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1
المؤلفون: Eirik Sundby, Kristin G. Nørsett, Bård Helge Hoff, Silje Henriksen, Jin Han
المصدر: European Journal of Medicinal Chemistry
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, hERG, Pharmacology, Cell Line, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Drug Discovery, medicine, Humans, Potency, Pyrroles, Epidermal growth factor receptor, Cell Proliferation, ADME, EGFR inhibitors, chemistry.chemical_classification, biology, Organic Chemistry, General Medicine, EGFR, Pyrrolopyrimidine, SAR, Metabolism, Erlotinib, ErbB Receptors, Pyrimidines, 030104 developmental biology, Enzyme, Biochemistry, chemistry, Drug Design, 030220 oncology & carcinogenesis, biology.protein, Efflux, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c170e443e60845774e85f6d7385051eTest
https://doi.org/10.1016/j.ejmech.2016.08.068Test -
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المؤلفون: Kristin G. Nørsett, Eirik Sundby, Sondre Nervik, Bård Helge Hoff, Jin Han, Svein Jacob Kaspersen
المصدر: European Journal of Medicinal Chemistry. 119:278-299
مصطلحات موضوعية: Protein Conformation, Stereochemistry, Stereoisomerism, 01 natural sciences, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Protein structure, Drug Discovery, medicine, Structure–activity relationship, Moiety, Amines, Protein Kinase Inhibitors, EGFR inhibitors, Pharmacology, 010405 organic chemistry, Kinase, Aryl, Organic Chemistry, General Medicine, 0104 chemical sciences, ErbB Receptors, Molecular Docking Simulation, Kinetics, Pyrimidines, chemistry, 030220 oncology & carcinogenesis, Erlotinib, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9efcd7efaa05464b58400b33c79f8fb6Test
https://doi.org/10.1016/j.ejmech.2016.04.054Test -
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المؤلفون: Kristin G. Nørsett, Ann Christin Reiersølmoen, Bård Helge Hoff, Eirik Sundby, Sarah Eckelt, Thomas Ihle Aarhus
المصدر: Bioorganic & Medicinal Chemistry Letters
مصطلحات موضوعية: Substituent, Cancer therapy, Molecular Dynamics Simulation, medicine.disease_cause, 01 natural sciences, Biochemistry, Cross-reactivity, Cell Line, chemistry.chemical_compound, Erlotinib Hydrochloride, Mice, Drug Discovery, medicine, Animals, Pyrroles, Epidermal growth factor receptor, Molecular Biology, Protein Kinase Inhibitors, EGFR inhibitors, Cell Proliferation, Binding Sites, biology, 010405 organic chemistry, Kinase, Aryl, Organic Chemistry, 0104 chemical sciences, ErbB Receptors, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Pyrimidines, chemistry, Cancer research, biology.protein, Erlotinib, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::92d45ff199e21667716bc31044df08faTest
http://hdl.handle.net/11250/2635253Test -
4
المؤلفون: F. Bysting, Bård Helge Hoff, Steffen Bugge, Eirik Sundby
المصدر: 18569-18577
RSC Advancesمصطلحات موضوعية: 010405 organic chemistry, Stereochemistry, Chemistry, General Chemical Engineering, Egfr inhibition, chemistry.chemical_element, General Chemistry, Highly selective, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, Catalysis, Solvent, 03 medical and health sciences, 0302 clinical medicine, 030220 oncology & carcinogenesis, Heck reaction, Isomerization, Palladium, EGFR inhibitors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4d473c3d1194cfd47119afacadfae6a8Test
https://hdl.handle.net/11250/2444444Test -
5
المؤلفون: Bård Helge Hoff, Ingri Ullestad Moen, Kent-Ove Kragseth Sylte, Steffen Bugge, Eirik Sundby
المصدر: European journal of medicinal chemistry. 94
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Models, Molecular, Chemistry, Stereochemistry, Organic Chemistry, Stereoisomerism, General Medicine, Combinatorial chemistry, ErbB Receptors, Structure-Activity Relationship, Activity measurements, Enzyme, Gefitinib, Pyrimidines, Binding efficiency, Drug Discovery, Retrospective analysis, medicine, Moiety, Protein Kinase Inhibitors, EGFR inhibitors, Epidermal growth factor receptor tyrosine kinase, medicine.drug, Retrospective Studies
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2da781867991cd3c09d954f90888555dTest
https://pubmed.ncbi.nlm.nih.gov/25768701Test -
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المؤلفون: Eirik Sundby, Synne Larsen, Unni Nonstad, Bård Helge Hoff, Geir Bjørkøy, Steffen Bugge, Svein Jacob Kaspersen
المصدر: European journal of medicinal chemistry. 75
مصطلحات موضوعية: Models, Molecular, Benzylamines, Pyrimidine, Stereochemistry, Mutant, Antineoplastic Agents, chemistry.chemical_compound, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Potency, Humans, IC50, Protein Kinase Inhibitors, EGFR inhibitors, Pharmacology, Chemistry, Organic Chemistry, General Medicine, In vitro, ErbB Receptors, Pyrimidines, Biochemistry, Cell culture, Erlotinib, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::076e87fc8ead7a1f45de3cc07f6b5422Test
https://pubmed.ncbi.nlm.nih.gov/24556149Test