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1
المؤلفون: Mirunalini Ravichandran, Subhiksha Subramanian
المصدر: Fundamental & Clinical Pharmacology. 36:72-80
مصطلحات موضوعية: Pharmacology, Nervous system, Orexins, Drug discovery, Neuropeptides, digestive, oral, and skin physiology, Optogenetics, Biology, Orexin receptor, Receptors, G-Protein-Coupled, medicine.anatomical_structure, nervous system, Orexin Receptors, Sleep Initiation and Maintenance Disorders, mental disorders, medicine, Drug approval, Humans, Pharmacology (medical), Receptor, Neuroscience, hormones, hormone substitutes, and hormone antagonists, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3940a00d6a047f0695b9a1c4ed9a95caTest
https://doi.org/10.1111/fcp.12723Test -
2
المؤلفون: Giorgio Bergamini, Michel A. Steiner, Catherine Roch, Martine Clozel
المصدر: Psychopharmacology
مصطلحات موضوعية: Pyrrolidines, Insomnia, Daridorexant, Allosteric regulation, Physical dependence, Review, Pharmacology, Doras, Nonclinical, Orexin Receptors, Sleep Initiation and Maintenance Disorders, Dual orexin receptor antagonist, medicine, Humans, Receptor, biology, Mechanism (biology), business.industry, Sleep architecture, Imidazoles, Antagonist, biology.organism_classification, Orexin receptor, Orexin, Orexin Receptor Antagonists, medicine.symptom, Sleep, business
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::98223dcb1d64e58042db5b10ea52358eTest
https://doi.org/10.1007/s00213-021-05954-0Test -
3
المؤلفون: Ann M. Decker, Catherine M. Kotz, Vijayakumar Mavanji, Tiffany L. Langston, Dehui Zhang, Yanan Zhang, Danni L. Harris, David A. Perrey
المصدر: J Med Chem
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, medicine.medical_treatment, Intraperitoneal injection, CHO Cells, Molecular Dynamics Simulation, Pharmacology, 01 natural sciences, Article, Mice, Structure-Activity Relationship, 03 medical and health sciences, Cricetulus, Orexin Receptors, Drug Discovery, medicine, Animals, Structure–activity relationship, Wakefulness, 030304 developmental biology, Sulfonamides, 0303 health sciences, Molecular Structure, biology, Chemistry, biology.organism_classification, medicine.disease, Small molecule, 0104 chemical sciences, Orexin, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Molecular Medicine, Female, Sleep, Narcolepsy
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::931ff980a0192e08e857b44e3b894b07Test
https://doi.org/10.1021/acs.jmedchem.1c00841Test -
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المؤلفون: Hitoshi Takahashi, Shunpei Moriya, Jun Ishigooka, Katsuji Nishimura, Makiko Yamada, Daiki Masukawa
المصدر: Journal of Pharmacological Sciences, Vol 145, Iss 2, Pp 198-201 (2021)
مصطلحات موضوعية: Male, 0301 basic medicine, medicine.medical_specialty, Noradrenalin transporter (Net), Gene Expression, Hippocampus, Biology, 03 medical and health sciences, 0302 clinical medicine, Dorsal raphe nucleus, Internal medicine, medicine, Animals, RNA, Messenger, Monoamine Oxidase, Dual orexin receptor antagonist (DORA), Pharmacology, Regulation of gene expression, Norepinephrine Plasma Membrane Transport Proteins, lcsh:RM1-950, Antagonist, Azepines, Orexin receptor, Orexin, Mice, Inbred C57BL, 030104 developmental biology, Monoamine neurotransmitter, Endocrinology, lcsh:Therapeutics. Pharmacology, Gene Expression Regulation, Molecular Medicine, Locus coeruleus, Benzimidazoles, Orexin Receptor Antagonists, 030217 neurology & neurosurgery
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e040ef606236d0a7f4ff3e0dba139ceTest
http://www.sciencedirect.com/science/article/pii/S1347861320301225Test -
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المؤلفون: Duffet, Loic, Tatarskiy, Petr V, Harada, Masaya, Williams, Elyse T, Hartrampf, Nina, Patriarchi, Tommaso
المساهمون: University of Zurich
المصدر: Cell Chemical Biology, 29 (12)
مصطلحات موضوعية: Pharmacology, Orexin-B, Neuropeptides, Photocage, G protein-coupled receptor, Genetically encoded sensors, Biosensor, Clinical Biochemistry, 10050 Institute of Pharmacology and Toxicology, 610 Medicine & health, Biochemistry, Drug Discovery, 570 Life sciences, biology, Molecular Medicine, Molecular Biology
وصف الملف: application/application/pdf; ZORA_pdf.pdf - application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::660fde800848fdd970de55ebf84199e8Test
https://pubmed.ncbi.nlm.nih.gov/36481097Test -
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المؤلفون: Yijia Cao, Tiange Yang, Yu Sun, Chenning Zhang, Yuxia Qu, Yikun Sun, Shiting Ni, Tianyi Li, Hao Wu, Renyun Zhao, Runhua Liu
المصدر: ACS Omega, Vol 6, Iss 13, Pp 9176-9187 (2021)
مصطلحات موضوعية: Honokiol, biology, GABAA receptor, General Chemical Engineering, Homovanillic acid, General Chemistry, Pharmacology, biology.organism_classification, Magnolol, Orexin receptor, Chemistry, chemistry.chemical_compound, Monoamine neurotransmitter, chemistry, Melanogaster, Drosophila melanogaster, QD1-999
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8d648d43aeeef00e9a0f26d77d793ebbTest
https://doi.org/10.1021/acsomega.1c00445Test -
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المصدر: Neuropsychopharmacology
مصطلحات موضوعية: Lateral hypothalamus, Biology, Article, Small hairpin RNA, Cocaine, Orexin Receptors, mental disorders, medicine, Animals, Receptor, Sensory cue, Pharmacology, Orexins, digestive, oral, and skin physiology, Ventral Tegmental Area, Antagonist, Receptor signaling, Orexin, Ventral tegmental area, Psychiatry and Mental health, medicine.anatomical_structure, nervous system, Hypothalamic Area, Lateral, Cues, Neuroscience, psychological phenomena and processes
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bb54b1dd103776b23b4a2105095711a1Test
https://europepmc.org/articles/PMC8782853Test/ -
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المصدر: Current Neuropharmacology
مصطلحات موضوعية: 0301 basic medicine, Central nervous system, CX3C Chemokine Receptor 1, Biology, Article, 03 medical and health sciences, 0302 clinical medicine, Antigens, CD, Orexin Receptors, CX3CR1, medicine, Animals, Humans, Pharmacology (medical), Receptor, CX3CL1, Pharmacology, Neurons, Brain Diseases, Cluster of differentiation, Microglia, Chemokine CX3CL1, Neurodegeneration, Brain, General Medicine, medicine.disease, Psychiatry and Mental health, 030104 developmental biology, medicine.anatomical_structure, Neurology, nervous system, CX3CL1-CX3CR1, depression, Schizophrenia, Parkinson’s disease, Neurology (clinical), Neuron, Chemokines, Neuroscience, Alzheimer’s disease, 030217 neurology & neurosurgery, CD200-CD200R
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c65888a4b5e1268af0bcc8acd6f9e63cTest
http://europepmc.org/articles/PMC7457436Test -
9
المؤلفون: Qiaochu Cheng, Yaguang Hu, Shan Gao, Ting Wei
المصدر: Inflammation Research. 68:945-955
مصطلحات موضوعية: Vascular Endothelial Growth Factor A, 0301 basic medicine, medicine.medical_treatment, Immunology, Becaplermin, Retinal Neovascularization, Retina, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Western blot, Antigens, CD, Orexin Receptors, medicine, Animals, Receptor, Pharmacology, Hyperoxia, medicine.diagnostic_test, biology, Microglia, Growth factor, Endothelial Cells, Retinal, Molecular biology, eye diseases, Mice, Inbred C57BL, Oxygen, Vitreous Body, Vascular endothelial growth factor, Disease Models, Animal, 030104 developmental biology, medicine.anatomical_structure, chemistry, 030220 oncology & carcinogenesis, biology.protein, Cytokines, sense organs, medicine.symptom, Platelet-derived growth factor receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9dd410bd6d87b791ab192c073a2c9e6cTest
https://doi.org/10.1007/s00011-019-01276-2Test -
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المؤلفون: Patrick M. Fuller, Melissa J. Chee, Elda Arrigoni
المصدر: Neuropharmacology. 154:34-49
مصطلحات موضوعية: 0301 basic medicine, Lateral hypothalamus, Melanin-concentrating hormone, Biology, Non-rapid eye movement sleep, Energy homeostasis, Arousal, Eating, 03 medical and health sciences, Cellular and Molecular Neuroscience, chemistry.chemical_compound, 0302 clinical medicine, Neural Pathways, Animals, Humans, Wakefulness, Pharmacology, Orexins, Orexin, 030104 developmental biology, chemistry, Hypothalamic Area, Lateral, GABAergic, Energy Metabolism, Sleep, Neuroscience, 030217 neurology & neurosurgery, Homeostasis
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::11359dcc3883d19f7eba4fc991425f35Test
https://doi.org/10.1016/j.neuropharm.2018.11.017Test