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1
المؤلفون: Martin F. Fromm, Georg Heinkele, Nicolas Simon, Ute Hofmann, Céline Verstuyft, Hartmut Glaeser, Monika Hitzl, Siegfried Drescher, Christian Schaefer, Thomas E. Mürdter, Oliver Burk, Michel Eichelbaum, Laurent Becquemont
المصدر: Clinical Pharmacology & Therapeutics. 79:449-460
مصطلحات موضوعية: Adult, Male, Digoxin, Midazolam, Enzyme Activators, In Vitro Techniques, Pharmacology, Cell Line, Cytochrome P-450 Enzyme System, Pharmacokinetics, Cell Line, Tumor, Leukocytes, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, RNA, Messenger, Intestinal Mucosa, P-glycoprotein, Pregnane X receptor, biology, CYP3A4, Chemistry, Ursodeoxycholic Acid, Ursodeoxycholic acid, Bioavailability, Intestines, Area Under Curve, biology.protein, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd638350525f5dd52169ddb3cf594f81Test
https://doi.org/10.1016/j.clpt.2006.01.005Test -
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المؤلفون: Pertti J. Neuvonen, Kari T. Kivistö, Julian B. S. Leathart, Mikko Niemi, Mikko Neuvonen, Janne T. Backman, Lauri I. Kajosaari, Ann K. Daly, Michel Eichelbaum
المصدر: Clinical Pharmacology & Therapeutics. 77:468-478
مصطلحات موضوعية: Adult, Male, Genotype, Cmax, Single-nucleotide polymorphism, Biology, Pharmacology, Polymorphism, Single Nucleotide, Cytochrome P-450 CYP2C8, Cytochrome P-450 Enzyme System, Piperidines, Pharmacokinetics, medicine, Cytochrome P-450 CYP3A, Humans, Hypoglycemic Agents, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, CYP2C8, Liver-Specific Organic Anion Transporter 1, Repaglinide, Organic anion-transporting polypeptide, biology.protein, ATP-Binding Cassette Transporters, Female, Aryl Hydrocarbon Hydroxylases, Carbamates, Genes, MDR, SLCO1B1, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e1a3de8b68a232f7346fef6a9756f07cTest
https://doi.org/10.1016/j.clpt.2005.01.018Test -
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المؤلفون: Reijo S. Tilvis, Timo E. Strandberg, Michel Eichelbaum, Matthias Schwab, Mikko Niemi, Martin F. Fromm, Kaisu H. Pitkälä, Florian Lang, Elke Schaeffeler, Kari T. Kivistö
المصدر: American Journal of PharmacoGenomics. 5:191-195
مصطلحات موضوعية: Male, medicine.medical_specialty, Pediatrics, Genotype, Blood Pressure, Single-nucleotide polymorphism, 030204 cardiovascular system & hematology, Polymorphism, Single Nucleotide, 03 medical and health sciences, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Internal medicine, Genetics, medicine, Cytochrome P-450 CYP3A, Humans, Medical history, CYP3A5, Alleles, Finland, Aged, 030304 developmental biology, Aged, 80 and over, Pharmacology, 0303 health sciences, Evidence-Based Medicine, Base Sequence, biology, business.industry, DNA, Odds ratio, 3. Good health, Genotype frequency, Blood pressure, Pharmacogenetics, Hypertension, biology.protein, Molecular Medicine, Female, SLCO1B1, business
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa88ccd12ae4965bdde5b34d8043596aTest
https://doi.org/10.2165/00129785-200505030-00005Test -
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المؤلفون: Martin F. Fromm, Michel Eichelbaum, Oliver Burk, Kari T. Kivistö, Oliver von Richter, Klaus P. Thon
المصدر: Clinical Pharmacology & Therapeutics. 75:172-183
مصطلحات موضوعية: Adult, Male, Enterocyte, Blotting, Western, Statistics, Nonparametric, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Intestine, Small, Cytochrome P-450 CYP3A, medicine, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, Aged, P-glycoprotein, Aged, 80 and over, Pharmacology, biology, CYP3A4, Cytochrome P450, Norverapamil, Middle Aged, Molecular biology, Enterocytes, medicine.anatomical_structure, Gene Expression Regulation, chemistry, Biochemistry, Hepatocyte, Hepatocytes, biology.protein, Duodenum, Female
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9bb8489a61cb545cebcfadb5ba7df9e3Test
https://doi.org/10.1016/j.clpt.2003.10.008Test -
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المؤلفون: Andreas K. Nussler, Kathrin Klein, Ulrich M. Zanger, Oliver Burk, Matthias Schwab, Renzo Wolbold, Peter Neuhaus, Michel Eichelbaum
المصدر: Hepatology. 38:978-988
مصطلحات موضوعية: Adult, Male, Drug, Receptors, Steroid, medicine.medical_specialty, media_common.quotation_subject, Receptors, Cytoplasmic and Nuclear, ATP-binding cassette transporter, Pharmacology, Sex Factors, Cytochrome P-450 Enzyme System, Internal medicine, Cytochrome P-450 CYP3A, medicine, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, RNA, Messenger, Receptor, Life Style, Constitutive Androstane Receptor, Aged, media_common, Pregnane X receptor, Hepatology, biology, CYP3A4, Pregnane X Receptor, Cytochrome P450, Middle Aged, Endocrinology, Liver, Verapamil, biology.protein, Female, Drug metabolism, Transcription Factors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2436915ecde8be75c9d5f021b7f3803bTest
https://doi.org/10.1002/hep.1840380424Test -
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المؤلفون: Julia Blievernicht, Ulrich M. Zanger, Jan G. Hengstler, Andreas K. Nussler, N Nussler, Matthias Schwab, Tanja Saussele, Kathrin Klein, Oliver Burk, Michel Eichelbaum
المصدر: Clinical pharmacology and therapeutics. 82(3)
مصطلحات موضوعية: Male, Receptors, Steroid, CYP2B6, Genotype, Blotting, Western, Dipyrone, Receptors, Cytoplasmic and Nuclear, Pharmacology, In Vitro Techniques, Catalysis, Cytochrome P-450 Enzyme System, Constitutive androstane receptor, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), Enzyme inducer, Cells, Cultured, Constitutive Androstane Receptor, Aged, Pregnane X receptor, biology, CYP3A4, Dose-Response Relationship, Drug, Chemistry, Reverse Transcriptase Polymerase Chain Reaction, Anti-Inflammatory Agents, Non-Steroidal, Pregnane X Receptor, Cytochrome P450 reductase, Oxidoreductases, N-Demethylating, DNA, Middle Aged, Metamizole, Isoenzymes, Cytochrome P-450 CYP2B6, Liver, Enzyme inhibitor, Enzyme Induction, biology.protein, Hepatocytes, Microsomes, Liver, RNA, Female, Aryl Hydrocarbon Hydroxylases, medicine.drug, Plasmids, Transcription Factors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f2732a57085a33507063701647d670fTest
https://pubmed.ncbi.nlm.nih.gov/17344806Test -
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المؤلفون: Kari T. Kivistö, Michel Eichelbaum, Karl Bodin, Mikko Niemi, Martin F. Fromm, Leif Bertilsson, Ulf Diczfalusy
المصدر: Karolinska Institutet
مصطلحات موضوعية: medicine.medical_specialty, ATP Binding Cassette Transporter, Subfamily B, Genotype, Organic Anion Transporters, Single-nucleotide polymorphism, Pharmacology, Cytochrome P-450 Enzyme System, Internal medicine, polycyclic compounds, Genetics, medicine, Cytochrome P-450 CYP3A, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, General Pharmacology, Toxicology and Pharmaceutics, Molecular Biology, Genetics (clinical), Antibacterial agent, Polymorphism, Genetic, biology, CYP3A4, Liver-Specific Organic Anion Transporter 1, Cytochrome P450, Hydroxycholesterols, Organic anion-transporting polypeptide, Endocrinology, Liver, Enzyme Induction, biology.protein, Molecular Medicine, Rifampin, SLCO1B1, Rifampicin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5313bd8a3a31d1de7bc93f990a49e9abTest
https://pubmed.ncbi.nlm.nih.gov/16847425Test -
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المؤلفون: Ulrich M. Zanger, Ina Koch, Jürgen Brockmöller, Regina Weil, Renzo Wolbold, Oliver Burk, Peter Neuhaus, Andreas K. Nuessler, Leszek Wojnowski, Michel Eichelbaum, Elisabeth Hustert
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 30(10)
مصطلحات موضوعية: Pharmacology, Messenger RNA, biology, CYP3A4, CYP3A, Pharmaceutical Science, Cytochrome P450, Gene Expression, Genetic Variation, Molecular biology, Isozyme, Isoenzymes, Cytochrome P-450 Enzyme System, Liver, Organ Specificity, Gene expression, biology.protein, Cytochrome P-450 CYP3A, Humans, RNA, Messenger, Gene, CYP3A7
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::28d5b00b276088c2629c6ddaf3444bc9Test
https://pubmed.ncbi.nlm.nih.gov/12228187Test -
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المؤلفون: Michel Eichelbaum, Heyo K. Kroemer, Ute Hofmann, Frank Bohnenstengel
المصدر: European journal of clinical pharmacology. 51(3-4)
مصطلحات موضوعية: In Vitro Techniques, Mixed Function Oxygenases, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Cytochrome P-450 CYP1A2, Cytochrome P-450 CYP3A, medicine, Chloroacetaldehyde, Humans, Pharmacology (medical), Antineoplastic Agents, Alkylating, Cyclophosphamide, Pharmacology, chemistry.chemical_classification, Unspecific monooxygenase, biology, Cytochrome P450, General Medicine, Prodrug, Enzyme, chemistry, Mechanism of action, Biochemistry, biology.protein, Microsome, medicine.symptom, Oxidation-Reduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58c77016958f8060e43d8a2404ffc68fTest
https://pubmed.ncbi.nlm.nih.gov/9010702Test