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المؤلفون: Judit Ovádi, Claudia A. Simões-Pires, Attila Lehotzky, Alessandra Nurisso, Philippe Bertrand, Muriel Cuendet, Nadine Martinet, Samuel Bouchet, Vincent Zwick, Christophe Blanquart
المساهمون: School of Pharmaceutical Sciences, Université de Lausanne (UNIL)-University of Geneva [Switzerland], Réseau épigénétique, Cancéropôle Grand-Ouest, Institut de Chimie des Milieux et Matériaux de Poitiers (IC2MP), Université de Poitiers-Institut national des sciences de l'Univers (INSU - CNRS)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Institut de Chimie de Nice (ICN), Université Nice Sophia Antipolis (... - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Côte d'Azur (UCA), Institute of Enzymology [Budapest], Research Centre for Natural Sciences, Hungarian Academy of Sciences (MTA)-Hungarian Academy of Sciences (MTA), Centre de Recherche en Cancérologie Nantes-Angers (CRCNA), Centre Hospitalier Universitaire d'Angers (CHU Angers), PRES Université Nantes Angers Le Mans (UNAM)-PRES Université Nantes Angers Le Mans (UNAM)-Hôtel-Dieu de Nantes-Institut National de la Santé et de la Recherche Médicale (INSERM)-Hôpital Laennec-Centre National de la Recherche Scientifique (CNRS)-Faculté de Médecine d'Angers-Centre hospitalier universitaire de Nantes (CHU Nantes), Authors thank the Centre National de la Recherche Scientifique– France, University of Poitiers, Region Poitou-Charentes (S.B. financial support), the Ligue Contre le Cancer: Committees of Vendée, et Charente-Maritime – France, ARSMeso44 – France, COST Actions CM1406 and CM1106 – Belgium and Hungarian OTKA Founds K-101039 and K-112144 for financial support. A.N. thanks the Excellence programme of the University of Geneva –Switzerland for financial support., Bernardo, Elizabeth, Université de Lausanne = University of Lausanne (UNIL)-Université de Genève = University of Geneva (UNIGE), Université Nice Sophia Antipolis (1965 - 2019) (UNS)
المصدر: Bioorganic and Medicinal Chemistry Letters
Bioorganic and Medicinal Chemistry Letters, Elsevier, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic and Medicinal Chemistry Letters, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic & Medicinal Chemistry Letters, Vol. 26, No 1 (2016) pp. 154-159مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Intrinsic activity, Formic Acid Esters, Stereochemistry, Clinical Biochemistry, Convergent synthesis, Pharmaceutical Science, [SDV.CAN]Life Sciences [q-bio]/Cancer, Alkenes, Hydroxamic Acids, Metathesis, Biochemistry, Histone Deacetylases, Catalysis, Dose-Response Relationship, Formic Acid Esters/chemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, [SDV.CAN] Life Sciences [q-bio]/Cancer, Models, Drug Discovery, Humans, Structure–activity relationship, Benzamides/chemistry, Benzamide, Molecular Biology, ddc:615, Dose-Response Relationship, Drug, Molecular Structure, biology, Organic Chemistry, Molecular, Alkenes/chemistry, 3. Good health, Histone Deacetylase Inhibitors, 030104 developmental biology, Tubulin, Histone Deacetylase Inhibitors/chemistry/pharmacology, Hydroxamic Acids/chemistry, chemistry, Benzamides, biology.protein, Molecular Medicine, Histone Deacetylases/metabolism, Drug, Selectivity
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::acc9fefa73c13b45a09cef22d951db0cTest
https://www.hal.inserm.fr/inserm-01299475/documentTest -
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المؤلفون: Jin Zhang, Zhanguo Gao, Weiping Jia, Aimin Xu, Huating Li, Xin Ye, Jianping Ye
المصدر: Diabetes
مصطلحات موضوعية: Male, Endocrinology, Diabetes and Metabolism, Mice, Obese, Mice, chemistry.chemical_compound, 0302 clinical medicine, Ketogenesis, Promoter Regions, Genetic, Hypolipidemic Agents, Mice, Knockout, chemistry.chemical_classification, 0303 health sciences, Sodium butyrate, Hep G2 Cells, 3. Good health, Butyrates, Liver, Ketone bodies, medicine.drug, Fibroblast Growth Factors - genetics - metabolism, medicine.medical_specialty, 030209 endocrinology & metabolism, Butyrate, Butyrates - pharmacology, Biology, Histone Deacetylases, 03 medical and health sciences, Internal medicine, Internal Medicine, medicine, Animals, Humans, Gene Expression Regulation - drug effects - physiology, PPAR alpha, Obesity, RNA, Messenger, 030304 developmental biology, Fatty acid, Histone Deacetylases - metabolism, HDAC3, Dietary Fats, Fibroblast Growth Factors, HEK293 Cells, Metabolism, Trichostatin A, Endocrinology, Gene Expression Regulation, chemistry, Histone deacetylase, Bezafibrate, Bezafibrate - pharmacology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a6611769b8da3912c3cf406adfaff4deTest
https://doi.org/10.2337/db11-0846Test -
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المؤلفون: Krishnan, Zhongjun Zhou, Baohua Liu
المصدر: Aging (Albany NY)
مصطلحات موضوعية: Premature aging, Aging - genetics, Aging, DNA Repair, Nuclear Proteins - chemistry - genetics - metabolism, DNA repair, Histone Acetylation, Senescence, Histone Deacetylases, Chromatin remodeling, Epigenesis, Genetic, Histones, Histone H4, Mice, Progeria, Prelamin A, Premature Aging, Humans, Animals, Histone code, Zmpste24, Protein Precursors, Lamin Type A - chemistry - genetics - metabolism, Hgps, Genetics, biology, Nuclear Proteins, Cell Biology, Lamin Type A, Histone Deacetylases - metabolism, Chromatin, Cell biology, Histone, Progeria - genetics - physiopathology, Research Perspective, Lamin A, Chromatin - chemistry - metabolism, biology.protein, Histones - metabolism, Epigenetics, DNA mismatch repair, Protein Precursors - chemistry - genetics - metabolism, DNA Damage
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2c47b742530234e85caa09b5d3770e13Test
https://doi.org/10.18632/aging.100399Test -
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المؤلفون: Fang Zhang, F. Donelson Smith, Alexandra C. Newton, Dario Diviani, Lorene K. Langeberg, John D. Scott, Joseph Soughayer, Michael R. Bristow, Maya T. Kunkel, Graeme K. Carnegie, Benjamin S. Pedroja
المصدر: Molecular Cell, vol. 32, no. 2, pp. 169-179
مصطلحات موضوعية: 14-3-3 Proteins/metabolism, A Kinase Anchor Proteins/genetics, A Kinase Anchor Proteins/metabolism, Active Transport, Cell Nucleus, Animals, COS Cells, Cardiomegaly/metabolism, Cell Line, Cercopithecus aethiops, Cyclic AMP-Dependent Protein Kinases/metabolism, Gene Expression Regulation, Guanine Nucleotide Exchange Factors/genetics, Guanine Nucleotide Exchange Factors/metabolism, Heart Ventricles/drug effects, Histone Deacetylases/metabolism, Humans, Models, Biological, Myocytes, Cardiac/drug effects, Myocytes, Cardiac/metabolism, Myogenic Regulatory Factors/metabolism, Phenylephrine/pharmacology, Phosphorylation, Protein Kinase C/metabolism, Proto-Oncogene Proteins/genetics, Proto-Oncogene Proteins/metabolism, RNA Interference, Rats, Signal Transduction, Heart Ventricles, A Kinase Anchor Proteins, Cardiomegaly, Biology, Histone Deacetylases, Article, Minor Histocompatibility Antigens, Phenylephrine, Proto-Oncogene Proteins, Chlorocebus aethiops, Guanine Nucleotide Exchange Factors, Myocytes, Cardiac, Kinase activity, Nuclear export signal, Molecular Biology, Protein Kinase C, Protein kinase C, Regulation of gene expression, Histone deacetylase 5, MEF2 Transcription Factors, Cell Biology, Cyclic AMP-Dependent Protein Kinases, Molecular biology, Cell biology, 14-3-3 Proteins, Myogenic Regulatory Factors, Histone deacetylase, Signal transduction
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::784529f321a20f89764ff93eefc37bb5Test
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المؤلفون: Michelandrea De Cesare, Muriel Cuendet, Sabrina Dallavalle, Vincent Zwick, Giuseppe Giannini, Alessandra Nurisso, Raffaella Cincinelli, Valentina Zuco, Loana Musso, Franco Zunino, Claudia A. Simões-Pires
المصدر: European Journal of Medicinal Chemistry, Vol. 112 (2016) pp. 99-105
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Antineoplastic Agents, Apoptosis, Drug Screening Assays, Hydroxamic Acids, Histone Deacetylases, Histone H4, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Neoplasms, Drug Discovery, Structure–activity relationship, Humans, Biphenyl Compounds/chemistry/pharmacology, Pharmacology, ddc:615, Neoplasms/drug therapy/metabolism, biology, Colonic Neoplasms/drug therapy/metabolism, Apoptosis/drug effects, Organic Chemistry, Biphenyl Compounds, Active site, Antitumor, General Medicine, HCT116 Cells, In vitro, Hydroxamic Acids/chemistry/pharmacology, Biphenyl compound, Histone Deacetylase Inhibitors, Molecular Docking Simulation, 030104 developmental biology, Histone Deacetylase Inhibitors/chemistry/pharmacology, chemistry, Biochemistry, Acetylation, Colonic Neoplasms, biology.protein, Histone Deacetylases/metabolism, Antineoplastic Agents/chemistry/pharmacology, Drug Screening Assays, Antitumor, Derivative (chemistry)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7c41240a5dcd709036f451727b80a3b2Test
https://pubmed.ncbi.nlm.nih.gov/26890116Test -
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المؤلفون: Zerzaihi, O., Chriett, S., Vidal, Hubert, Pirola, L.
المساهمون: Cardiovasculaire, métabolisme, diabétologie et nutrition (CarMeN), Institut National de la Recherche Agronomique (INRA)-Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Institut National des Sciences Appliquées de Lyon (INSA Lyon), Université de Lyon-Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Hospices Civils de Lyon (HCL)-Institut National de la Santé et de la Recherche Médicale (INSERM)
المصدر: ISSN: 0829-8211.
مصطلحات موضوعية: Promoter Regions, Genetic, Humans, Animals, Rats, Acetylation, Gene Expression Regulation, Transcription Initiation Site, Class Ia Phosphatidylinositol 3-Kinase/metabolism, Hexokinase/metabolism, Histone Deacetylases/metabolism, Histones/*metabolism, Insulin Receptor Substrate Proteins/metabolism, Insulin/*metabolism/pharmacology, Muscle Fibers, Skeletal/drug effects/*metabolism, Phosphatidylinositol 3-Kinases/metabolism, [SDV]Life Sciences [q-bio]
العلاقة: hal-01859362; https://hal.science/hal-01859362Test
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المؤلفون: Mathieu Boxus, Julie Lodewick, Françoise Bex, Carla Sampaio, Lucas Willems, Anne-Sophie Rinaldi, Pierre P. Roger, Katia Coulonval
المصدر: Retrovirology, 10
Retrovirologyمصطلحات موضوعية: Gene Products, tax -- metabolism, CDK4, Fibroblasts -- virology, Human T-lymphotropic virus 1 -- pathogenicity, Lysine -- metabolism, Tax, SUMO protein, P300-CBP Transcription Factors, Histone Deacetylases, p300-CBP Transcription Factors -- metabolism, Transformation, Cell Line, Ubiquitin, Virology, Animals, Humans, p300-CBP Transcription Factors, Kinase activity, Human T-lymphotropic virus 1, Histone deacetylase 5, Leukemia, biology, Physiologie de la régulation, Research, Lysine, Retinoblastoma protein, Virologie médicale, Acetylation, Gene Products, tax, Fibroblasts, Sciences bio-médicales et agricoles, Cell Transformation, Viral, Cell biology, Rats, Infectious Diseases, HTLV-1, Immunology, biology.protein, Phosphorylation, Histone Deacetylases -- metabolism, Protein Processing, Post-Translational
وصف الملف: 1 full-text file(s): application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ee701f71482c8e8e3732ac7a311293eTest
http://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/149587Test -
48دورية أكاديمية
المؤلفون: Grabiec, Aleksander M., Reedquist, Kris A.
المصدر: Grabiec , A M & Reedquist , K A 2010 , ' Histone deacetylases in RA: Epigenetics and epiphenomena ' , Arthritis Research and Therapy , vol. 12 , no. 5 , 142 . https://doi.org/10.1186/ar3137Test
مصطلحات موضوعية: Arthritis, Enzymologic, Epigenesis, Gene Expression, Gene Expression Regulation, Genetic, Histone Deacetylases, Histone Deacetylases: metabolism, Humans, Rheumatoid, Rheumatoid: enzymology, Rheumatoid: immunology, Rheumatoid: pathology, Tumor Necrosis Factor-alpha, Tumor Necrosis Factor-alpha: biosynthesis
الإتاحة: https://doi.org/10.1186/ar3137Test
https://research.manchester.ac.uk/en/publications/1353a854-a490-4f53-bbef-37ce0df6012aTest
http://arthritis-research.com/content/12/5/142Test
http://www.ncbi.nlm.nih.gov/pubmed/20959025Test http://www.pubmedcentral.nih.gov/articlerender.fcgi?artid=2991004Test\&tool=pmcentrez\&rendertype=abstract -
49دورية أكاديمية
المؤلفون: Marmolino, Daniele, Acquaviva, Fabio
المصدر: Cerebellum, 8 (3
مصطلحات موضوعية: Neurologie, Sciences bio-médicales et agricoles, Animals, Antioxidants -- pharmacology -- therapeutic use, Chlorofluorocarbons, Methane -- pharmacology -- therapeutic use, Enzyme Inhibitors -- pharmacology -- therapeutic use, Friedreich Ataxia -- drug therapy -- genetics -- therapy, Gene Silencing -- physiology, Heterochromatin -- metabolism, Histone Deacetylases -- metabolism, Histones -- metabolism, Humans, Iron -- metabolism, Iron Chelating Agents -- pharmacology -- therapeutic use, Iron-Binding Proteins -- genetics, Models, Biological, PPAR gamma -- metabolism, Signal Transduction -- drug effects, Transcription Factors -- metabolism, Trinucleotide Repeats -- genetics, Frataxin, Friedreich's ataxia, FXN gene, GAA triplet repeat, Neurodegeneration
وصف الملف: No full-text files
العلاقة: uri/info:doi/10.1007/s12311-008-0084-2; uri/info:pmid/19165552; uri/info:scp/68449096810; http://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/148500Test
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المؤلفون: Denis, Hélène, Deplus, Rachel, Putmans, Pascale, Yamada, Michiyuki, Métivier, Raphaël, Fuks, François
المصدر: Molecular and cellular biology, 29 (18
مصطلحات موضوعية: Sciences bio-médicales et agricoles, Acetylation -- drug effects, Cell Line, Chromatin -- metabolism, Chromatin Immunoprecipitation, Estradiol -- pharmacology, Histone Deacetylases -- metabolism, Histones -- metabolism, Humans, Hydrolases -- metabolism, Imines -- metabolism, Promoter Regions, Genetic -- genetics, Protein Binding -- drug effects
وصف الملف: 1 full-text file(s): application/pdf
العلاقة: uri/info:doi/10.1128/MCB.00285-09; uri/info:pii/MCB.00285-09; uri/info:pmid/19581286; uri/info:scp/70249133329; uri/info:pmcid/PMC2738279; https://dipot.ulb.ac.be/dspace/bitstream/2013/50502/1/PMC2738279.pdfTest; http://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/50502Test