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المؤلفون: Annette N. Chiang, Disha Joshi, Peter Wipf, Mads B. Larsen, Raymond A. Frizzell, Jeffrey L. Brodsky, Clare Hill, Jennifer L. Goeckeler-Fried, Rajiah Aldrin Denny, Eric J. Sorscher
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Protein Folding, Ubiquitin-activating enzyme, Clinical Biochemistry, Pharmaceutical Science, Cystic Fibrosis Transmembrane Conductance Regulator, Endoplasmic-reticulum-associated protein degradation, Protein degradation, Biochemistry, Benzoates, Article, Structure-Activity Relationship, Ubiquitin, Drug Discovery, Humans, Furans, Molecular Biology, Integral membrane protein, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Ubiquitination, Cystic fibrosis transmembrane conductance regulator, Protein ubiquitination, Cell biology, biology.protein, Molecular Medicine, Pyrazoles, Protein folding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9acacfc386f55a26c851fd71b6ecd340Test
https://pubmed.ncbi.nlm.nih.gov/34246753Test -
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المؤلفون: Carly S. Mazzone, Antonio Dominguez-Meijide, Jeffrey L. Brodsky, Mary Liang, Tiago F. Outeiro, Annette N. Chiang, David Newhouse, Peter Wipf, Nathan M. Kendsersky, Megan E. Yates, Patrick G. Needham, Caterina Masaracchia, Alexandra Manos-Turvey, Jennifer L. Goeckeler-Fried
المصدر: Bioorganic & Medicinal Chemistry. 27:79-91
مصطلحات موضوعية: Protein Folding, Clinical Biochemistry, Mutant, Cystic Fibrosis Transmembrane Conductance Regulator, Enzyme Activators, Pharmaceutical Science, Pyrimidinones, Saccharomyces cerevisiae, Protein aggregation, 01 natural sciences, Biochemistry, Article, Structure-Activity Relationship, Cell Line, Tumor, Cellular stress response, Drug Discovery, Humans, HSP70 Heat-Shock Proteins, Molecular Biology, Adenosine Triphosphatases, Molecular Structure, biology, 010405 organic chemistry, Activator (genetics), Chemistry, Organic Chemistry, HEK 293 cells, Esters, Cystic fibrosis transmembrane conductance regulator, 3. Good health, 0104 chemical sciences, Hsp70, Cell biology, 010404 medicinal & biomolecular chemistry, HEK293 Cells, Proteostasis, alpha-Synuclein, biology.protein, Molecular Medicine, Protein Multimerization
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c6e5c63d4a71c5b638613d360a3ee103Test
https://doi.org/10.1016/j.bmc.2018.11.011Test