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المؤلفون: Matucci, R., Ottaviani, M. F., Barbieri, M., Elisabetta Cerbai, Mugelli, A.
المصدر: Università degli studi di Firenze-IRIS
Scopus-Elsevierمصطلحات موضوعية: Male, Dose-Response Relationship, Drug, Free Radicals, Nifedipine, Myocardium, Electron Spin Resonance Spectroscopy, Heart, Calcium Channel Blockers, Membrane Potentials, Rats, Electrophysiology, Cardiomyocytes, Darodipine, Electron spin resonance, L-type calcium current, Oxygen radicals, Papers, Animals, Rats, Wistar, Reactive Oxygen Species
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::fd0ea03f8ff522202140d52f1794d636Test
http://hdl.handle.net/11392/1696111Test -
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المؤلفون: Simona Saponara, Massimo Baroni, Domenico Spinelli, Barbara Cosimelli, Elda Severi, Pierfranco Ioan, Camillo Rosano, Roberta Budriesi, Fabio Fusi, Rosanna Matucci, Emanuele Carosati, Simon Cross, Maria Frosini, Maurizio Viale, Alberto Chiarini, Matteo Micucci
المساهمون: Spinelli, D., Budriesi, R., Cosimelli, B., Severi, E., Micucci, M., Baroni, M., Fusi, F., Ioan, P., Cross, S., Frosini, M., Saponara, S., Matucci, R., Rosano, C., Viale, M., Chiarini, A., Carosati, E., Domenico, Spinelli, Roberta, Budriesi, Cosimelli, Barbara, Elda, Severi, Matteo, Micucci, Massimo, Baroni, Fabio, Fusi, Pierfranco, Ioan, Simon, Cro, Maria, Frosini, Simona, Saponara, Rosanna, Matucci, Camillo, Rosano, Maurizio, Viale, Alberto, Chiarini, Emanuele, Carosati
المصدر: Molecules, Vol 19, Iss 10, Pp 16543-16572 (2014)
Molecules
Volume 19
Issue 10
Pages 16543-16572مصطلحات موضوعية: oxadiazolothiazinones, Pharmaceutical Science, Quantitative Structure-Activity Relationship, Multidrug resistance, ternary complex, Analytical Chemistry, Heterocyclic Compounds, Drug Discovery, Ternary complex, L-type calcium channel, Oxadiazoles, Chemistry, Calcium Channel Blockers, Molecular Docking Simulation, Subfamily B, Chemistry (miscellaneous), docking, Molecular Medicine, ATP Binding Cassette Transporter, Subfamily B, Animals, Guinea Pigs, Heart Atria, Muscle, Smooth, Structural Homology, Protein, Muscle, Smooth, Pharmacophore, structure-activity relationship, L-type calcium channels, oxadiazolothiazinone, P-glycoprotein, Quantitative structure–activity relationship, Stereochemistry, In silico, negative inotropic activity, ATP Binding Cassette Transporter, Fingerprints for Ligands and Proteins (FLAP), L-Type Calcium Channels (LTCC), Article, lcsh:QD241-441, lcsh:Organic chemistry, Homology modeling, Physical and Theoretical Chemistry, multidrug resistance (MDR1), 3D-QSAR, Structural Homology, Virtual screening, Calcium channel, Protein, Organic Chemistry, Combinatorial chemistry, Docking (molecular), pharmacophore modeling
وصف الملف: application/pdf; STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::61554762b7203fa9fbc751ecaa3e5b93Test
https://hdl.handle.net/11576/2696050Test -
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المؤلفون: Fabio Fusi, Domenico Spinelli, Alberto Chiarini, Raffaella Spisani, Emanuele Carosati, Philip J. Stephens, Maria Frosini, Roberta Budriesi, Gabriele Cruciani, Francesco Gasparrini, Barbara Cosimelli, Frank J. Devlin, Alessia Ciogli, Pierfranco Ioan, Rosanna Matucci
المساهمون: Carosati, E, Cruciani, G, Chiarini, A, Budriesi, R, Ioan, P, Spisani, R, Spinelli, D, Cosimelli, Barbara, Fusi, F, Frosini, M, Matucci, R, Gasparrini, F, Ciogli, A, STEPHENS P., J, Devlin, F. J.
مصطلحات موضوعية: binding, Calcium Channels, L-Type, calcium channel antagonist, Stereochemistry, drug design, In silico, Guinea Pigs, Drug Evaluation, Preclinical, Ligands, Structure-Activity Relationship, chemotypes, ligand channel interaction, medicinal chemistry, Drug Discovery, Animals, Myocytes, Cardiac, Heart Atria, Calcium entry, Virtual screening, Oxadiazoles, Binding Sites, Molecular Structure, Chemistry, Calcium channel, diltiazem, Absolute configuration, Muscle, Smooth, Stereoisomerism, Papillary Muscles, Calcium Channel Blockers, virtual screening, circular dichroism, Databases as Topic, Vibrational circular dichroism, calcium entry blocker, Molecular Medicine, Female, synthesi
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::766918fe8cc1cd3e9d24046cf16cf76aTest
http://hdl.handle.net/11588/102166Test