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1
المؤلفون: Janine Holze, Dina Manetti, Christian Tränkle, Klaus Mohr, Elisabetta Teodori, Maria Vittoria Martino, Cristina Bellucci, Maria Novella Romanelli, Giulio Vistoli, Jessica Welzel, Silvia Dei, Angelica Mazzolari, Marta Nesi, Ulrike Bartz, Rosanna Matucci
المصدر: European journal of pharmacology. 883
مصطلحات موضوعية: 0301 basic medicine, Carbachol, Allosteric regulation, CHO Cells, Muscarinic Antagonists, Muscarinic Agonists, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Cricetulus, Muscarinic acetylcholine receptor, medicine, Cyclic AMP, Animals, Humans, Phosphorylation, Receptor, Extracellular Signal-Regulated MAP Kinases, Pharmacology, Molecular Structure, Chemistry, Muscarinic antagonist, Receptors, Muscarinic, Molecular Docking Simulation, Kinetics, 030104 developmental biology, Docking (molecular), Guanosine 5'-O-(3-Thiotriphosphate), Biophysics, Cholinergic, Dimerization, 030217 neurology & neurosurgery, medicine.drug, Protein Binding, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b88ca14a4fbf7a1acd767dca1e4963fcTest
https://pubmed.ncbi.nlm.nih.gov/32534072Test -
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المؤلفون: Hongwei Li, Philipp Risel, Shoji Maeda, Harald Hübner, Brian K. Kobilka, Jonas Kaindl, Changwen Jin, Xiaogang Niu, Yunfei Hu, Peter Gmeiner, Jun Xu
المصدر: Molecular cell. 75(1)
مصطلحات موضوعية: Protein Conformation, alpha-Helical, Magnetic Resonance Spectroscopy, Pyridines, Allosteric regulation, Genetic Vectors, Gene Expression, Biology, Molecular Dynamics Simulation, Spodoptera, Ligands, 03 medical and health sciences, 0302 clinical medicine, Muscarinic acetylcholine receptor, Thiadiazoles, Arrestin, Sf9 Cells, Animals, Humans, Protein Interaction Domains and Motifs, Cloning, Molecular, Receptor, Molecular Biology, 030304 developmental biology, G protein-coupled receptor, 0303 health sciences, Receptor, Muscarinic M2, Binding Sites, Pilocarpine, Cell Biology, Nuclear magnetic resonance spectroscopy, Isoxazoles, Ligand (biochemistry), Transmembrane protein, Acetylcholine, Recombinant Proteins, Quaternary Ammonium Compounds, Kinetics, Biophysics, Thermodynamics, Carbachol, Protein Conformation, beta-Strand, Baculoviridae, 030217 neurology & neurosurgery, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::01fc3cac70fdf8f2cac7dce55b1d8dd0Test
https://pubmed.ncbi.nlm.nih.gov/31103421Test -
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المؤلفون: Deborah L. Smith, Sarah J. Neal, Lei Zhang, Jeremy R. Edgerton, Jennifer E. Davoren, Sarah Grimwood, John T. Lazzaro, Chewah Lee
المصدر: Molecular Pharmacology. 90:177-187
مصطلحات موضوعية: Male, 0301 basic medicine, Carbachol, Allosteric modulator, Pyridines, Stereochemistry, Allosteric regulation, CHO Cells, Isoindoles, Hippocampus, Rats, Sprague-Dawley, Radioligand Assay, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Allosteric Regulation, Cricetinae, Muscarinic acetylcholine receptor, medicine, Radioligand, Animals, Humans, Fluorometry, Pharmacology, Membranes, Chemistry, Ligand binding assay, Receptor, Muscarinic M1, N-Methylscopolamine, Acetylcholine, Electrophysiological Phenomena, Kinetics, HEK293 Cells, 030104 developmental biology, Positron-Emission Tomography, Autoradiography, Molecular Medicine, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59a4cbb153c3abcd01cb4427f9543370Test
https://doi.org/10.1124/mol.116.104737Test -
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المؤلفون: Gergő Gulyás, J. Tóth, László Hunyady, Péter Várnai, Gerald R.V. Hammond, Dániel J. Tóth, Tamas Balla, András Balla
المصدر: Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids. 1861:177-187
مصطلحات موضوعية: Phosphatidylinositol 4,5-Diphosphate, 0301 basic medicine, Lipolysis, Recombinant Fusion Proteins, Biosensing Techniques, Inositol 1,4,5-Trisphosphate, Muscarinic Agonists, Biology, Transfection, Article, 03 medical and health sciences, chemistry.chemical_compound, Phosphatidylinositol Phosphates, Chlorocebus aethiops, Fluorescence Resonance Energy Transfer, Animals, Humans, Inositol, Protein kinase A, Molecular Biology, Protein Kinase C, Protein kinase C, G protein-coupled receptor, Feedback, Physiological, Receptor, Muscarinic M3, Epidermal Growth Factor, Phospholipase C, Hydrolysis, Muscarinic acetylcholine receptor M3, Lipid metabolism, Cell Biology, Receptors, Muscarinic, Up-Regulation, Cell biology, Enzyme Activation, ErbB Receptors, Kinetics, HEK293 Cells, 030104 developmental biology, chemistry, Type C Phospholipases, COS Cells, Carbachol, Phosphatidylinositol 3-Kinase, Signal transduction, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dbee06da5cb4310f631bbb9f90b7802bTest
https://doi.org/10.1016/j.bbalip.2015.12.005Test -
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المؤلفون: Norihiro Yoshida, Eri Jojima, Hiroyuki Saito, Tatsuya Haga
المصدر: Biomedical Research. 35:185-192
مصطلحات موضوعية: Dynamins, Time Factors, G-Protein-Coupled Receptor Kinase 2, media_common.quotation_subject, education, Gene Expression, Plasma protein binding, General Biochemistry, Genetics and Molecular Biology, Muscarinic acetylcholine receptor, Humans, Protein Interaction Domains and Motifs, Receptor, Internalization, Cells, Cultured, media_common, Dynamin, Receptor, Muscarinic M2, Receptor, Muscarinic M4, Chemistry, HEK 293 cells, Muscarinic acetylcholine receptor M2, General Medicine, Cell biology, Kinetics, HEK293 Cells, Carbachol, Intracellular, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::affdfb006164c1e9c8cc4cc1ef567fdfTest
https://doi.org/10.2220/biomedres.35.185Test -
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المؤلفون: Owen N, Vickery, Catarina A, Carvalheda, Saheem A, Zaidi, Andrei V, Pisliakov, Vsevolod, Katritch, Ulrich, Zachariae
المصدر: Structure (London, England : 1993). 26(1)
مصطلحات موضوعية: Protein Conformation, alpha-Helical, Receptor, Muscarinic M2, Binding Sites, Ion Transport, Amino Acid Motifs, Sodium, Static Electricity, Cations, Monovalent, Molecular Dynamics Simulation, Ligands, Article, Kinetics, Phosphatidylcholines, Humans, Thermodynamics, Carbachol, Protein Interaction Domains and Motifs, Hydrophobic and Hydrophilic Interactions, Ion Channel Gating, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::6812cfb204cf6332bb01eb9b201a9831Test
https://pubmed.ncbi.nlm.nih.gov/29249607Test -
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المؤلفون: Gregory W. Sawyer, Frederick J. Ehlert, Jon P. Hart
المصدر: Journal of Pharmacological and Toxicological Methods. 53:219-233
مصطلحات موضوعية: Atropine, Time Factors, Carbachol, Recombinant Fusion Proteins, CHO Cells, Muscarinic Antagonists, Ligands, Toxicology, Binding, Competitive, Radioligand Assay, Cricetinae, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Receptor, Furin, Pharmacology, Microscopy, Confocal, Models, Statistical, Dose-Response Relationship, Drug, biology, Chemistry, Chinese hamster ovary cell, Cell Membrane, Receptor, Muscarinic M1, Muscarinic acetylcholine receptor M1, Fusion protein, Protein Structure, Tertiary, Kinetics, Membrane, Biochemistry, Mutation, biology.protein, Biophysics, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::72df4f795369e87002386cc47e8710b2Test
https://doi.org/10.1016/j.vascn.2005.08.006Test -
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المؤلفون: James W. Wells, Paul S.-H. Park, Chi Shing Sum
المصدر: Journal of Biological Chemistry. 277:36188-36203
مصطلحات موضوعية: Agonist, Insecta, Time Factors, Carbachol, Protein Conformation, Swine, medicine.drug_class, G protein, Blotting, Western, Muscarinic Agonists, Ligands, Biochemistry, Cell Line, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Enzyme Inhibitors, Receptor, Molecular Biology, Receptor, Muscarinic M2, Chemistry, Oxotremorine, Sulfhydryl Reagents, Parasympatholytics, Muscarinic acetylcholine receptor M2, Cell Biology, N-Methylscopolamine, Ligand (biochemistry), Precipitin Tests, Receptors, Muscarinic, Quinuclidinyl Benzilate, Kinetics, Models, Chemical, Ethylmaleimide, Biophysics, Protein Binding, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19951c77d8cefaaf54595a5860027acfTest
https://doi.org/10.1074/jbc.m201731200Test -
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المؤلفون: Markus Frings, Paschal A. Oude Weernink, Marie-Luise Mono, Martina Schmidt, Yuanjian Guo, Karl Jakobs, Sandrine Evellin, Li Han
المصدر: Journal of Biological Chemistry. 275:32603-32610
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Protein Kinase C-alpha, medicine.drug_class, Inositol Phosphates, Stimulation, Inositol 1,4,5-Trisphosphate, Transfection, Biochemistry, Receptor tyrosine kinase, Cell Line, chemistry.chemical_compound, Adenosine Triphosphate, GTP-Binding Proteins, Internal medicine, Protein Kinase C beta, Lysophosphatidic acid, Muscarinic acetylcholine receptor, medicine, Humans, Molecular Biology, Protein Kinase C, Protein kinase C, G protein-coupled receptor, Platelet-Derived Growth Factor, Receptor, Muscarinic M3, Receptor, Muscarinic M2, Epidermal Growth Factor, Phospholipase C, biology, Receptor Protein-Tyrosine Kinases, Cell Biology, Receptors, Muscarinic, Recombinant Proteins, Cell biology, Isoenzymes, Kinetics, Endocrinology, chemistry, Type C Phospholipases, biology.protein, Carbachol
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca2452a38c3cbdbeb5c9054b1a3c7c82Test
https://doi.org/10.1074/jbc.m004784200Test -
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المؤلفون: Helen P. Meijer, Jack A. Groot, Judith C. J. Oprins
المصدر: American Journal of Physiology-Cell Physiology. 278:C463-C472
مصطلحات موضوعية: medicine.medical_specialty, Indoles, Carbachol, Physiology, Muscarinic Agonists, Pharmacology, Biology, Cell Line, Membrane Potentials, Maleimides, Internal medicine, Muscarinic acetylcholine receptor, Phospholipase D, medicine, Humans, Enzyme Inhibitors, Intestinal Mucosa, Receptor, Protein Kinase C, Protein kinase C, Tumor Necrosis Factor-alpha, Cell Membrane, Cell Biology, Muscarinic acetylcholine receptor M1, Apical membrane, Propranolol, Receptors, Muscarinic, Kinetics, Endocrinology, Signal transduction, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cab6dc4371692400206b76539bcb4bd5Test
https://doi.org/10.1152/ajpcell.2000.278.3.c463Test