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المؤلفون: Christelle David, Nele Vandervoort, Damien Fleury, Denis Annoot, Laëtitia Cherel, Willem Jan Hengeveld, Thierry Christophe, Sameh H. Soror, Agnès Marie Joncour, Christopher Gaëtan Housseman, Alain Monjardet, R Galien, Patrick Mollat, Reginald Brys, Veronique Roncoroni, Luce Lepissier, Natacha Bienvenu, Lionel Vercheval, Alexandre Wohlkonig, Christophe Peixoto, Jörg Heiermann, Katja Conrath, Mia Jans, Sandrine Le Tallec, Bertrand Heckmann, Robert Touitou, Nicolas Desroy, Jan Steyaert, Virginie Labeguere, Gregor Pilzak, Ellen van der Aar, Xavier Marie Bock, Nicolas Triballeau, Emanuelle Wakselman
المساهمون: Department of Bio-engineering Sciences, Structural Biology Brussels
المصدر: Journal of Medicinal Chemistry. 60:7371-7392
مصطلحات موضوعية: Male, 0301 basic medicine, Phosphodiesterase Inhibitors, Pyridines, Stereochemistry, Inflammation, 01 natural sciences, Cocrystal, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, Lysophosphatidic acid, Hydrolase, medicine, Animals, Humans, Structure–activity relationship, chemistry.chemical_classification, Phosphoric Diester Hydrolases, 010405 organic chemistry, Chemistry, Drug discovery, Imidazoles, Lysophosphatidylcholines, Rats, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, Enzyme, Biochemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Lysophospholipids, Autotaxin, medicine.symptom
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c1bab957aedfbab6da364d90d0e33f16Test
https://doi.org/10.1021/acs.jmedchem.7b00647Test -
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المؤلفون: John G. Logan, Silvia Marino, Patrick Mollat, Ryan T. Bishop, Aymen I. Idris
مصطلحات موضوعية: 0301 basic medicine, musculoskeletal diseases, Cancer Research, Time Factors, Osteolysis, β-Catenin, Osteoclasts, Apoptosis, Bone Neoplasms, Breast Neoplasms, 03 medical and health sciences, chemistry.chemical_compound, Breast cancer, Osteogenesis, Osteoclast, medicine, Animals, Humans, Parthenolide, Oncology & Carcinogenesis, Bone, beta Catenin, Cell Proliferation, Mice, Inbred BALB C, Osteoblasts, Dose-Response Relationship, Drug, Chemistry, NF-kappa B, Bone metastasis, Cell Differentiation, Osteoblast, medicine.disease, Mice, Inbred C57BL, 030104 developmental biology, medicine.anatomical_structure, Oncology, Catenin, Immunology, MCF-7 Cells, Cancer research, Female, Sesquiterpenes, 1112 Oncology And Carcinogenesis, Signal Transduction, NFκB
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ce26b1fead8a0082887cd6b411262742Test
http://hdl.handle.net/10044/1/53123Test -
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المؤلفون: Nele Vandervoort, Xavier Marie Bock, Patrick Mollat, Jovica Ralić, Alain Monjardet, Nicolas Triballeau, Thierry Christophe, Ellen van der Aar, Marieke Lamers, Boska Hrvacic, Nicolas Desroy, Bertrand Heckmann, Line Oste, Emilie Rondet, Virginie Labeguere, Roland Blanque, Veronique Roncoroni, Christopher Gaëtan Housseman, Sandrine Le Tallec, Natacha Bienvenu, C. Cottereaux, M. Auberval, Reginald Brys, Laëtitia Cherel, Emanuelle Wakselman, Picolet Olivier Laurent, Jean-Marie Grassot, Agnès Marie Joncour, Christophe Peixoto, Denis Annoot
مصطلحات موضوعية: 0301 basic medicine, hERG, Pharmacology, autoaxin inhibitor, LPA, pulmonary fibrosis, bleomycin-induced model in mice, 03 medical and health sciences, Idiopathic pulmonary fibrosis, chemistry.chemical_compound, Mice, 0302 clinical medicine, In vivo, Drug Discovery, Pulmonary fibrosis, medicine, Animals, Humans, Thiazole, Mice, Knockout, Lung, medicine.diagnostic_test, biology, Chemistry, Phosphoric Diester Hydrolases, Imidazoles, medicine.disease, Idiopathic Pulmonary Fibrosis, Rats, 030104 developmental biology, Bronchoalveolar lavage, medicine.anatomical_structure, Pyrimidines, 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), Autotaxin
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04c6f6e80895c7ca93e77aad9243c383Test
https://www.bib.irb.hr/981523Test -
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المؤلفون: Reginald Brys, Emanuelle Wakselman, Lionel Vercheval, Christelle David, Nele Vandervoort, Laëtitia Cherel, Christopher Gaëtan Housseman, Luce Lepissier, Natacha Bienvenu, Mia Jans, Alain Monjardet, Agnès Marie Joncour, Nicolas Desroy, Gregor Pilzak, Willem Jan Hengeveld, Sandrine Le Tallec, Ellen van der Aar, Bertrand Heckmann, Nicolas Triballeau, Jan Steyaert, Patrick Mollat, Veronique Roncoroni, Virginie Labeguere, Sameh H. Soror, Damien Fleury, Thierry Christophe, Christophe Peixoto, Xavier Marie Bock, Denis Annoot, Jörg Heiermann, Katja Conrath, R Galien, Robert Touitou, Alexandre Wohlkonig
المصدر: Journal of Medicinal Chemistry. 61:4270-4270
مصطلحات موضوعية: chemistry.chemical_compound, Series (mathematics), chemistry, Stereochemistry, Drug Discovery, Pyridine, Molecular Medicine, Structure–activity relationship, Autotaxin
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::93dee812f5866eca6cabf47d605a46ceTest
https://doi.org/10.1021/acs.jmedchem.8b00579Test -
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المؤلفون: Paulette Bichet, Patrick Mollat, Edoardo Sarubbi, Cécile Capdevila
المصدر: Protein Expression and Purification. 19:197-201
مصطلحات موضوعية: Insecta, Recombinant Fusion Proteins, Sf9, Plasma protein binding, Biology, Chromatography, Affinity, Mass Spectrometry, Cell Line, chemistry.chemical_compound, Affinity chromatography, Animals, Polyacrylamide gel electrophoresis, Chromatography, High Pressure Liquid, Glutathione Transferase, fungi, Glutathione, Molecular biology, Fusion protein, Glutathione S-transferase, chemistry, Biochemistry, biology.protein, Electrophoresis, Polyacrylamide Gel, Baculoviridae, Glutathione binding, Protein Binding, Biotechnology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::214598e530c97184b05855ce1216fa09Test
https://doi.org/10.1006/prep.2000.1239Test -
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المؤلفون: Francois Nique, Denis Guédin, Nicolas Triballeau, Eric Duval, Jean-Michel Lemoullec, Denis Annoot, Catherine Robin-Jagerschmidt, Maxime Thauvin, Jean-Michel Lefrancois, Thierry Prangé, Laurence Michoux, Philippe Clément-Lacroix, Damien Fleury, Pierre Deprez, Patrick Mollat, Séverine Hebbe, Dominique Minet, Christophe Peixoto
المصدر: Journal of medicinal chemistry. 55(19)
مصطلحات موضوعية: Male, Models, Molecular, Transcriptional Activation, medicine.medical_specialty, Antiandrogens, Hydantoin, Peptide, Pharmacology, Crystallography, X-Ray, Binding, Competitive, Bone and Bones, Transactivation, chemistry.chemical_compound, Structure-Activity Relationship, Anabolic Agents, Internal medicine, Drug Discovery, medicine, Androgen Receptor Antagonists, Potency, Animals, Humans, Muscle, Skeletal, chemistry.chemical_classification, Hydantoins, Prostate, Stereoisomerism, In vitro, Rats, Androgen receptor, Drug Partial Agonism, Endocrinology, Selective androgen receptor modulator, chemistry, Receptors, Androgen, Androgens, Molecular Medicine, Orchiectomy, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ac608008905445d4f9b1a1f2414f5434Test
https://pubmed.ncbi.nlm.nih.gov/22897611Test -
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المؤلفون: Rony Nehmé, Robert Bittman, Hélène Faure, Martial Ruat, Michel Bidet, Marine Ciantar, Lionel Bretillon, Patrick Mollat, Isabelle Mus-Veteau, Olivier Joubert, Benoît Lacombe
المساهمون: Institute of Developmental Biology and Cancer (IBDC), Université Nice Sophia Antipolis (... - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Centre National de la Recherche Scientifique (CNRS)-Université Côte d'Azur (UCA), Université Henri Poincaré - Nancy 1 (UHP), Laboratory of Molecular Biology, Medical Research Council, Galapagos SASU, Centre des Sciences du Goût et de l'Alimentation [Dijon] (CSGA), Institut National de la Recherche Agronomique (INRA)-Université de Bourgogne (UB)-AgroSup Dijon - Institut National Supérieur des Sciences Agronomiques, de l'Alimentation et de l'Environnement-Centre National de la Recherche Scientifique (CNRS), Neurobiologie & Développement (N&D), Centre National de la Recherche Scientifique (CNRS), Institut de Neurobiologie Alfred Fessard (INAF), Department of Chemistry and Biochemistry, State University of New York (SUNY), Université Côte d'Azur (UCA)-Université Côte d'Azur (UCA)-Centre National de la Recherche Scientifique (CNRS), Cibles thérapeutiques, formulation et expertise pré-clinique du médicament (CITHEFOR), Université de Lorraine (UL), Centre des Sciences du Goût et de l'Alimentation (CSGA), Institut National de la Recherche Agronomique (INRA)-Université de Bourgogne (UB)-Centre National de la Recherche Scientifique (CNRS), Institute of Developmental Biology and Cancer ( IBDC ), Centre National de la Recherche Scientifique ( CNRS ) -Université Nice Sophia Antipolis ( UNS ), Université Côte d'Azur ( UCA ) -Université Côte d'Azur ( UCA ), Université Henri Poincaré - Nancy 1 ( UHP ), Centre des Sciences du Goût et de l'Alimentation [Dijon] ( CSGA ), Institut National de la Recherche Agronomique ( INRA ) -Université de Bourgogne ( UB ) -AgroSup Dijon - Institut National Supérieur des Sciences Agronomiques, de l'Alimentation et de l'Environnement-Centre National de la Recherche Scientifique ( CNRS ), Neurobiologie & Développement ( N&D ), Centre National de la Recherche Scientifique ( CNRS ), Institut de Neurobiologie Alfred Fessard ( INAF ), The State University of New York ( SUNY ), ProdInra, Migration
المصدر: PLoS ONE
PLoS ONE, Public Library of Science, 2011, 6 (9), pp.e23834. ⟨10.1371/journal.pone.0023834⟩
European Biophysics Journal
8. EBSA European Biophysics Congress
8. EBSA European Biophysics Congress, Aug 2011, Budapest, Hungary. 1 p
HAL
PLoS ONE, Vol 6, Iss 9, p e23834 (2011)
PLoS ONE, Public Library of Science, 2011, 6 (9), pp.e23834. 〈10.1371/journal.pone.0023834〉
Plos One 9 (6), . (2011)مصطلحات موضوعية: cilium, lcsh:Medicine, yeast, Biochemistry, Receptors, G-Protein-Coupled, Transmembrane Transport Proteins, Mice, chemistry.chemical_compound, 0302 clinical medicine, Molecular Cell Biology, [SDV.IDA]Life Sciences [q-bio]/Food engineering, Membrane Receptor Signaling, Biomacromolecule-Ligand Interactions, Sonic hedgehog, lcsh:Science, ComputingMilieux_MISCELLANEOUS, 0303 health sciences, Multidisciplinary, Mechanisms of Signal Transduction, Veratrum Alkaloids, [SDV.IDA] Life Sciences [q-bio]/Food engineering, drosophila, Smoothened Receptor, Lipids, Hedgehog signaling pathway, Cell biology, Sterols, Alimentation et Nutrition, embryonic structures, cil, Membranes and Sorting, [SDV.NEU]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC], Signal transduction, vesicular trafficking, Signal Transduction, Research Article, primary cilium, Patched Receptors, Patched, signal-transduction, animal structures, Cyclopamine, [SPI.GPROC] Engineering Sciences [physics]/Chemical and Process Engineering, Biophysics, Receptors, Cell Surface, pathway activation, Saccharomyces cerevisiae, transduction du signal, Biology, 03 medical and health sciences, sonic hedgehog, lipid, Animals, Humans, Food and Nutrition, Hedgehog Proteins, [SPI.GPROC]Engineering Sciences [physics]/Chemical and Process Engineering, 030304 developmental biology, protein signals, Cell Membrane, lcsh:R, Proteins, cholesterol, Biological Transport, Transmembrane Proteins, sterol-sensing domain, chemistry, [ SDV.NEU ] Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC], NIH 3T3 Cells, cell trafficking, cells, biology.protein, lcsh:Q, Smoothened, 030217 neurology & neurosurgery
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5e0bcbd5426269bceb20005767504a4cTest
https://hal.archives-ouvertes.fr/hal-00637248Test -
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المؤلفون: Petra Simic, Maala Krishnan, Slobodan Vukicevic, Patrick Mollat, Euphemie Landao-Bassonga, Stuart H. Ralston, Aymen I. Idris
مصطلحات موضوعية: musculoskeletal diseases, medicine.medical_specialty, Cell Survival, Ovariectomy, Osteoporosis, Osteoclasts, IKK, TAK1, NFκB, osteoblast, osteoporosis, IκB kinase, Biochemistry, Bone resorption, Inhibitory Concentration 50, Mice, chemistry.chemical_compound, Osteoclast, Quinoxalines, Internal medicine, Bone cell, Genetics, medicine, Animals, Humans, Parthenolide, Bone Resorption, Enzyme Inhibitors, Molecular Biology, Cells, Cultured, Anti-Inflammatory Agents, Non-Steroidal, Imidazoles, Cell Differentiation, Osteoblast, medicine.disease, Triterpenes, I-kappa B Kinase, Cell biology, Enzyme Activation, Endocrinology, medicine.anatomical_structure, chemistry, Celastrol, Female, Pentacyclic Triterpenes, Sesquiterpenes, Signal Transduction, Biotechnology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cb841405b96f7ac3788a4c5d9fe76aa2Test
https://www.bib.irb.hr/552039Test -
9Identification of hydrogen sulfide releasing compounds as novel antiresorptive and antitumour agents
المؤلفون: Aymen I. Idris, Anna Sparatore, Stuart H. Ralston, J. Frantzias, Patrick Mollat, P. Del Soldato
المصدر: Bone. 48:S44
مصطلحات موضوعية: chemistry.chemical_compound, Histology, Physiology, Chemistry, Endocrinology, Diabetes and Metabolism, Hydrogen sulfide, Identification (biology), Combinatorial chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::12e1d599a8f5862d5728f43bfc7559a6Test
https://doi.org/10.1016/j.bone.2010.10.125Test