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1دورية أكاديميةThe HIV-1 Capsid-Targeted Inhibitor GSK878 Alters Selection of Target Sites for HIV DNA Integration.
المؤلفون: Marquis, Kaitlin A., Everett, John, Cantu, Adrian, McFarland, Alexander, Sherrill-Mix, Scott, Krystal, Mark, Parcella, Kyle, Gillis, Eric, Fridell, Robert A., Bushman, Frederic D.
المصدر: AIDS Research & Human Retroviruses; Feb2024, Vol. 40 Issue 2, p114-126, 13p
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2دورية أكاديمية
المؤلفون: Parcella, Kyle1 (AUTHOR) kyle.e.parcella@viivhealthcare.com, Patel, Manoj1 (AUTHOR), Tu, Yong2 (AUTHOR), Eastman, Kyle2 (AUTHOR), Peese, Kevin1 (AUTHOR), Gillis, Eric1 (AUTHOR), Belema, Makonen2 (AUTHOR), Dicker, Ira B.1 (AUTHOR), McAuliffe, Brian1 (AUTHOR), Ding, Bo1 (AUTHOR), Falk, Paul1 (AUTHOR), Simmermacher, Jean1 (AUTHOR), Parker, Dawn D.1 (AUTHOR), Sivaprakasam, Prasanna2 (AUTHOR), Khan, Javed A.2 (AUTHOR), Kish, Kevin2 (AUTHOR), Lewis, Hal2 (AUTHOR), Hanumegowda, Umesh1 (AUTHOR), Jenkins, Susan1 (AUTHOR), Kadow, John F.1 (AUTHOR)
المصدر: Bioorganic & Medicinal Chemistry. Aug2022, Vol. 67, pN.PAG-N.PAG. 1p.
مصطلحات موضوعية: *HIV, *INTEGRASE inhibitors, *STRUCTURE-activity relationships, *LEAD compounds, *IMIDAZOPYRIDINES, *PHARMACOKINETICS