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المؤلفون: Yen-Der Li, Michelle W. Ma, Muhammad Murtaza Hassan, Kedar Puvar, Mingxing Teng, Brittany Sandoval, Ryan Lumpkin, Scott B. Ficarro, Michelle Y. Wang, Shawn Xu, Brian J. Groendyke, Logan H. Sigua, Isidoro Tavares, Charles Zou, Jonathan M. Tsai, Paul M. Park, Hojong Yoon, Radosław P. Nowak, Jarrod A. Marto, Jun Qi, Katherine A. Donovan, Mikołaj Słabicki, Nathanael S. Gray, Eric S. Fischer, Benjamin L. Ebert
المصدر: Cancer Research. 83:3424-3424
مصطلحات موضوعية: Cancer Research, Oncology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::c3a5b6eba7ac746545c7a80669b65a86Test
https://doi.org/10.1158/1538-7445.am2023-3424Test -
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المؤلفون: Li Wang, Scott B. Ficarro, Hao Wu, John M. Hatcher, Jarrod A. Marto, Nathanael S. Gray, Steven P. Treon, Sara J. Buhrlage, Guang Yang
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: biology, 010405 organic chemistry, Kinase, Organic Chemistry, Interleukin, medicine.disease, 01 natural sciences, Biochemistry, 0104 chemical sciences, Lymphoma, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, chemistry, Cell culture, hemic and lymphatic diseases, Ibrutinib, Drug Discovery, medicine, biology.protein, Cancer research, Cytotoxic T cell, Bruton's tyrosine kinase, B-cell lymphoma
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::22b6a1d71c35abaa77c3807f4aa62aa6Test
https://doi.org/10.1021/acsmedchemlett.0c00378Test -
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المؤلفون: Kun Ping Lu, Hyuk-Soo Seo, Yujin Chun, Christopher M. Browne, Theresa D. Manz, Xiao Zhen Zhou, Zainab M. Doctor, Xiaolan Lian, Zoe C. Yeoh, Shin Kibe, Scott B. Ficarro, Nir London, Benika J. Pinch, Nicholas E. Vangos, Behnam Nabet, Stephen Buratowski, Dina Daitchman, Shingo Kozono, Daniel Zaidman, Nathanael S. Gray, Jarrod A. Marto, Mikaela L. Mohardt, Li Tan, Sirano Dhe-Paganon, Ezekiel A. Geffken
المصدر: Nature chemical biology
مصطلحات موضوعية: endocrine system diseases, Cell Survival, Protein Conformation, Mutant, Antineoplastic Agents, Crystallography, X-Ray, medicine.disease_cause, Article, Proto-Oncogene Proteins p21(ras), Mice, 03 medical and health sciences, Cell Line, Tumor, medicine, Animals, Humans, Cysteine, Viability assay, Enzyme Inhibitors, Molecular Biology, 030304 developmental biology, 0303 health sciences, Chemistry, 030302 biochemistry & molecular biology, HEK 293 cells, Cancer, Cell Biology, medicine.disease, digestive system diseases, Gene Expression Regulation, Neoplastic, NIMA-Interacting Peptidylprolyl Isomerase, Pancreatic Neoplasms, Cell Transformation, Neoplastic, HEK293 Cells, Cell culture, Drug Design, NIH 3T3 Cells, Cancer research, PIN1, KRAS, Carcinogenesis, Carcinoma, Pancreatic Ductal
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6565cbd6de180dcf92ba1d74b5e545e0Test
https://doi.org/10.1038/s41589-020-0550-9Test -
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المؤلفون: Sara J. Buhrlage, William C. Hahn, Sumner Perera, Ellen Weisberg, Robert S. Magin, Kenneth C. Anderson, Dharminder Chauhan, Arghya Ray, Wai Cheung Chan, Nathan J. Schauer, Laura M. Doherty, Björn Stolte, Sirano Dhe-Paganon, Rebekka M. Roberts, Jarrod A. Marto, Wanyi Hu, Sarah A. Boswell, James D. Griffin, Scott B. Ficarro, Peter K. Sorger, Andrew O. Giacomelli, Jianing Li, Kimberly Stegmaier, Roxana E. Iacob, Kyle T. McKay, John R. Engen, Xiaoxi Liu
المصدر: Scientific Reports, Vol 10, Iss 1, Pp 1-15 (2020)
Scientific Reportsمصطلحات موضوعية: lcsh:Medicine, Antineoplastic Agents, Apoptosis, Article, Target validation, Deubiquitinating enzyme, Ubiquitin-Specific Peptidase 7, 03 medical and health sciences, 0302 clinical medicine, Ubiquitin, Cell Line, Tumor, Humans, Cytotoxic T cell, PTEN, Protease Inhibitors, lcsh:Science, Cell Proliferation, 030304 developmental biology, 0303 health sciences, Multidisciplinary, biology, Chemistry, Small molecules, lcsh:R, Ubiquitination, 3. Good health, Cell culture, 030220 oncology & carcinogenesis, Cancer cell, FOXO4, MCF-7 Cells, biology.protein, Cancer research, Mdm2, lcsh:Q, Tumor Suppressor Protein p53
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::89403c0f98aeff7c94fa67b62b62d125Test
http://link.springer.com/article/10.1038/s41598-020-62076-xTest -
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المؤلفون: Evon Poon, Anli Yang, Xiao Zhou, Efrat Resnick, Daniel Zaidman, Roni Oren, Yann Jamin, Shingo Kozono, Colin J. Daniel, Ellen M. Langer, Shijie He, Behnam Nabet, Yu-Hong Chen, Christopher M. Browne, Hyuk-Soo Seo, Louis Chesler, Kun Ping Lu, Benika J. Pinch, Rosalie C. Sears, Shin Kibe, Liat Stoler-Barak, Ziv Shulman, Nir London, Samuel Sidi, Christian Dubiella, Thomas Look, Nicholas E. Vangos, Kazuhiro Koikawa, Xiaolan Lian, Chunhui Wang, Nathaniel Gray, Trevor Manz, Jarrod A. Marto, Richa B. Shah, Ezekiel A. Geffken, Sirano Dhe-Paganon, Scott B. Ficarro
مصطلحات موضوعية: 0303 health sciences, Chemistry, Tumor initiation, medicine.disease, 3. Good health, 03 medical and health sciences, 0302 clinical medicine, Downregulation and upregulation, In vivo, Tumor progression, 030220 oncology & carcinogenesis, Neuroblastoma, Cancer cell, Cancer research, medicine, PIN1, Chemoproteomics, 030304 developmental biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e3ceb5d0f3a7e590d161df59af1ffd9Test
https://doi.org/10.1101/2020.03.20.998443Test -
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المؤلفون: Baishan Jiang, Scott B. Ficarro, Tinghu Zhang, Zhixiang He, Yang Gao, Nathanael S. Gray, Jarrod A. Marto, Jianwei Che, Jie Jiang
المصدر: Cell chemical biology. 27(12)
مصطلحات موضوعية: Models, Molecular, MAP Kinase Kinase 4, Clinical Biochemistry, Cell, Amino Acid Motifs, MAP Kinase Kinase 7, Biology, medicine.disease_cause, Biochemistry, Cell Line, Tumor, Drug Discovery, medicine, Humans, Kinome, Molecular Biology, Protein Kinase Inhibitors, Cell Proliferation, Pharmacology, Kinase, Dual inhibitor, medicine.anatomical_structure, Covalent bond, Drug Design, Cancer research, Molecular Medicine, Phosphorylation, Carcinogenesis, Cysteine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::049342c225539a7c75034388e9726fbbTest
https://pubmed.ncbi.nlm.nih.gov/32916088Test -
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المؤلفون: Sirano Dhe-Paganon, Benika J. Pinch, Mark W. Zimmerman, Richa B. Shah, Kun Ping Lu, Jarrod A. Marto, Shuning He, Eriko Koide, Daniel Zaidman, Christopher M. Browne, Ziv Shulman, Barbara Martins da Costa, Christian Dubiella, Evon Poon, Guillaume Adelmant, Nir London, Xiao Zhen Zhou, Chu Wang, Ellen M. Langer, Kazuhiro Koikawa, Theresa D. Manz, Thomas Look, Xiaolan Lian, Hyuk-Soo Seo, Annan Yang, Louis Chesler, Ezekiel A. Geffken, Liat Stoler-Barak, Shin Kibe, Efrat Resnick, Nicholas E. Vangos, Shabnam Sharifzadeh, Shingo Kozono, Colin J. Daniel, Scott B. Ficarro, Roni Oren, Ying Chen, Nathanael S. Gray, Rosalie C. Sears, Samuel Sidi, Adi Rogel, Zainab M. Doctor, Behnam Nabet, Yann Jamin
المصدر: Nat Chem Biol
مصطلحات موضوعية: Cell Survival, Antineoplastic Agents, Apoptosis, Article, Proto-Oncogene Proteins c-myc, 03 medical and health sciences, Mice, Structure-Activity Relationship, Downregulation and upregulation, In vivo, Pancreatic cancer, Neuroblastoma, medicine, Tumor Cells, Cultured, Animals, Humans, Chemoproteomics, Enzyme Inhibitors, Molecular Biology, 030304 developmental biology, Cell Proliferation, 0303 health sciences, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, 030302 biochemistry & molecular biology, Cancer, Cell Biology, Neoplasms, Experimental, medicine.disease, Mice, Inbred C57BL, NIMA-Interacting Peptidylprolyl Isomerase, Tumor progression, Cancer research, PIN1, Drug Screening Assays, Antitumor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8338cdca0db7efbd0dc3ed699641997fTest
https://pubmed.ncbi.nlm.nih.gov/34040180Test -
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المؤلفون: Guangyan Du, Jianwei Che, Tinghu Zhang, Nathanael S. Gray, Henning Nathaniel, Scott B. Ficarro, Jie Jiang, Jarrod A. Marto, Andrew J. Aguirre, Deepak Gurbani, Suman Rao, Kenneth D. Westover, Peter K. Sorger, Annan Yang
المصدر: J Med Chem
مصطلحات موضوعية: AAA Domain, 01 natural sciences, Article, 03 medical and health sciences, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Anilides, Amino Acid Sequence, Cysteine, Protein Kinase Inhibitors, 030304 developmental biology, Cell Proliferation, 0303 health sciences, Molecular Structure, Kinase, Chemistry, 0104 chemical sciences, Dasatinib, Mice, Inbred C57BL, 010404 medicinal & biomolecular chemistry, Pyrimidines, src-Family Kinases, Cell culture, Drug Design, Cancer research, Molecular Medicine, Signal transduction, Drug Screening Assays, Antitumor, Bosutinib, Proto-oncogene tyrosine-protein kinase Src, medicine.drug, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::590fc495fb569d9115bb1caa5ba74b3cTest
https://pubmed.ncbi.nlm.nih.gov/31935084Test -
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المؤلفون: Martin S. Tallman, Ross L. Levine, Andrei V. Krivtsov, Jarrod A. Marto, Casie Reed, Conor O’Donnell, Alex Kentsis, Christina Y. Yim, Fiona C. Brown, Mithat Gonen, Gayle P. Pouliot, Richard Koche, Peter Romanienko, Barbara Spitzer, Craig McCarthy, Crystal Stutzke, Josée Hébert, Elisabeth Paietta, Willie Mark, Anthony Letai, Vincent-Philippe Lavallée, Guy Sauvageau, Elisa de Stanchina, Paolo Cifani, Venkatraman E. Seshan, Patrick Bhola, Ari Melnick, Eric Still, Shehana Gunasekera, Scott A. Armstrong, Sumiko Takao, Scott B. Ficarro
المصدر: Cancer Discovery. 8:478-497
مصطلحات موضوعية: Proteomics, 0301 basic medicine, Myeloid, Antineoplastic Agents, Mice, Transgenic, Article, Cell Line, Mice, 03 medical and health sciences, 0302 clinical medicine, hemic and lymphatic diseases, medicine, Animals, Humans, MEF2C, Phosphorylation, Transcription factor, Gene Expression Regulation, Leukemic, MEF2 Transcription Factors, Kinase, business.industry, Myeloid leukemia, Cancer, medicine.disease, Leukemia, Myeloid, Acute, Leukemia, 030104 developmental biology, medicine.anatomical_structure, Oncology, Drug Resistance, Neoplasm, 030220 oncology & carcinogenesis, Cancer research, business, Protein Processing, Post-Translational
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d25f36a31ccd798c9866696a88aca7dbTest
https://doi.org/10.1158/2159-8290.cd-17-1271Test -
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المؤلفون: Sofia Dust, Jie Jiang, Kanchan Anand, Jarrod A. Marto, Tinghu Zhang, Nathanael S. Gray, Ines H. Kaltheuner, Bo Kyung Alex Seong, Nicholas Kwiatkowski, Matthias Geyer, Fleur M. Ferguson, Baishan Jiang, Kimberly Stegmaier, Scott B. Ficarro, Ann Katrin Greifenberg, Amanda Balboni Iniguez
المصدر: European Journal of Medicinal Chemistry. 221:113481
مصطلحات موضوعية: Male, DNA damage, RNA polymerase II, 01 natural sciences, Mice, Structure-Activity Relationship, 03 medical and health sciences, Downregulation and upregulation, Transcription (biology), CDC2 Protein Kinase, Drug Discovery, Animals, Humans, Structure–activity relationship, Anilides, Protein Kinase Inhibitors, Cells, Cultured, 030304 developmental biology, Pharmacology, 0303 health sciences, Dose-Response Relationship, Drug, Molecular Structure, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, General Medicine, Cyclin-Dependent Kinases, 0104 chemical sciences, Pyrimidines, Protein kinase domain, Cancer cell, Microsomes, Liver, biology.protein, Cancer research, CDK12
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ee0596e688b658a34bb628083ae27aa6Test
https://doi.org/10.1016/j.ejmech.2021.113481Test