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1
المؤلفون: José N. Nobrega, Tarek K. Rajji, Bruce G. Pollock, Roger Raymond
المصدر: Journal of Pharmacological and Toxicological Methods. 112:107118
مصطلحات موضوعية: Agonist, Carbachol, medicine.drug_class, Pharmacology, Toxicology, Fluorescence, Calcium in biology, Cricetulus, Cricetinae, medicine, Animals, Humans, Fluorometry, Pharmacokinetics, Receptors, Cholinergic, Cognitive decline, Acetylcholine receptor, Chemistry, Receptor, Muscarinic M1, Antagonist, Muscarinic acetylcholine receptor M1, Radioactivity, Pharmaceutical Preparations, Cholinergic, Calcium, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::162de83b3e6b13d4403ffbc148be4f20Test
https://doi.org/10.1016/j.vascn.2021.107118Test -
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المؤلفون: Jelena Momirov, Alena Randáková, John Boulos, Jan Jakubík, John M. Boulos
المصدر: Chemical Biology & Drug Design. 91:93-104
مصطلحات موضوعية: 0301 basic medicine, Carbachol, Pyridines, Pilot Projects, CHO Cells, Muscarinic Antagonists, Pharmacology, Ligands, Biochemistry, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Allosteric Regulation, Cricetinae, Drug Discovery, Muscarinic acetylcholine receptor M5, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M4, medicine, Animals, Humans, Protein Isoforms, Binding Sites, Chemistry, Organic Chemistry, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, N-Methylscopolamine, Receptors, Muscarinic, 030104 developmental biology, Drug Design, Acetylcholinesterase, Molecular Medicine, Pharmacophore, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::47b579d475c0acbbac04c6b9a5286c50Test
https://doi.org/10.1111/cbdd.13059Test -
3
المؤلفون: Deborah L. Smith, Sarah J. Neal, Lei Zhang, Jeremy R. Edgerton, Jennifer E. Davoren, Sarah Grimwood, John T. Lazzaro, Chewah Lee
المصدر: Molecular Pharmacology. 90:177-187
مصطلحات موضوعية: Male, 0301 basic medicine, Carbachol, Allosteric modulator, Pyridines, Stereochemistry, Allosteric regulation, CHO Cells, Isoindoles, Hippocampus, Rats, Sprague-Dawley, Radioligand Assay, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Allosteric Regulation, Cricetinae, Muscarinic acetylcholine receptor, medicine, Radioligand, Animals, Humans, Fluorometry, Pharmacology, Membranes, Chemistry, Ligand binding assay, Receptor, Muscarinic M1, N-Methylscopolamine, Acetylcholine, Electrophysiological Phenomena, Kinetics, HEK293 Cells, 030104 developmental biology, Positron-Emission Tomography, Autoradiography, Molecular Medicine, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59a4cbb153c3abcd01cb4427f9543370Test
https://doi.org/10.1124/mol.116.104737Test -
4
المؤلفون: Alexey Pronin, Vladlen Z. Slepak, Qiang Wang
مصطلحات موضوعية: 0301 basic medicine, Agonist, Male, medicine.medical_specialty, endocrine system, Carbachol, medicine.drug_class, CHO Cells, Muscarinic Antagonists, Pharmacology, Muscarinic Agonists, Muscarinic agonist, 03 medical and health sciences, Mice, 0302 clinical medicine, Cricetulus, Internal medicine, Cricetinae, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Receptor, Receptor, Muscarinic M3, Dose-Response Relationship, Drug, Chemistry, Pilocarpine, Muscarinic acetylcholine receptor M3, Articles, Mice, Inbred C57BL, 030104 developmental biology, Endocrinology, HEK293 Cells, Molecular Medicine, Signal transduction, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f3f7b56792ce0ac740d905ede9a46a8cTest
https://europepmc.org/articles/PMC5635516Test/ -
5
المؤلفون: Sandra Den Hoedt, Christopher J. Langmead, Patrick R. Gentry, Arthur Christopoulos, Patrick M. Sexton, Alice E. Berizzi, Patricia Rueda
المصدر: Molecular pharmacology. 90(4)
مصطلحات موضوعية: 0301 basic medicine, Agonist, Atropine, Allosteric modulator, Carbachol, Indazoles, Indoles, medicine.drug_class, Inositol Phosphates, Allosteric regulation, CHO Cells, Pharmacology, Partial agonist, 03 medical and health sciences, Radioligand Assay, 0302 clinical medicine, Cricetulus, Allosteric Regulation, Cricetinae, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Sulfonamides, Receptor, Muscarinic M5, Phenoxybenzamine, Chemistry, Imidazoles, Cooperative binding, Acetylcholine, 030104 developmental biology, Molecular Medicine, 030217 neurology & neurosurgery, Allosteric Site, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b19f52c9c1d4b178ccd5a931c85b98f1Test
https://pubmed.ncbi.nlm.nih.gov/27461343Test -
6
المؤلفون: Giulio Vistoli, Laura Raimondi, Rosanna Matucci, Annunziatina Laurino
مصطلحات موضوعية: 0301 basic medicine, Male, medicine.medical_specialty, 3-iodothyrothyronamine, Urinary Bladder, Muscarinic receptors, Muscarinic Antagonists, Pharmacology, 03 medical and health sciences, Internal medicine, Catalytic Domain, Cricetinae, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M5, medicine, Muscarinic acetylcholine receptor M4, Thyronines, Animals, Humans, Phosphorylation, Receptor, Thyroid, Mitogen-Activated Protein Kinase 1, Receptor, Muscarinic M3, Mitogen-Activated Protein Kinase 3, Chemistry, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, Acetylcholine, Rats, Molecular Docking Simulation, 3-iodothyroacetic acid, 030104 developmental biology, Endocrinology, Carbachol, medicine.drug, Muscle Contraction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c01eb65ef66fdd7244b6881399adb955Test
http://hdl.handle.net/2158/1079396Test -
7
المؤلفون: Banu Aydın, Beki Kan, Hülya Cabadak
المصدر: Journal of Receptors and Signal Transduction. 31:26-32
مصطلحات موضوعية: Atropine, Time Factors, Carbachol, Blotting, Western, CHO Cells, Muscarinic Antagonists, Pharmacology, Biology, Biochemistry, Cricetulus, Cricetinae, Leukemia, Myelogenous, Chronic, BCR-ABL Positive, Muscarinic acetylcholine receptor M5, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M4, medicine, Animals, Humans, RNA, Messenger, Molecular Biology, Receptor, Muscarinic M3, Receptor, Muscarinic M2, Receptor, Muscarinic M4, Gene Expression Regulation, Leukemic, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Cell Biology, Muscarinic acetylcholine receptor M1, Receptors, Muscarinic, Molecular biology, K562 Cells, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9b63df4355a2850eba289bba9aae9935Test
https://doi.org/10.3109/10799893.2010.506484Test -
8
المؤلفون: Paola Casarosa, Tobias Kiechle, Michael P. Pieper, Florian Gantner, Peter Sieger
المصدر: Journal of Pharmacology and Experimental Therapeutics. 333:201-209
مصطلحات موضوعية: medicine.medical_specialty, Carbachol, Drug Inverse Agonism, Protein Conformation, CHO Cells, Muscarinic Antagonists, Muscarinic Agonists, Pharmacology, Cricetulus, Genes, Reporter, Cricetinae, Internal medicine, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Inverse agonist, Luciferases, Inositol phosphate, Receptor, Receptor, Muscarinic M3, chemistry.chemical_classification, Chinese hamster ovary cell, Muscarinic acetylcholine receptor M3, Up-Regulation, Transcription Factor AP-1, Endocrinology, chemistry, Molecular Medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::958e2574802614bd5fa77fba50aceb13Test
https://doi.org/10.1124/jpet.109.163188Test -
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المؤلفون: Pavel Michal, Esam E. El-Fakahany, Vladimír Rudajev, Vladimír Doležal
المصدر: European Journal of Pharmacology. 606:50-60
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Carbachol, Membrane permeability, G protein, medicine.drug_class, CHO Cells, Muscarinic Antagonists, Second Messenger Systems, Article, Cricetulus, GTP-Binding Proteins, Cricetinae, Internal medicine, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Receptor, Acetylcholine receptor, Pharmacology, Receptor, Muscarinic M2, Chemistry, Cell Membrane, beta-Cyclodextrins, Muscarinic acetylcholine receptor M2, N-Methylscopolamine, Molecular biology, Acetylcholine, Cholesterol, Endocrinology, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::74a35ddb8c291e0e65da44336769465eTest
https://doi.org/10.1016/j.ejphar.2009.01.028Test -
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المؤلفون: Elmar M Udarbe Zamora, Jing Liu, Carey Pope
المصدر: Journal of Toxicology and Environmental Health, Part A. 71:1440-1447
مصطلحات موضوعية: Health, Toxicology and Mutagenesis, media_common.quotation_subject, CHO Cells, Muscarinic Agonists, Pharmacology, Biology, Toxicology, Muscarinic agonist, Cricetulus, Species Specificity, Cricetinae, Muscarinic acetylcholine receptor M5, Enzyme-linked receptor, Animals, Humans, Phosphorylation, Receptor, Internalization, G protein-coupled receptor, media_common, Receptor, Muscarinic M2, Parasympatholytics, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, N-Methylscopolamine, Immunohistochemistry, Rats, Cell biology, Carbachol, Chlorpyrifos
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::afa50f9f986a317bf82fb780feff2a7dTest
https://doi.org/10.1080/15287390802328887Test