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1
المؤلفون: Andrea Cavalli, Anna Minarini, Antonino Cattaneo, Michela Rosini, Andrea Tarozzi, Vincenza Andrisano, Maria Laura Bolognesi, Patrizia Hrelia, Giorgio Lenaz, Rita Banzi, Manuela Bartolini, Christian Bergamini, Carlo Melchiorre, Romana Fato, Vincenzo Tumiatti, Maurizio Recanatini
المساهمون: Bolognesi ML, Banzi R, Bartolini M, Cavalli A, Tarozzi A, Andrisano V, Minarini A, Rosini M, Tumiatti V, Bergamini C, Fato R, Lenaz G, Hrelia P, Cattaneo A, Recanatini M, Melchiorre C., Bolognesi, Ml, Banzi, R, Bartolini, M, Cavalli, A, Tarozzi, A, Andrisano, V, Minarini, A, Rosini, M, Tumiatti, V, Bergamini, C, Fato, R, Lenaz, G, Hrelia, P, Cattaneo, Antonino, Recanatini, M, Melchiorre, C.
المصدر: Journal of medicinal chemistry. 50(20)
مصطلحات موضوعية: Models, Molecular, Amyloid beta, Plasma protein binding, medicine.disease_cause, Ligands, Antioxidants, MULTITARGET, Cell Line, Substrate Specificity, chemistry.chemical_compound, Structure-Activity Relationship, Alzheimer Disease, Drug Discovery, medicine, NAD(P)H Dehydrogenase (Quinone), Polyamines, Structure–activity relationship, Humans, Binding site, Butyrylcholinesterase, Amyloid beta-Peptides, Binding Sites, biology, Chemistry, Quinones, medicine.disease, AMYLOID-BETA, Acetylcholinesterase, Oxidative Stress, Biochemistry, ALZHEIMER'S DISEASE, biology.protein, Molecular Medicine, Cholinesterase Inhibitors, Alzheimer's disease, Reactive Oxygen Species, Oxidative stress, Protein Binding
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f1ae0f0f5155ca76a5f3596bd588cb39Test
https://pubmed.ncbi.nlm.nih.gov/17850125Test -
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المساهمون: Melchiorre C, Bolognesi ML, Minarini A, Rosini M, Tumiatti V
المصدر: Journal of Medicinal Chemistry. 53:5906-5914
مصطلحات موضوعية: Structure-Activity Relationship, Chemistry, Drug discovery, Drug Design, Models, Animal, Drug Discovery, Polyamines, Animals, Molecular Medicine, Design strategy, Ligands, Ligand (biochemistry), Combinatorial chemistry
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::22b5c2965b7f4133b33fcaddd8fb04e3Test
https://doi.org/10.1021/jm100293fTest -
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المؤلفون: Carlo Melchiorre, Maria Laura Bolognesi, Anna Minarini, Michela Rosini, Elena Simoni, Vincenzo Tumiatti
المساهمون: Bolognesi M.L., Simoni E., Rosini M., Minarini A., Tumiatti V., Melchiorre C
مصطلحات موضوعية: Drug, media_common.quotation_subject, Computational biology, Disease, Pharmacology, Ligands, Alzheimer Disease, Alkanes, medicine, Ethylamines, Animals, Humans, Enzyme Inhibitors, media_common, Amyloid beta-Peptides, Thioctic Acid, Drug discovery, business.industry, General Medicine, DRUG DISCOVERY, Tacrine, Molecular targets, Acetylcholinesterase, business, NEURODEGENERATIVE DISEASES, medicine.drug
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fd763a546e1db61961b2fdbedbe66576Test
http://hdl.handle.net/11585/108616Test -
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المؤلفون: Gianpaolo Chiriano, Maria Laura Bolognesi, Giovanni Bottegoni, Manfred Windisch, Vincenzo Tumiatti, Michela Rosini, Carlo Melchiorre, Manuela Bartolini, Andrea Cavalli, Vincenza Andrisano, Valentina Maestri, Anna Minarini, Stefan Czvitkovich, Francesca Mancini
المساهمون: Bolognesi ML, Chiriano G, Bartolini M, Mancini F, Bottegoni G, Maestri V, Czvitkovich S, Windisch M, Cavalli A, Minarini A, Rosini M, Tumiatti V, Andrisano V, Melchiorre C.
مصطلحات موضوعية: Models, Molecular, Aché, Stereochemistry, Cell Survival, Molecular Conformation, In Vitro Techniques, Ligands, Bivalent (genetics), chemistry.chemical_compound, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Alkanes, Ethylamines, Animals, Humans, Neurons, Amyloid beta-Peptides, ALZHEIMER’S DISEASE, Affinities, language.human_language, In vitro, Peptide Fragments, APP metabolism, Monomer, chemistry, Butyrylcholinesterase, Amyloid aggregation, language, Acetylcholinesterase, Molecular Medicine, Cholinesterase Inhibitors, Amyloid Precursor Protein Secretases, Chickens, Protein Binding
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6915ab35436d2c99c205c324dfb6ba17Test
http://hdl.handle.net/11585/109307Test -
5
المؤلفون: Vincenza Andrisano, Michela Rosini, Maria Laura Bolognesi, Manuela Bartolini, Carlo Melchiorre, Romana Fato, Giorgio Lenaz, Andrea Cavalli, Christian Bergamini
المساهمون: Bolognesi ML, Cavalli A, Bergamini C, Fato R, Lenaz G, Rosini M, Bartolini M, Andrisano V, Melchiorre C.
مصطلحات موضوعية: Antioxidant, medicine.drug_class, Ubiquinone, medicine.medical_treatment, Submitochondrial Particles, Carboxamide, Ligands, Antioxidants, Electron Transport, chemistry.chemical_compound, Alzheimer Disease, Cell Line, Tumor, Drug Discovery, Alkanes, medicine, Ethylamines, Humans, Amyloid beta-Peptides, biology, Thioctic Acid, Rational design, Acetylcholinesterase, Benzoquinone, Lipoic acid, chemistry, Biochemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Reactive Oxygen Species, Function (biology), Protein Binding
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::059ee8f15e58e064ed3cec87811cd724Test
http://hdl.handle.net/11585/84134Test -
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المؤلفون: Maria Laura Bolognesi, Manuela Bartolini, Carlo Melchiorre, Vincenza Andrisano, Andrea Cavalli, Maurizio Recanatini, Michela Rosini, Luca Valgimigli
المساهمون: Bolognesi ML, Cavalli A, Valgimigli L, Bartolini M, Rosini M, Andrisano V, Recanatini M, Melchiorre C
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Ligands, Ferric Compounds, Structure-Activity Relationship, chemistry.chemical_compound, Alzheimer Disease, Drug Discovery, medicine, Humans, Structure–activity relationship, Binding site, Chelating Agents, Amyloid beta-Peptides, Binding Sites, biology, Biological activity, Acetylcholinesterase, Peptide Fragments, chemistry, Acetylcholinesterase inhibitor, Biochemistry, Enzyme inhibitor, Butyrylcholinesterase, Drug Design, Tacrine, biology.protein, Thermodynamics, Molecular Medicine, Cholinesterase Inhibitors, Lead compound, Copper, medicine.drug
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6e7b237e16654741393b4fff129e7597Test
http://hdl.handle.net/11585/52760Test -
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المؤلفون: Maria Laura Bolognesi, Vincenza Andrisano, Rita Banzi, Carlo Melchiorre, Manuela Bartolini
المساهمون: BOLOGNESI M. L., ANDRISANO V., BARTOLINI M., BANZI R., MELCHIORRE C.
مصطلحات موضوعية: Aché, Drug Evaluation, Preclinical, Ligands, Biochemistry, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, Polyamines, Structure–activity relationship, Humans, Fluorometry, chemistry.chemical_classification, Amyloid beta-Peptides, biology, Hydrolysis, Biological activity, Acetylcholinesterase, In vitro, language.human_language, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, language, Molecular Medicine, Cholinesterase Inhibitors, Polyamine, Dimerization, Propidium
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd0aac2a7b660a7816e77ebb0a839385Test
http://hdl.handle.net/11585/1821Test