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المؤلفون: Yin-Ru Li, Yan-Bing Zhang, Yuan Liu, Xu Liu, Xiao-Jing Pang, Jian Song, Guang-Xi Yu, Sai-Yang Zhang, Wen-Bo Liu
المصدر: Molecules
Volume 26
Issue 13
Molecules, Vol 26, Iss 4047, p 4047 (2021)مصطلحات موضوعية: Stereochemistry, Pharmaceutical Science, Quantitative Structure-Activity Relationship, macromolecular substances, 01 natural sciences, Microtubules, Article, Analytical Chemistry, Tubulin binding, 03 medical and health sciences, chemistry.chemical_compound, QD241-441, Microtubule, Heterocyclic Compounds, Tubulin, Cell Line, Tumor, Drug Discovery, medicine, Colchicine, Humans, Physical and Theoretical Chemistry, colchicine binding site, Heterocyclic derivatives, 030304 developmental biology, Cell Proliferation, 0303 health sciences, N-containing heterocyclics, Binding Sites, biology, 010405 organic chemistry, Drug discovery, Organic Chemistry, Cancer, medicine.disease, Tubulin Modulators, 0104 chemical sciences, chemistry, Chemistry (miscellaneous), Cell culture, biology.protein, anti-proliferative activity, Molecular Medicine, vicinal diaryl, CA-4, Protein Binding
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::909eb39ab405236ab838402a6867341cTest
https://pubmed.ncbi.nlm.nih.gov/34279387Test -
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المؤلفون: Zahra Sadat Nazifi, Aref G Ghahsare, S. M. R. Nazifi
المصدر: Current organic synthesis. 16(8)
مصطلحات موضوعية: Xanthene, Cyclic compound, Biological Products, Molecular Structure, 010405 organic chemistry, Drug Compounding, Organic Chemistry, Anti-Inflammatory Agents, Antineoplastic Agents, 010402 general chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, chemistry.chemical_compound, Structure-Activity Relationship, chemistry, Anti-Infective Agents, Xanthenes, Alzheimer Disease, Drug Design, Animals, Humans, Hypoglycemic Agents, Heterocyclic derivatives
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d74d39e6087479e0c4e7b24d724ddb9dTest
https://pubmed.ncbi.nlm.nih.gov/31984917Test -
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المؤلفون: Su Huo, Penglong Wang, Xuehao Tian, Yuhao Gu, Jinchai Qi, Wen Li, Hongshan Chen, Ziqi Dai, Nana Han, Yu-Qin Yang, Feng Gao, Xiaojing Liu, Qianwen Wu, Haimin Lei, Tianxin Xie
المصدر: Molecules
Volume 25
Issue 4
Molecules, Vol 25, Iss 4, p 948 (2020)مصطلحات موضوعية: BA-nitrogen heterocyclic derivatives, Pharmaceutical Science, Antineoplastic Agents, Article, Analytical Chemistry, Flow cytometry, lcsh:QD241-441, HeLa, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, lcsh:Organic chemistry, betulinic acid, Neoplasms, Betulinic acid, Drug Discovery, medicine, Humans, Cytotoxic T cell, Physical and Theoretical Chemistry, Cytotoxicity, IC50, antitumor, 030304 developmental biology, 0303 health sciences, biology, medicine.diagnostic_test, Cytotoxins, flow cytometry, Organic Chemistry, Hep G2 Cells, biology.organism_classification, Triterpenes, In vitro, Hela, Biochemistry, chemistry, Chemistry (miscellaneous), Apoptosis, 030220 oncology & carcinogenesis, Molecular Medicine, Drug Screening Assays, Antitumor, Pentacyclic Triterpenes, HeLa Cells
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c12f57ef45dd776a937437792b273f91Test
https://doi.org/10.3390/molecules25040948Test -
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المؤلفون: Gianluigi Franci, Rosana Alvarez, A. R. de Lera, Lucia Altucci, J. G. Denis, Jose M. Aurrecoechea
المساهمون: Denis, Jg, Franci, G, Altucci, Lucia, Aurrecoechea, Jm, de Lera, Ár, Álvarez, R.
المصدر: Organic & Biomolecular Chemistry. 13:2800-2810
مصطلحات موضوعية: Indoles, biology, Chemistry, Stereochemistry, Organic Chemistry, epigenetic drugs, U937 Cells, Oxidative phosphorylation, Benzazepines, Biochemistry, Benzazepine, sirtuin, Structure-Activity Relationship, chemistry.chemical_compound, Sirtuin 1, Cyclization, Sirtuin, biology.protein, Humans, Physical and Theoretical Chemistry, Oxidation-Reduction, Heterocyclic derivatives, epigenetic
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::da88404d33bd4e42879376bbe50abf9aTest
https://doi.org/10.1039/c4ob02493aTest -
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المؤلفون: Anna E. Koziol, David Collu, Filippo Iuliano, Piotr Tomaszewski, Michał Jóźwiak, Daniel Szulczyk, Tadeusz Lis, Marta Struga
المصدر: Molecules : A Journal of Synthetic Chemistry and Natural Product Chemistry
Molecules; Volume 22; Issue 3; Pages: 409
Molecules, Vol 22, Iss 3, p 409 (2017)مصطلحات موضوعية: Models, Molecular, Pharmaceutical Science, Oxadiazole, biological activity, Microbial Sensitivity Tests, 010402 general chemistry, Ring (chemistry), Crystallography, X-Ray, 01 natural sciences, Article, Analytical Chemistry, X-ray crystal structure analysis, Cell Line, lcsh:QD241-441, chemistry.chemical_compound, Structure-Activity Relationship, 1,2,4-triazole, lcsh:Organic chemistry, Anti-Infective Agents, Drug Discovery, Thiadiazoles, 1,3,4-oxadiazole, Organic chemistry, Humans, Physical and Theoretical Chemistry, Candida albicans, Cytotoxicity, Heterocyclic derivatives, Cells, Cultured, 1,3,4-thiadiazole, Oxadiazoles, biology, Bacteria, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Fungi, Thiourea, 1,2,4-Triazole, thiourea, Triazoles, biology.organism_classification, In vitro, 0104 chemical sciences, chemistry, Chemistry (miscellaneous), HIV-1, Molecular Medicine
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::12f7b65a32faf0720e27b39f0a9d03caTest
http://europepmc.org/articles/PMC6155191Test -
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المؤلفون: Claudia Gargini, Sara Del Carlo, Clementina Manera, Ilaria Piano, Marco Macchia, Riccardo Ghidoni, Simone Bertini, Maria Digiacomo, Giuseppe Saccomanni, Giuseppe Matteo Campisi
المصدر: Molecules : A Journal of Synthetic Chemistry and Natural Product Chemistry
Molecules, Vol 22, Iss 7, p 1198 (2017)مصطلحات موضوعية: 0301 basic medicine, Magnetic Resonance Spectroscopy, Serine C-Palmitoyltransferase, Pharmaceutical Science, SPT, High-performance liquid chromatography, Analytical Chemistry, Substrate Specificity, HPLC, enzymatic assay, screening, serine palmitoyl transferase, Serine, lcsh:QD241-441, 03 medical and health sciences, chemistry.chemical_compound, lcsh:Organic chemistry, Myriocin, Drug Discovery, Transferase, Humans, Fluorometry, Physical and Theoretical Chemistry, Enzyme Inhibitors, Derivatization, Heterocyclic derivatives, Chromatography, High Pressure Liquid, Chromatography, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Communication, Organic Chemistry, Extraction (chemistry), Reproducibility of Results, 030104 developmental biology, HEK293 Cells, Chemistry (miscellaneous), Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c11799c59b6a3ffdc501fb7c08a6ac32Test
http://hdl.handle.net/11568/876789Test -
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المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry. 28:240-266
مصطلحات موضوعية: Pharmacology, Molecular Structure, Antitubercular Agents, Antineoplastic Agents, General Medicine, Antimicrobial, Ring (chemistry), Antimalarials, chemistry.chemical_compound, Anti-Infective Agents, Benzothiazole, chemistry, Drug Discovery, Humans, Organic chemistry, Benzothiazoles, Enzyme Inhibitors, Thiazole, Heterocyclic derivatives
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4c335708cb19e2b8390ed1af878a4c58Test
https://doi.org/10.3109/14756366.2012.720572Test -
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المؤلفون: Srikanth Yellamelli Valli Venkata, Naseer Ahmed Khan Mohammed, Kashi Reddy Methuku, Kamal Ahmed, Farheen Sultana
المصدر: Expert Opinion on Investigational Drugs. 21:619-635
مصطلحات موضوعية: Pharmacology, Molecular Structure, Bicyclic molecule, Antineoplastic Agents, General Medicine, chemistry.chemical_compound, Benzothiazole, chemistry, Biological profile, Neoplasms, Biological property, Animals, Humans, Moiety, Organic chemistry, Pharmacology (medical), Benzothiazoles, Pharmacophore, Heterocyclic derivatives, Conjugate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4353d34da8973488fceb1adfa5c49713Test
https://doi.org/10.1517/13543784.2012.676043Test -
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المؤلفون: Abeer A. Mohamed, Rafat M. Mohareb
المصدر: Molecules
Molecules, Vol 15, Iss 5, Pp 3602-3617 (2010)
Molecules; Volume 15; Issue 5; Pages: 3602-3617مصطلحات موضوعية: pyridine, Stereochemistry, Pyridines, Pharmaceutical Science, 1,3,4-triazine, Antineoplastic Agents, CNS cancer, Article, Analytical Chemistry, lcsh:QD241-441, Pyridazine, chemistry.chemical_compound, Structure-Activity Relationship, hydrazide-hydrazone, lcsh:Organic chemistry, Heterocyclic Compounds, Drug Discovery, Pyridine, Tumor Cells, Cultured, Structure–activity relationship, Humans, Physical and Theoretical Chemistry, Heterocyclic derivatives, pyridazine, antitumor, Antitumor activity, Chemistry, Triazines, Organic Chemistry, Acetophenones, Hydrazines, Chemistry (miscellaneous), Molecular Medicine, Non small cell, Drug Screening Assays, Antitumor, Acetophenone
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::732768f85e4ae3e3747c9be80c55cecbTest
http://europepmc.org/articles/PMC6263350Test -
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المؤلفون: Yoshio Hamada, Yoshiaki Kiso, Jeffrey-Tri Nguyen, Kenji Suzuki
المصدر: Bioorganicmedicinal chemistry. 21(21)
مصطلحات موضوعية: Quantitative structure–activity relationship, Stereochemistry, Isostere, Clinical Biochemistry, Pharmaceutical Science, Quantitative Structure-Activity Relationship, Ring (chemistry), Biochemistry, chemistry.chemical_compound, Heterocyclic Compounds, mental disorders, Drug Discovery, Thiadiazoles, Moiety, Aspartic Acid Endopeptidases, Humans, Tetrazole, Protease Inhibitors, Molecular Biology, Heterocyclic derivatives, Chemistry, Organic Chemistry, Substrate (chemistry), Hydrogen Bonding, Combinatorial chemistry, Recombinant Proteins, Benzamides, β secretase, Molecular Medicine, Amyloid Precursor Protein Secretases, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5b2ccdf7a426aa6ba2a62a4cf92d12ecTest
https://pubmed.ncbi.nlm.nih.gov/23993670Test