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1دورية أكاديمية
المؤلفون: Ritesh P. Bhole, Govinda O. Joshi, Harshad S. Kapare, Rupesh V. Chikhale, Somdatta Chaudhari
المصدر: Results in Chemistry, Vol 8, Iss , Pp 101615- (2024)
مصطلحات موضوعية: Covalent drugs, Targeted covalent inhibition (TCI), Disease-related proteins, Two-step inhibition process, Toxicity mitigation strategies, Chemistry, QD1-999
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2211715624003114Test; https://doaj.org/toc/2211-7156Test
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2دورية أكاديمية
المصدر: Results in Chemistry, Vol 6, Iss , Pp 101143- (2023)
مصطلحات موضوعية: Metastatic Castration Resistant prostate cancer, Enzalutamide, Nonsteroidal antiandrogens, AR, F786L mutation, Chemistry, QD1-999
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S221171562300382XTest; https://doaj.org/toc/2211-7156Test
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3دورية أكاديميةFacile and efficient synthesis of benzoxazole derivatives using novel catalytic activity of PEG-SO3H
المؤلفون: Rupesh V. Chikhale, Amit M. Pant, Sunil S. Menghani, Pankaj G. Wadibhasme, Pramod B. Khedekar
المصدر: Arabian Journal of Chemistry, Vol 10, Iss 5, Pp 715-725 (2017)
مصطلحات موضوعية: Poly (ethylene glycol)-bound sulfonic acid (PEG-SO3H), 2-Aminobenzoxazole, Benzoxazole derivatives, Chemistry, QD1-999
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S187853521400135XTest; https://doaj.org/toc/1878-5352Test
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المؤلفون: S. Jadhav, R.P. Bhole, C.G. Bonde, Rupesh V. Chikhale, Y. Shinde
المصدر: Қарағанды университетінің хабаршысы. Химия сериясы, Vol 103, Iss 3, Pp 21-26 (2021)
مصطلحات موضوعية: Drug, Vitamin, vitamin d3, synthesis, Chemistry, molecular modeling, media_common.quotation_subject, 5-fluorouracil acetic acid, General Chemistry, molecular docking, Pharmacology, chemistry.chemical_compound, vitamin-drug conjugate, QD1-999, media_common, Conjugate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::65b1b291bea631af94d1626ef59532deTest
https://chemistry -vestnik.ksu.kz/apart/2021-103-3/02.pdf -
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المؤلفون: Pramod B. Khedekar, Rupesh V. Chikhale, Mohit D. Umare
المصدر: ChemMedChem. 16:3136-3148
مصطلحات موضوعية: Tuberculosis, medicine.drug_class, Antibiotics, Antitubercular Agents, Microbial Sensitivity Tests, Biology, Biochemistry, Bacterial cell structure, Mycolic acid, Microbiology, Bacterial Proteins, Drug Discovery, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, High potential, Pharmacology, chemistry.chemical_classification, Molecular Structure, Organic Chemistry, Membrane Transport Proteins, Transporter, Mycobacterium tuberculosis, medicine.disease, chemistry, Drug development, Membrane protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6faf1f5274eb492c1e015d93d449025eTest
https://doi.org/10.1002/cmdc.202100359Test -
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المؤلفون: Siham A. Alissa, Hassna Mohammed Alhajri, Shuchi Nagar, Tahani Mazyad Almutairi, Rupesh V. Chikhale, Surajit Ghosh, Hans Raj Bhat, Ataul Islam, Fatmah A.S. Alasmary, Anshul Shakya
المصدر: Molecular Diversity
مصطلحات موضوعية: Camostat, Virtual screening, medicine.medical_treatment, 030303 biophysics, Molecular Dynamics Simulation, medicine.disease_cause, urologic and male genital diseases, Catalysis, Inorganic Chemistry, Hydrophobic effect, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, Morus alba Linn, medicine, Serine, Humans, Protease Inhibitors, Physical and Theoretical Chemistry, Molecular Biology, TMPRSS2, 030304 developmental biology, Coronavirus, chemistry.chemical_classification, 0303 health sciences, Protease, Chemistry, SARS-CoV-2, Organic Chemistry, General Medicine, Virus Internalization, Transmembrane Protease Serine 2, Transmembrane protein, Amino acid, COVID-19 Drug Treatment, Molecular Docking Simulation, Biochemistry, Molecular docking, Original Article, Morus, Information Systems
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4b424b8446533b2a50245d81fa96e292Test
http://europepmc.org/articles/PMC8009078Test -
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المؤلفون: Manish M. Wanjari, Rupali S. Prasad, Rajesh B. Patil, Suhas R. Dhaswadikar, Saurabh K. Sinha, Nilambari S. Gurav, Rupesh V. Chikhale, Satyendra K. Prasad, Shailendra S. Gurav, Anshul Shakya
المصدر: Journal of Biomolecular Structure & Dynamics
Journal of Biomolecular Structure and Dynamicsمصطلحات موضوعية: 0303 health sciences, Indian Ayurveda, Coronavirus disease 2019 (COVID-19), Binding free energy, biology, Chemistry, Stereochemistry, In silico, Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2), Shatavari, Molecular docking, nCov-2019, 030303 biophysics, Endoribonuclease, General Medicine, biology.organism_classification, 03 medical and health sciences, Pandemic disease, Docking (molecular), Structural Biology, Asparagus racemosus, Antiviral, Molecular Biology, Binding affinities, Research Article
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e988f509ad066a969b7997b222adf7e6Test
http://europepmc.org/articles/PMC7335809Test -
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المؤلفون: Saurabh K. Sinha, Rupesh V. Chikhale, Rajesh B. Patil, Muniappan Ayyanar, Shailendra S. Gurav, Manish M. Wanjari, Satyendra K. Prasad, Pukar Khanal, Nilambari S. Gurav
المصدر: Phytomedicine Plus, Vol 1, Iss 3, Pp 100095-(2021)
Phytomedicine Plusمصطلحات موضوعية: COVID19, medicine.medical_treatment, Biology, Pharmacology, Article, chemistry.chemical_compound, Other systems of medicine, Myricetin, Molecular Dynamics, medicine, Potency, Amlaki, Protease, Pandemic, Myricetin, Chlorogenic acid, medicine.disease, Quercitrin, chemistry, Docking (molecular), Phyllanthus emblica, Emblica officinalis, Signal transduction, Cytokine storm, Ayurveda, RZ201-999
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9480cab318ac55a742948949bd5ec9fbTest
http://www.sciencedirect.com/science/article/pii/S2667031321000774Test -
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المصدر: Bioorganic chemistry. 115
مصطلحات موضوعية: Enoyl-acyl carrier protein reductase, Antitubercular Agents, Microbial Sensitivity Tests, Reductase, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Structure–activity relationship, Humans, Inhibins, Molecular Biology, Fatty acid synthesis, chemistry.chemical_classification, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Drug discovery, INHA, Organic Chemistry, Mycobacterium tuberculosis, Acyl carrier protein, Enzyme, biology.protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e7e398c0a0f3b48b9d086508aa0c6b61Test
https://pubmed.ncbi.nlm.nih.gov/34392175Test -
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المؤلفون: Tahani Mazyad Almutairi, Chandrakant G. Bonde, Ritesh P. Bhole, Ravindra D. Wavhale, Fatmah Ali Asmary, Rupesh V. Chikhale, Hassna Mohammed Alhajri
المصدر: Heliyon, Vol 7, Iss 3, Pp e06227-(2021)
Heliyonمصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.drug_class, 03 medical and health sciences, chemistry.chemical_compound, Prostate cancer, 0302 clinical medicine, Castration Resistance, Binding energy calculations, LNCaP, medicine, Enzalutamide, lcsh:Social sciences (General), lcsh:Science (General), IC50, Multidisciplinary, Trifluoromethyl, Chemistry, Molecular dynamics simulations, Imidazolidinone derivatives, medicine.disease, Hybrid molecules, Androgen receptor, 030104 developmental biology, Molecular docking, Cancer research, lcsh:H1-99, 030217 neurology & neurosurgery, Research Article, lcsh:Q1-390
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62d6205eea10c7bce1e5f175062c6266Test
https://ueaeprints.uea.ac.uk/id/eprint/79458Test/