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1دورية أكاديمية
المؤلفون: Krieger, Viktoria, Hamacher, Alexandra, Gertzen, Christoph, Senger, Johanna, Zwinderman, Martijn, Marek, Martin, Romier, Christophe, Dekker, Frank, Kurz, Thomas, Jung, Manfred, Gohlke, Holger, Kassack, Matthias, Hansen, Finn
المساهمون: Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Université de Strasbourg (UNISTRA)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Institut de génétique et biologie moléculaire et cellulaire (IGBMC), Université Louis Pasteur - Strasbourg I-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)
المصدر: Journal of Medical Chemistry ; https://hal.science/hal-03682266Test ; Journal of Medical Chemistry, 2017, 60 (13), pp.5493-5506. ⟨10.1021/acs.jmedchem.7b00197⟩ ; http://www.ncbi.nlm.nih.gov/pubmed/28574690Test
مصطلحات موضوعية: Antineoplastic Agents/chemical synthesis/chemistry/*pharmacology, Cell Line, Tumor, Cell Proliferation/drug effects, Dose-Response Relationship, Drug, Drug Design, Drug Screening Assays, Antitumor, Histone Deacetylase Inhibitors/chemical synthesis/chemistry/*pharmacology, Histone Deacetylases/*metabolism, Humans, Models, Molecular, Molecular Structure, Peptoids/chemical synthesis/chemistry/*pharmacology, Small Molecule Libraries/chemical synthesis/chemistry/*pharmacology, Structure-Activity Relationship, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology
العلاقة: hal-03682266; https://hal.science/hal-03682266Test
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2دورية أكاديمية
المؤلفون: Stenzel, Katharina, Hamacher, Alexandra, Hansen, Finn, Gertzen, Christoph, Senger, Johanna, Marquardt, Viktoria, Marek, Linda, Marek, Martin, Romier, Christophe, Remke, Marc, Jung, Manfred, Gohlke, Holger, Kassack, Matthias, Kurz, Thomas
المساهمون: Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Université de Strasbourg (UNISTRA)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Institut de génétique et biologie moléculaire et cellulaire (IGBMC), Université Louis Pasteur - Strasbourg I-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)
المصدر: ISSN: 0022-2623.
مصطلحات موضوعية: Dose-Response Relationship, Drug, Drug Screening Assays, Antitumor, Histone Deacetylase Inhibitors/chemical synthesis/chemistry/*pharmacology, Histone Deacetylases/*metabolism, Humans, Molecular Docking Simulation, Molecular Structure, Structure-Activity Relationship, Antineoplastic Agents/chemistry/*pharmacology, Apoptosis/drug effects, Cell Line, Tumor, Cell Proliferation/drug effects, Cisplatin/chemistry/*pharmacology, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology
العلاقة: hal-03691179; https://hal.science/hal-03691179Test
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المؤلفون: Finn K. Hansen, Christophe Romier, Linda Marek, Martin Marek, Manfred Jung, Christoph G. W. Gertzen, Johanna Senger, Katharina Stenzel, Viktoria Marquardt, Marc Remke, Thomas Kurz, Alexandra Hamacher, Holger Gohlke, Matthias U. Kassack
المساهمون: Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Université de Strasbourg (UNISTRA)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Institut de génétique et biologie moléculaire et cellulaire (IGBMC), Université Louis Pasteur - Strasbourg I-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)
المصدر: Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2017, 60 (13), pp.5334-5348. ⟨10.1021/acs.jmedchem.6b01538⟩مصطلحات موضوعية: 0301 basic medicine, Histone Deacetylases/*metabolism, Antineoplastic Agents, Apoptosis, Pharmacology, Drug Screening Assays, Cisplatin/chemistry/*pharmacology, Histone Deacetylases, Cell Line, Dose-Response Relationship, Cell Proliferation/drug effects, 03 medical and health sciences, Structure-Activity Relationship, Antineoplastic Agents/chemistry/*pharmacology, Cell Line, Tumor, Drug Discovery, medicine, Urea, Structure–activity relationship, Humans, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology, Histone Deacetylase Inhibitors/chemical synthesis/chemistry/*pharmacology, Cell Proliferation, Cisplatin, Tumor, Dose-Response Relationship, Drug, Molecular Structure, Cell growth, Chemistry, Apoptosis/drug effects, HDAC8, Antitumor, Squamous carcinoma, Histone Deacetylase Inhibitors, Molecular Docking Simulation, 030104 developmental biology, Cell culture, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor, Drug, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fae45bc45d6f85c20596af1b3e2cbe58Test
https://hal.archives-ouvertes.fr/hal-03691179Test -
4دورية أكاديمية
المؤلفون: Cincinelli, Raffaella, Zwick, Vincent, Musso, Loana, Zuco, Valentina, De Cesare, Michelandrea, Zunino, Franco, Simoes Avello, Claudia, Nurisso, Alessandra, Giannini, Giuseppe, Cuendet, Muriel, Dallavalle, Sabrina
المصدر: ISSN: 0223-5234 ; European journal of medicinal chemistry, vol. 112 (2016) p. 99-105.
مصطلحات موضوعية: info:eu-repo/classification/ddc/615, Antineoplastic Agents/chemistry/pharmacology, Apoptosis/drug effects, Biphenyl Compounds/chemistry/pharmacology, Colonic Neoplasms/drug therapy/metabolism, Drug Screening Assays, Antitumor, HCT116 Cells, Histone Deacetylase Inhibitors/chemistry/pharmacology, Histone Deacetylases/metabolism, Humans, Hydroxamic Acids/chemistry/pharmacology, Molecular Docking Simulation, Neoplasms/drug therapy/metabolism, Structure-Activity Relationship
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/26890116; https://archive-ouverte.unige.ch/unige:94976Test; unige:94976
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5دورية أكاديمية
المؤلفون: Zwick, Vincent, Simoes Avello, Claudia, Cuendet, Muriel
المصدر: ISSN: 1475-6366 ; Journal of enzyme inhibition and medicinal chemistry, vol. 31, no. sup1 (2016) p. 209-214.
مصطلحات موضوعية: info:eu-repo/classification/ddc/615, Chromatography, High Pressure Liquid, Dose-Response Relationship, Drug, Drug Evaluation, Preclinical/methods, HeLa Cells, Histone Deacetylase 1/antagonists & inhibitors/metabolism, Histone Deacetylase Inhibitors/analysis/chemistry/pharmacology, Histone Deacetylases/metabolism, Humans, Molecular Conformation, Spectrometry, Mass, Electrospray Ionization, Structure-Activity Relationship
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/27149362; https://archive-ouverte.unige.ch/unige:94975Test; unige:94975
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المؤلفون: Muriel Cuendet, Claudia A. Simões-Pires, Vincent Zwick
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 31, No sup1 (2016) pp. 209-214
مصطلحات موضوعية: 0301 basic medicine, Spectrometry, Mass, Electrospray Ionization, High-throughput screening, Cell, Drug Evaluation, Preclinical, Molecular Conformation, Histone Deacetylase 1, Pharmacology, Histone Deacetylase 6, Histone Deacetylases, Dose-Response Relationship, 03 medical and health sciences, Structure-Activity Relationship, Histone Deacetylase Inhibitors/analysis/chemistry/pharmacology, Drug Discovery, medicine, Humans, Chromatography, High Pressure Liquid, chemistry.chemical_classification, Histone Deacetylase 1/antagonists & inhibitors/metabolism, ddc:615, Chromatography, Dose-Response Relationship, Drug, biology, Drug discovery, Spectrometry, Electrospray Ionization, Cancer, General Medicine, HDAC6, Mass, medicine.disease, Histone Deacetylase Inhibitors, 030104 developmental biology, medicine.anatomical_structure, Histone, Enzyme, chemistry, Preclinical/methods, High Pressure Liquid, biology.protein, Drug Evaluation, Histone deacetylase, Histone Deacetylases/metabolism, Drug, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::883ab462cbcd9a7751ca36c6ff377bbeTest
https://archive-ouverte.unige.ch/unige:94975Test -
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المؤلفون: Judit Ovádi, Claudia A. Simões-Pires, Attila Lehotzky, Alessandra Nurisso, Philippe Bertrand, Muriel Cuendet, Nadine Martinet, Samuel Bouchet, Vincent Zwick, Christophe Blanquart
المساهمون: School of Pharmaceutical Sciences, Université de Lausanne (UNIL)-University of Geneva [Switzerland], Réseau épigénétique, Cancéropôle Grand-Ouest, Institut de Chimie des Milieux et Matériaux de Poitiers (IC2MP), Université de Poitiers-Institut national des sciences de l'Univers (INSU - CNRS)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Institut de Chimie de Nice (ICN), Université Nice Sophia Antipolis (... - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Côte d'Azur (UCA), Institute of Enzymology [Budapest], Research Centre for Natural Sciences, Hungarian Academy of Sciences (MTA)-Hungarian Academy of Sciences (MTA), Centre de Recherche en Cancérologie Nantes-Angers (CRCNA), Centre Hospitalier Universitaire d'Angers (CHU Angers), PRES Université Nantes Angers Le Mans (UNAM)-PRES Université Nantes Angers Le Mans (UNAM)-Hôtel-Dieu de Nantes-Institut National de la Santé et de la Recherche Médicale (INSERM)-Hôpital Laennec-Centre National de la Recherche Scientifique (CNRS)-Faculté de Médecine d'Angers-Centre hospitalier universitaire de Nantes (CHU Nantes), Authors thank the Centre National de la Recherche Scientifique– France, University of Poitiers, Region Poitou-Charentes (S.B. financial support), the Ligue Contre le Cancer: Committees of Vendée, et Charente-Maritime – France, ARSMeso44 – France, COST Actions CM1406 and CM1106 – Belgium and Hungarian OTKA Founds K-101039 and K-112144 for financial support. A.N. thanks the Excellence programme of the University of Geneva –Switzerland for financial support., Bernardo, Elizabeth, Université de Lausanne = University of Lausanne (UNIL)-Université de Genève = University of Geneva (UNIGE), Université Nice Sophia Antipolis (1965 - 2019) (UNS)
المصدر: Bioorganic and Medicinal Chemistry Letters
Bioorganic and Medicinal Chemistry Letters, Elsevier, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic and Medicinal Chemistry Letters, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic & Medicinal Chemistry Letters, Vol. 26, No 1 (2016) pp. 154-159مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Intrinsic activity, Formic Acid Esters, Stereochemistry, Clinical Biochemistry, Convergent synthesis, Pharmaceutical Science, [SDV.CAN]Life Sciences [q-bio]/Cancer, Alkenes, Hydroxamic Acids, Metathesis, Biochemistry, Histone Deacetylases, Catalysis, Dose-Response Relationship, Formic Acid Esters/chemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, [SDV.CAN] Life Sciences [q-bio]/Cancer, Models, Drug Discovery, Humans, Structure–activity relationship, Benzamides/chemistry, Benzamide, Molecular Biology, ddc:615, Dose-Response Relationship, Drug, Molecular Structure, biology, Organic Chemistry, Molecular, Alkenes/chemistry, 3. Good health, Histone Deacetylase Inhibitors, 030104 developmental biology, Tubulin, Histone Deacetylase Inhibitors/chemistry/pharmacology, Hydroxamic Acids/chemistry, chemistry, Benzamides, biology.protein, Molecular Medicine, Histone Deacetylases/metabolism, Drug, Selectivity
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::acc9fefa73c13b45a09cef22d951db0cTest
https://www.hal.inserm.fr/inserm-01299475/documentTest -
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المؤلفون: Michelandrea De Cesare, Muriel Cuendet, Sabrina Dallavalle, Vincent Zwick, Giuseppe Giannini, Alessandra Nurisso, Raffaella Cincinelli, Valentina Zuco, Loana Musso, Franco Zunino, Claudia A. Simões-Pires
المصدر: European Journal of Medicinal Chemistry, Vol. 112 (2016) pp. 99-105
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Antineoplastic Agents, Apoptosis, Drug Screening Assays, Hydroxamic Acids, Histone Deacetylases, Histone H4, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Neoplasms, Drug Discovery, Structure–activity relationship, Humans, Biphenyl Compounds/chemistry/pharmacology, Pharmacology, ddc:615, Neoplasms/drug therapy/metabolism, biology, Colonic Neoplasms/drug therapy/metabolism, Apoptosis/drug effects, Organic Chemistry, Biphenyl Compounds, Active site, Antitumor, General Medicine, HCT116 Cells, In vitro, Hydroxamic Acids/chemistry/pharmacology, Biphenyl compound, Histone Deacetylase Inhibitors, Molecular Docking Simulation, 030104 developmental biology, Histone Deacetylase Inhibitors/chemistry/pharmacology, chemistry, Biochemistry, Acetylation, Colonic Neoplasms, biology.protein, Histone Deacetylases/metabolism, Antineoplastic Agents/chemistry/pharmacology, Drug Screening Assays, Antitumor, Derivative (chemistry)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7c41240a5dcd709036f451727b80a3b2Test
https://pubmed.ncbi.nlm.nih.gov/26890116Test -
9دورية أكاديمية
المؤلفون: Deschamps, N., Simões-Pires, C.A., Carrupt, P.A., Nurisso, A.
المصدر: Drug Discovery Today, vol. 20, no. 6, pp. 736-742
مصطلحات موضوعية: Animals, Binding Sites, Catalytic Domain, Drug Design, Histone Deacetylase Inhibitors/chemistry, Histone Deacetylase Inhibitors/metabolism, Histone Deacetylases/chemistry, Histone Deacetylases/metabolism, Humans, Isoenzymes, Ligands, Models, Molecular, Protein Binding, Protein Conformation, Structure-Activity Relationship, Substrate Specificity
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/25597521; info:eu-repo/semantics/altIdentifier/eissn/1878-5832; https://serval.unil.ch/notice/serval:BIB_B0902461421BTest; urn:issn:1359-6446
الإتاحة: https://doi.org/10.1016/j.drudis.2015.01.004Test
https://serval.unil.ch/notice/serval:BIB_B0902461421BTest