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1
المؤلفون: Martin F. Fromm, Georg Heinkele, Nicolas Simon, Ute Hofmann, Céline Verstuyft, Hartmut Glaeser, Monika Hitzl, Siegfried Drescher, Christian Schaefer, Thomas E. Mürdter, Oliver Burk, Michel Eichelbaum, Laurent Becquemont
المصدر: Clinical Pharmacology & Therapeutics. 79:449-460
مصطلحات موضوعية: Adult, Male, Digoxin, Midazolam, Enzyme Activators, In Vitro Techniques, Pharmacology, Cell Line, Cytochrome P-450 Enzyme System, Pharmacokinetics, Cell Line, Tumor, Leukocytes, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, RNA, Messenger, Intestinal Mucosa, P-glycoprotein, Pregnane X receptor, biology, CYP3A4, Chemistry, Ursodeoxycholic Acid, Ursodeoxycholic acid, Bioavailability, Intestines, Area Under Curve, biology.protein, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd638350525f5dd52169ddb3cf594f81Test
https://doi.org/10.1016/j.clpt.2006.01.005Test -
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المؤلفون: Martin F. Fromm, Michel Eichelbaum, Oliver Burk, Kari T. Kivistö, Oliver von Richter, Klaus P. Thon
المصدر: Clinical Pharmacology & Therapeutics. 75:172-183
مصطلحات موضوعية: Adult, Male, Enterocyte, Blotting, Western, Statistics, Nonparametric, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Intestine, Small, Cytochrome P-450 CYP3A, medicine, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, Aged, P-glycoprotein, Aged, 80 and over, Pharmacology, biology, CYP3A4, Cytochrome P450, Norverapamil, Middle Aged, Molecular biology, Enterocytes, medicine.anatomical_structure, Gene Expression Regulation, chemistry, Biochemistry, Hepatocyte, Hepatocytes, biology.protein, Duodenum, Female
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9bb8489a61cb545cebcfadb5ba7df9e3Test
https://doi.org/10.1016/j.clpt.2003.10.008Test -
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المؤلفون: Andreas K. Nussler, Kathrin Klein, Ulrich M. Zanger, Oliver Burk, Matthias Schwab, Renzo Wolbold, Peter Neuhaus, Michel Eichelbaum
المصدر: Hepatology. 38:978-988
مصطلحات موضوعية: Adult, Male, Drug, Receptors, Steroid, medicine.medical_specialty, media_common.quotation_subject, Receptors, Cytoplasmic and Nuclear, ATP-binding cassette transporter, Pharmacology, Sex Factors, Cytochrome P-450 Enzyme System, Internal medicine, Cytochrome P-450 CYP3A, medicine, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, RNA, Messenger, Receptor, Life Style, Constitutive Androstane Receptor, Aged, media_common, Pregnane X receptor, Hepatology, biology, CYP3A4, Pregnane X Receptor, Cytochrome P450, Middle Aged, Endocrinology, Liver, Verapamil, biology.protein, Female, Drug metabolism, Transcription Factors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2436915ecde8be75c9d5f021b7f3803bTest
https://doi.org/10.1002/hep.1840380424Test -
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المؤلفون: Peter Neuhaus, Kathrin Klein, Ulrich M. Zanger, Thomas E. Mürdter, Andreas K. Nussler, Janet K. Coller, Niels Krebsfaenger, Michel Eichelbaum, Renzo Wolbold
المصدر: British Journal of Clinical Pharmacology. 57:105-111
مصطلحات موضوعية: Pharmacology, biology, CYP3A4, Metabolite, Cytochrome P450, Antiestrogen, Isozyme, chemistry.chemical_compound, chemistry, medicine, biology.protein, Microsome, Pharmacology (medical), Troleandomycin, Tamoxifen, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::95dc15953869e1814871426e345d4a4bTest
https://doi.org/10.1046/j.1365-2125.2003.01970.xTest -
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المؤلفون: Julia Blievernicht, Ulrich M. Zanger, Jan G. Hengstler, Andreas K. Nussler, N Nussler, Matthias Schwab, Tanja Saussele, Kathrin Klein, Oliver Burk, Michel Eichelbaum
المصدر: Clinical pharmacology and therapeutics. 82(3)
مصطلحات موضوعية: Male, Receptors, Steroid, CYP2B6, Genotype, Blotting, Western, Dipyrone, Receptors, Cytoplasmic and Nuclear, Pharmacology, In Vitro Techniques, Catalysis, Cytochrome P-450 Enzyme System, Constitutive androstane receptor, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), Enzyme inducer, Cells, Cultured, Constitutive Androstane Receptor, Aged, Pregnane X receptor, biology, CYP3A4, Dose-Response Relationship, Drug, Chemistry, Reverse Transcriptase Polymerase Chain Reaction, Anti-Inflammatory Agents, Non-Steroidal, Pregnane X Receptor, Cytochrome P450 reductase, Oxidoreductases, N-Demethylating, DNA, Middle Aged, Metamizole, Isoenzymes, Cytochrome P-450 CYP2B6, Liver, Enzyme inhibitor, Enzyme Induction, biology.protein, Hepatocytes, Microsomes, Liver, RNA, Female, Aryl Hydrocarbon Hydroxylases, medicine.drug, Plasmids, Transcription Factors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f2732a57085a33507063701647d670fTest
https://pubmed.ncbi.nlm.nih.gov/17344806Test -
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المؤلفون: Kari T. Kivistö, Michel Eichelbaum, Karl Bodin, Mikko Niemi, Martin F. Fromm, Leif Bertilsson, Ulf Diczfalusy
المصدر: Karolinska Institutet
مصطلحات موضوعية: medicine.medical_specialty, ATP Binding Cassette Transporter, Subfamily B, Genotype, Organic Anion Transporters, Single-nucleotide polymorphism, Pharmacology, Cytochrome P-450 Enzyme System, Internal medicine, polycyclic compounds, Genetics, medicine, Cytochrome P-450 CYP3A, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, General Pharmacology, Toxicology and Pharmaceutics, Molecular Biology, Genetics (clinical), Antibacterial agent, Polymorphism, Genetic, biology, CYP3A4, Liver-Specific Organic Anion Transporter 1, Cytochrome P450, Hydroxycholesterols, Organic anion-transporting polypeptide, Endocrinology, Liver, Enzyme Induction, biology.protein, Molecular Medicine, Rifampin, SLCO1B1, Rifampicin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5313bd8a3a31d1de7bc93f990a49e9abTest
https://pubmed.ncbi.nlm.nih.gov/16847425Test -
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المؤلفون: Mitchell A. Avery, Oliver Burk, Andreas K. Nussler, Michel Eichelbaum, Elke Schaeffeler, Katja A. Arnold, Ekaterina Efimova, Bonnie A. Avery, Martin F. Fromm
المصدر: Molecular pharmacology. 67(6)
مصطلحات موضوعية: Receptors, Steroid, CYP2B6, Receptors, Cytoplasmic and Nuclear, Pharmacology, Cell Line, Antimalarials, Mice, Cytochrome P-450 Enzyme System, parasitic diseases, Constitutive androstane receptor, Chlorocebus aethiops, medicine, Animals, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Artemisinin, Receptor, Constitutive Androstane Receptor, Pregnane X receptor, biology, CYP3A4, Dose-Response Relationship, Drug, Pregnane X Receptor, Cytochrome P450, Artemisinins, Nuclear receptor, Gene Expression Regulation, Enzyme Induction, COS Cells, biology.protein, Hepatocytes, Molecular Medicine, Sesquiterpenes, medicine.drug, Transcription Factors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::10bca50b1ece1cda198358894228f9edTest
https://pubmed.ncbi.nlm.nih.gov/15761118Test -
8
المؤلفون: Ulrich M. Zanger, Ina Koch, Jürgen Brockmöller, Regina Weil, Renzo Wolbold, Oliver Burk, Peter Neuhaus, Andreas K. Nuessler, Leszek Wojnowski, Michel Eichelbaum, Elisabeth Hustert
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 30(10)
مصطلحات موضوعية: Pharmacology, Messenger RNA, biology, CYP3A4, CYP3A, Pharmaceutical Science, Cytochrome P450, Gene Expression, Genetic Variation, Molecular biology, Isozyme, Isoenzymes, Cytochrome P-450 Enzyme System, Liver, Organ Specificity, Gene expression, biology.protein, Cytochrome P-450 CYP3A, Humans, RNA, Messenger, Gene, CYP3A7
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::28d5b00b276088c2629c6ddaf3444bc9Test
https://pubmed.ncbi.nlm.nih.gov/12228187Test -
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المؤلفون: Heyo K. Kroemer, Michel Eichelbaum, Dagmar Busse, Martin F. Fromm
المصدر: Hepatology (Baltimore, Md.). 24(4)
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Administration, Oral, Biological Availability, Pharmacology, Pharmacokinetics, Oral administration, Internal medicine, medicine, Humans, Drug Interactions, Hepatology, CYP3A4, biology, Chemistry, Cytochrome P450, Stereoisomerism, Drug interaction, Bioavailability, Endocrinology, Liver, Verapamil, Enzyme Induction, Injections, Intravenous, biology.protein, Rifampin, Digestive System, Drug metabolism, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd04922015a5fa9d7b442e51a33b00c1Test
https://pubmed.ncbi.nlm.nih.gov/8855178Test -
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المؤلفون: Dagmar Busse, Jose Cosme, Philippe Beaune, HeyoK. Kroemer, Michel Eichelbaum, D. Busse, H.K. Kroemer, M. Eichelbaum
المصدر: Naunyn-Schmiedeberg's archives of pharmacology. 353(1)
مصطلحات موضوعية: Metabolite, Biology, Pharmacology, Sulfaphenazole, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, medicine, Humans, CYP3A4, CYP1A2, Cytochrome P450, Norverapamil, General Medicine, Calcium Channel Blockers, Isoenzymes, Kinetics, chemistry, Liver, Verapamil, Dealkylation, biology.protein, Microsome, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c1ec03472c21ba0a93780fa2afa8ceb5Test
https://pubmed.ncbi.nlm.nih.gov/8750925Test