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1دورية أكاديمية
المؤلفون: Silva, Daniel, Mendes, Eduarda, Summers, Eleanor J., Neca, Ana, Jacinto, Ana C., Reis, Telma, Agostinho, Paula, Bolea, Irene, Jimeno, M. Luisa, Mateus, M. Luisa, Oliveira-Campos, Ana M. F., Unzeta, Mercedes, Marco-Contelles, José, Majekova, Magdalena, Ramsay, Rona R., Carreiras, M. Carmo
المصدر: Silva , D , Mendes , E , Summers , E J , Neca , A , Jacinto , A C , Reis , T , Agostinho , P , Bolea , I , Jimeno , M L , Mateus , M L , Oliveira-Campos , A M F , Unzeta , M , Marco-Contelles , J , Majekova , M , Ramsay , R R & Carreiras , M C 2019 , ' Synthesis, biological evaluation, and molecular modeling of nitrile-containing compounds : exploring multiple activities as anti-Alzheimer agents ' , Drug Development Research , vol. Early View ....
مصطلحات موضوعية: Nitrile-containing compounds, Alzheimer's disease, MAO inhibitors, Cholinesterase inhibitors, Aβ1-42 disaggregating agents, In silico study
وصف الملف: application/pdf
العلاقة: https://research-portal.st-andrews.ac.uk/en/researchoutput/synthesis-biological-evaluation-and-molecular-modeling-of-nitrilecontaining-compoundsTest(a2bf3daa-a7f7-4a16-9729-e4ef09695e3a).html
الإتاحة: https://doi.org/10.1002/ddr.21594Test
https://research-portal.st-andrews.ac.uk/en/researchoutput/synthesis-biological-evaluation-and-molecular-modeling-of-nitrilecontaining-compoundsTest(a2bf3daa-a7f7-4a16-9729-e4ef09695e3a).html
https://research-repository.st-andrews.ac.uk/bitstream/10023/20525/1/Silva2019acceptedDDR.pdfTest -
2دورية أكاديمية
المؤلفون: Silva, Daniel, Mendes, Eduarda, Summers, Eleanor J., Neca, Ana, Jacinto, Ana C., Reis, Telma, Agostinho, Paula, Bolea, Irene, Jimeno, M. Luisa, Mateus, M. Luisa, Oliveira-Campos, Ana M. F., Unzeta, Mercedes, Marco-Contelles, José, Majekova, Magdalena, Ramsay, Rona R., Carreiras, M. Carmo
المساهمون: University of St Andrews. Biomedical Sciences Research Complex, University of St Andrews. School of Biology
مصطلحات موضوعية: Nitrile-containing compounds, Alzheimer's disease, MAO inhibitors, Cholinesterase inhibitors, Aβ1-42 disaggregating agents, In silico study, RM Therapeutics. Pharmacology, NDAS, RM
وصف الملف: application/pdf
العلاقة: Drug Development Research; 260556740; a2bf3daa-a7f7-4a16-9729-e4ef09695e3a; 85071395167; 000484141800001; Silva , D , Mendes , E , Summers , E J , Neca , A , Jacinto , A C , Reis , T , Agostinho , P , Bolea , I , Jimeno , M L , Mateus , M L , Oliveira-Campos , A M F , Unzeta , M , Marco-Contelles , J , Majekova , M , Ramsay , R R & Carreiras , M C 2019 , ' Synthesis, biological evaluation, and molecular modeling of nitrile-containing compounds : exploring multiple activities as anti-Alzheimer agents ' , Drug Development Research , vol. Early View , DDR-19-0121.R1 . https://doi.org/10.1002/ddr.21594Test; ORCID: /0000-0003-1535-4904/work/61369941; https://hdl.handle.net/10023/20525Test
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المؤلفون: Dgachi, Youssef, Martin, H., Martin, Hélène, Malek, R, Jun, D., Janockova, Jana, Sepsova, Vendula, Soukup, Ondrej, Iriepa, Isabel, Moraleda, Ignacio, Maalej, Enma, Carreiras, M. Carmo, Refouvelet, B., Chabchoub, Fakher, Marco-Contelles, José, Ismaili, Lhassane
المساهمون: Ministerio de Economía, Industria y Competitividad (España), European Commission
المصدر: Digital.CSIC. Repositorio Institucional del CSIC
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Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 163-170 (2019)
Journal of Enzyme Inhibition and Medicinal Chemistryمصطلحات موضوعية: Models, Molecular, 0301 basic medicine, medicine.drug_class, Short Communication, tacrine, Pharmacology, 01 natural sciences, Neuroprotection, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Kojic acid, Drug Discovery, medicine, alzheimer disease, Humans, Structure–activity relationship, IC50, Dose-Response Relationship, Drug, Molecular Structure, kojic acid, 010405 organic chemistry, business.industry, lcsh:RM1-950, General Medicine, multitarget small molecules, medicine.disease, Acetylcholinesterase, Multitarget small molecules, 0104 chemical sciences, Neuroprotective Agents, 030104 developmental biology, lcsh:Therapeutics. Pharmacology, chemistry, Acetylcholinesterase inhibitor, Drug Design, Tacrine, Cholinesterase Inhibitors, Alzheimer's disease, Alzheimer disease, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d0f01cc1d23157fa3d81d0133cfe5701Test
http://hdl.handle.net/10261/175021Test -
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المؤلفون: Ignacio Moraleda, Rafael León, Manuela García, M. Carmo Carreiras, Vincenza Andrisano, Carla Martins, Cristóbal de los Ríos, Enrique Gálvez, José Marco-Contelles, Abdelouhaid Samadi, Javier Egea, Mourad Chioua, Manuela Bartolini, Isabel Iriepa
المساهمون: Martins C., Carreiras M. C., Leon R., de Los Rios C., Bartolini M., Andrisano V., Iriepa I., Moraleda I., Galvez E., Garcia M., Egea J., Samadi A., Chioua M., Marco-Contelles J.
المصدر: European journal of medicinal chemistry. 46(12)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, ACHE/BUCHE INHIBITORS, chemistry.chemical_compound, Alzheimer Disease, Drug Discovery, medicine, Humans, Butyrylcholinesterase, Cholinesterase, Pharmacology, chemistry.chemical_classification, NEUROPROTECTION, biology, ALZHEIMER’S DISEASE, Organic Chemistry, Active site, General Medicine, Acetylcholinesterase, Enzyme, chemistry, Docking (molecular), Tacrine, biology.protein, Aminoquinolines, Amine gas treating, Cholinesterase Inhibitors, medicine.drug
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7af52204ef77d6ab74f638461fa32ff0Test
https://pubmed.ncbi.nlm.nih.gov/22000936Test