita S., Katzenellenbogen, John A., Nettles, Kendall W.

المصدر: Proceedings of the National Academy of Sciences of the United States of America; 6/11/2024, Vol. 121 Issue 24, p1-50, 50p

مصطلحات موضوعية: HOMODIMERS, LIGAND binding (Biochemistry), LIGANDS (Biochemistry), MOLECULAR dynamics, BINDING sites

2

دورية أكاديمية

Optimization of the preparation of fluorine-18-labeled steroid receptor ligands 16alpha-[¹⁸F]fluoroestradiol (FES), [¹⁸F]fluoro furanyl norprogesterone (FFNP), and 16beta-[¹⁸F]fluoro-5alpha-dihydrotestosterone (FDHT) as radiopharmaceuticals

المؤلفون: Zhou, Dong, Lin, Mai, Yasui, Norio, Al ‐ Qahtani, Mohammed H., Dence, Carmen S., Schwarz, Sally, Katzenellenbogen, John A.

المصدر: Journal of Labelled Compounds & Radiopharmaceuticals; May2014, Vol. 57 Issue 5, p371-377, 7p

مصطلحات موضوعية: FLUORINE, STEROID receptors, LIGANDS (Biochemistry), ESTRADIOL, PROGESTERONE, STANOLONE, RADIOPHARMACEUTICALS

3

دورية أكاديمية

Estrogen receptor β ligands: Recent advances and biomedical applications.

المؤلفون: Minutolo, Filippo, Macchia, Marco, Katzenellenbogen, Benita S., Katzenellenbogen, John A.

المصدر: Medicinal Research Reviews; May2011, Vol. 31 Issue 3, p364-442, 79p, 8 Charts, 76 Graphs

مصطلحات موضوعية: ESTROGEN receptors, PATHOLOGY, LIGANDS (Biochemistry), STEROID hormones, SEX hormones, THERAPEUTICS

4

دورية أكاديمية

A dual-acceptor time-resolved Föster resonance energy transfer assay for simultaneous determination of thyroid hormone regulation of corepressor and coactivator binding to the thyroid hormone receptor: Mimicking the cellular context of thyroid hormone action

المؤلفون: Jeyakumar, M.¹, Katzenellenbogen, John A. jkatzene@uiuc.edu

المصدر: Analytical Biochemistry. Mar2009, Vol. 386 Issue 1, p73-78. 6p.

مصطلحات موضوعية: *THYROID hormones, *ENERGY transfer, *HORMONE receptors, *LIGANDS (Biochemistry), *FLUORESCEIN, *HIGH throughput screening (Drug development)

5

دورية أكاديمية

NFκB selectivity of estrogen receptor ligands revealed by comparative crystallographic analyses.

المؤلفون: Nettles, Kendall W., Bruning, John B., Gil, German, Nowak, Jason, Sharma, Sanjay K., Hahm, Johnnie B., Kulp, Kristen, Hochberg, Richard B., Haibing Zhou, Katzenellenbogen, John A., Katzenellenbogen, Benita S., Younchang Kim, Joachmiak, Andrzej, Greene, Geoffrey L.

المصدر: Nature Chemical Biology; Apr2008, Vol. 4 Issue 4, p241-247, 7p, 4 Diagrams, 3 Graphs

مصطلحات موضوعية: ESTROGEN receptors, LIGANDS (Biochemistry), BIOCHEMISTRY, HORMONE receptors, GENE expression

6

دورية أكاديمية

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism.

المؤلفون: Shiau, Andrew K., Barstad, Danielle, Radek, James T., Meyers, Marvin J., Nettles, Kendall W., Katzenellenbogen, Benita S., Katzenellenbogen, John A., Agard, David A., Greene, Geoffrey L.

المصدر: Nature Structural Biology; May2002, Vol. 9 Issue 5, p359, 6p

مصطلحات موضوعية: LIGANDS (Biochemistry), ESTROGEN receptors, ESTROGEN antagonists

7

دورية أكاديمية

Corrigendum: NFκB selectivity of estrogen receptor ligands revealed by comparative crystallographic analyses.

المؤلفون: Nettles, Kendall W, Bruning, John B, Gil, German, Nowak, Jason, Sharma, Sanjay K, Hahm, Johnnie B, Kulp, Kristen, Hochberg, Richard B, Zhou, Haibing, Katzenellenbogen, John A, Katzenellenbogen, Benita S, Kim, Younchang, Joachimiak, Andrzej, Greene, Geoffrey L

المصدر: Nature Chemical Biology; Jun2008, Vol. 4 Issue 6, p379-379, 1p, 1 Graph

مصطلحات موضوعية: LIGANDS (Biochemistry)

8

دورية أكاديمية

Synthesis and evaluation of aryl-substituted diarylpropionitriles, selective ligands for estrogen receptor β, as positron-emission tomographic imaging agents

المؤلفون: Moon, Byung Seok^1,2, Carlson, Kathryn E.³, Katzenellenbogen, John A.³, Choi, Tae Hyun¹, Chi, Dae Yoon⁴, Kim, Jung Young¹, Cheon, Gi Jeong¹, Koh, Hun Yeong², Lee, Kyo Chul¹ kyochul@kirams.re.kr, An, Gwangil¹ gwangil@kirams.re.kr

المصدر: Bioorganic & Medicinal Chemistry. May2009, Vol. 17 Issue 9, p3479-3488. 10p.

مصطلحات موضوعية: *ORGANIC synthesis, *LIGANDS (Biochemistry), *ESTROGEN receptors, *POSITRON emission, *POSITRON emission tomography, *BREAST tumors

9

دورية أكاديمية

Exploration of the bicyclo[3.3.1]nonane system as a template for the development of new ligands for the estrogen receptor

المؤلفون: Muthyala, Rajeev S.¹, Carlson, Kathryn E.¹, Katzenellenbogen, John A. jkatzene@uiuc.edu

المصدر: Bioorganic & Medicinal Chemistry Letters. Dec2003, Vol. 13 Issue 24, p4485. 4p.

مصطلحات موضوعية: *CYCLIC compounds, *LIGANDS (Biochemistry), *ESTROGEN receptors

10

دورية أكاديمية

Adamantyl Antiestrogens with Novel Side Chains Reveal a Spectrum of Activities in Suppressing Estrogen Receptor Mediated Activities in Breast Cancer Cells.

المؤلفون: Jian Min¹, Guillen, Valeria Sanabria², Sharma, Abhishek¹, Yuechao Zhao², Yvonne Ziegler², Ping Gong², Mayne, Christopher G.³, Srinivasan, Sathish⁴, Sung Hoon Kim¹, Carlson, Kathryn E.¹, Nettles, Kendall W.⁴, Katzenellenbogen, Benita S.², Katzenellenbogen, John A.¹ jkatzene@illinois.edu

المصدر: Journal of Medicinal Chemistry. 7/27/2017, Vol. 60 Issue 14, p6321-6336. 16p.

مصطلحات موضوعية: *ESTROGEN antagonists, *BREAST cancer treatment, *LYMPHADENECTOMY, *LIGANDS (Biochemistry), *BIOCHEMISTRY, *THERAPEUTICS

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