-
1
المؤلفون: Dominika E. Butler, Anne T. Collins, Matthew S. Simms, Christopher R. Marlein, Barry R. Davies, Fiona M. Frame, Norman J. Maitland, Hannah F. Walker, Vincent M. Mann
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, MAPK/ERK pathway, medicine.medical_specialty, autophagy, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Internal medicine, LNCaP, medicine, PTEN, Protein kinase B, PI3K/AKT/mTOR pathway, biology, business.industry, Kinase, AKT, RPTOR, medicine.disease, prostate cancer, 030104 developmental biology, Endocrinology, Oncology, 030220 oncology & carcinogenesis, MAPK signalling, Cancer research, biology.protein, mTOR, business, Research Paper, RAS
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4954da09786e316b749b3fba977b5899Test
http://europepmc.org/articles/PMC5593594Test -
2
المؤلفون: Charlene Fallan, Derek Barratt, Gillian M. Lamont, Elaine Cadogan, Frederick W. Goldberg, Mercedes Vazquez-Chantada, Antonio Ramos Montoya, Anna Cronin, Simon J. Hollingsworth, Andrew D. Campbell, D. Beattie, Raymond AstraZeneca R D Alderley Finlay, Jacqueline H. L. Fok, Emma Dean, Joanna Harding, Jane Norris, Attilla Ting, Barry R. Davies
المصدر: Cancer Research. 79:DDT01-02
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Kinase, DNA damage, DNA repair, Poly ADP ribose polymerase, Olaparib, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Oncology, chemistry, In vivo, 030220 oncology & carcinogenesis, Cancer research, Growth inhibition, IC50
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::55596045c1b3fd811eba667906d5e018Test
https://doi.org/10.1158/1538-7445.am2019-ddt01-02Test -
3
المؤلفون: Michael Ittmann, Peter S. Nelson, Paul D. Smith, Barry R. Davies, Shu Feng, Longjiang Shao, Ilsa Coleman, Patricia Castro
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, MAPK/ERK pathway, Male, STAT3 Transcription Factor, medicine.medical_specialty, kinase inhibitor, Mice, SCID, Fibroblast growth factor, Piperazines, 03 medical and health sciences, Internal medicine, Cell Line, Tumor, Antineoplastic Combined Chemotherapy Protocols, medicine, Animals, Humans, Pyrroles, Receptor, Fibroblast Growth Factor, Type 1, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein kinase B, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Cell Proliferation, Dose-Response Relationship, Drug, Kinase, business.industry, Fibroblast growth factor receptor 1, AKT, fibroblast growth factors, Prostatic Neoplasms, prostate cancer, Xenograft Model Antitumor Assays, 3. Good health, Tumor Burden, 030104 developmental biology, Endocrinology, Pyrimidines, Oncology, Fibroblast growth factor receptor, Benzamides, Cancer research, Pyrazoles, Signal transduction, business, Proto-Oncogene Proteins c-akt, signal transduction, Research Paper
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a286cbf59b00d90c15d81932e9cb0d4eTest
https://pubmed.ncbi.nlm.nih.gov/28008155Test -
4
المؤلفون: Neil H. James, Valeria Follia, Ankur Karmokar, Barry R. Davies, Jacqueline H. L. Fok, Emma Dean, Mercedes Vazquez-Chantada, Simon J. Hollingsworth, Antonio Ramos-Montoya, Lenka Oplustil O'Connor, Paul W. G. Wijnhoven, Anna Staniszewska, Elaine Cadogan
المصدر: Cancer Research. 79:3506-3506
مصطلحات موضوعية: Protein kinase complex, Cancer Research, Chemistry, Kinase, Cell growth, DNA damage, Cell, Olaparib, chemistry.chemical_compound, medicine.anatomical_structure, Oncology, PARP inhibitor, medicine, Cancer research, Growth inhibition
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::fed19919befdfb163b13b2d262815543Test
https://doi.org/10.1158/1538-7445.am2019-3506Test -
5
المؤلفون: Emma Dean, Antonio Ramos-Montoya, Elaine Cadogan, Jacqueline H. L. Fok, Lenka Oplustil O'Connor, Barry R. Davies, Neil H. James, Paul Winjhoven, Valeria Follia, Ankur Karmokar, Anna Staniszewska, Mercedes Vazquez-Chantada, Simon J. Hollingsworth
المصدر: Cancer Research. 79:3505-3505
مصطلحات موضوعية: Protein kinase complex, A549 cell, Cancer Research, chemistry.chemical_compound, Oncology, DNA damage, Chemistry, Kinase, DNA repair, Poly ADP ribose polymerase, Cancer research, Growth inhibition, Olaparib
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::d3da36654f442068097cfc48c3d5f6e7Test
https://doi.org/10.1158/1538-7445.am2019-3505Test -
6
المؤلفون: Eeva Sommer, Dario R. Alessi, Barry R. Davies, Darren Cross, Sylvie Guichard, Hannah Dry
المصدر: Biochemical Journal. 452:499-508
مصطلحات موضوعية: Molecular Sequence Data, Breast Neoplasms, Signal transduction inhibitor, Protein Serine-Threonine Kinases, Biology, Biochemistry, mTORC2, Immediate early protein, Immediate-Early Proteins, Predictive Value of Tests, Cell Line, Tumor, Animals, Humans, Amino Acid Sequence, Protein Kinase Inhibitors, Molecular Biology, Protein kinase B, PI3K/AKT/mTOR pathway, Cell Proliferation, Sheep, Cell growth, Kinase, Cell Biology, Growth Inhibitors, HEK293 Cells, Drug Resistance, Neoplasm, Cancer research, Phosphorylation, Female, Proto-Oncogene Proteins c-akt
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ac6f9cdd02b445a137e64a9f423bfc8aTest
https://doi.org/10.1042/bj20130342Test -
7
المؤلفون: Morris Jeffrey James, Gordon S. Currie, Jason Grant Kettle, Claire Crafter, Clare Lane, Ken Page, Peter Ballard, Linette Ruston, Hannah Dry, Martin Pass, Andrew G. Leach, Ryan Greenwood, Matt Addie, Judit E. Debreczeni, Johnson Paul David, Barry R. Davies, Gillian M. Lamont, Donald J. Ogilvie, David Buttar, Philippa Dudley, Richard W. A. Luke, Stuart E. Pearson
المصدر: Journal of Medicinal Chemistry. 56:2059-2073
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, hERG, Administration, Oral, Carboxamide, Pharmacology, Inhibitory Concentration 50, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Humans, Structure–activity relationship, Pyrroles, Protein Kinase Inhibitors, Protein kinase B, biology, Chemistry, Kinase, Xenograft Model Antitumor Assays, Pyrimidines, Biochemistry, biology.protein, Molecular Medicine, Phosphorylation, Female, Proto-Oncogene Proteins c-akt, Drug metabolism
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9e89f0e75ec3075ae6b777ac8b9c2c94Test
https://doi.org/10.1021/jm301762vTest -
8
المؤلفون: Kazuto Nishio, Marco A. De Velasco, Hirotsugu Uemura, Yurie Kura, Kazuhiro Yoshimura, Barry R. Davies, Kazuhiro Yoshikawa, Naomi Ando Ando, Noriko Sato, Masahiro Nozawa
المصدر: Cancer Research. 78:4825-4825
مصطلحات موضوعية: Cancer Research, biology, Combination therapy, Kinase, business.industry, Cancer, medicine.disease, Prostate cancer, medicine.anatomical_structure, Oncology, Prostate, Tumor progression, medicine, Cancer research, biology.protein, PTEN, business, Protein kinase B
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::a11e2e4db32c493b2a4ebc7a83102750Test
https://doi.org/10.1158/1538-7445.am2018-4825Test -
9
المصدر: Clinical Cancer Research. 10:4874-4884
مصطلحات موضوعية: Male, MAPK/ERK pathway, Cancer Research, medicine.medical_specialty, Cell Survival, Mice, Nude, Protein Serine-Threonine Kinases, Mice, Gefitinib, Epidermal growth factor, Cell Line, Tumor, Proto-Oncogene Proteins, Internal medicine, medicine, Animals, Humans, Epidermal growth factor receptor, Phosphorylation, Protein Kinase Inhibitors, Protein kinase B, Cell Proliferation, Bladder cancer, Dose-Response Relationship, Drug, biology, Kinase, business.industry, Cell Cycle, DNA, medicine.disease, Xenograft Model Antitumor Assays, ErbB Receptors, Endocrinology, Urinary Bladder Neoplasms, Oncology, Cell culture, Quinazolines, Cancer research, biology.protein, Mitogen-Activated Protein Kinases, business, Proto-Oncogene Proteins c-akt, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b8ea0bb535841df71020973beb7fe6bTest
https://doi.org/10.1158/1078-0432.ccr-04-0034Test -
10
المؤلفون: Barry R. Davies, Noriko Sato, Naomi Ando, Kazuto Nishio, Yurie Kura, Marco A. De Velasco, Hirotsugu Uemura, Kazuhiro Yoshikawa, Dennis Huszar, Kazuko Sakai, Koichi Sugimoto, Kazuhiro Yoshimura, Masahiro Nozawa
المصدر: Cancer Research. 77:1096-1096
مصطلحات موضوعية: Cancer Research, Programmed cell death, biology, business.industry, Kinase, Cancer, medicine.disease, Prostate cancer, Oncology, Apoptosis, medicine, Cancer research, biology.protein, PTEN, Phosphorylation, business, Protein kinase B
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::13c2e4ef43cf3a07ddb74fe4dcec5712Test
https://doi.org/10.1158/1538-7445.am2017-1096Test