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المؤلفون: Peter Orth, Bandarpalle B. Shankar, Daniel Lundell, Corey O. Strickland, Vinay Girijavallabhan, Chaoyang Dai, Joseph A. Kozlowski, Janeta Popovici-Muller, Brian J. Lavey, Jing Sun, Shiying Chen, Dansu Li, John J. Piwinski, Razia Rizvi, M. Arshad Siddiqui, Kristin E. Rosner, Lianyun Zhao, Zhuyan Guo, Wong Michael K C, Neng-Yang Shih, Xiaoda Niu
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3172-3176
مصطلحات موضوعية: Pyrrolidines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Carboxamide, ADAM17 Protein, Tartrate, Biochemistry, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Oral administration, Amide, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Tartrates, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, Amides, Rats, Enzyme Activation, ADAM Proteins, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5ffe3fdf02a5dba0580b311b55f7fe2Test
https://doi.org/10.1016/j.bmcl.2011.01.002Test -
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المؤلفون: Bandarpalle B. Shankar, Ling Tong, Himanshu Shah, Wensheng Yu, Jing Sun, De-Yi Yang, Guowei Zhou, Lei Chen, Feltz Robert, Kristin E. Rosner, Xiaoda Niu, Neng-Yang Shih, Shelby Umland, Zhuyan Guo, John J. Piwinski, Seong Heon Kim, Dansu Li, Razia Rizvi, Peter Orth, Aneta Kosinski, Wong Michael K C, Joseph A. Kozlowski, Daniel Lundell, M. Arshad Siddiqui, Brian J. Lavey
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5286-5289
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Hydantoin, ADAM17 Protein, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Hydrolase, Animals, Structure–activity relationship, Enzyme Inhibitors, Molecular Biology, biology, Organic Chemistry, Active site, Biological activity, Rats, ADAM Proteins, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Selectivity
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0544f42865077bfcb9c1747073ba2311Test
https://doi.org/10.1016/j.bmcl.2010.06.134Test -
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المؤلفون: Gopinadhan N. Anilkumar, Qingbei Zeng, Brian F. Mcguinness, Chung-Her Jenh, Guizhen Dong, Lisa Guise Zawacki, Inna Schulman, Yueheng Jiang, Seong Heon Kim, Yuefei Shao, Youheng Shu, Wong Michael K C, Doug W. Hobbs, Stuart B. Rosenblum, Neng-Yang Shih, James W. Hall, Carolyn DiIanni Carroll, Wensheng Yu, Joseph A. Kozlowski
المصدر: Bioorganicmedicinal chemistry letters. 21(5)
مصطلحات موضوعية: Receptors, CXCR3, Stereochemistry, medicine.drug_class, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CXCR3, Biochemistry, Piperazines, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, stomatognathic system, Piperidines, immune system diseases, Drug Discovery, medicine, Moiety, Humans, skin and connective tissue diseases, Receptor, Molecular Biology, IC50, Piperazine, Molecular Structure, Organic Chemistry, Antagonist, hemic and immune systems, In vitro, stomatognathic diseases, chemistry, Molecular Medicine, Piperidine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9894b320a60ce2053010ea1122688132Test
https://pubmed.ncbi.nlm.nih.gov/21277198Test -
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المؤلفون: Feltz Robert, Kristin E. Rosner, De-Yi Yang, Janeta Popovici-Muller, Daniel Lundell, M. Arshad Siddiqui, Peter Orth, John J. Piwinski, Bandarpalle B. Shankar, Shelby Umland, Guowei Zhou, Zhuyan Guo, Ling Tong, Vincent S. Madison, Razia Rizvi, Xiaoda Niu, Neng-Yang Shih, Chaoyang Dai, Joseph A. Kozlowski, Wong Michael K C, Seong Heon Kim, Dansu Li, Jing Sun, Vinay Girijavallabhan, Lei Chen, Brian J. Lavey, Wensheng Yu
المصدر: Bioorganicmedicinal chemistry letters. 20(6)
مصطلحات موضوعية: Models, Molecular, Denticity, Zinc binding, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, chemistry.chemical_element, Hydantoin, Zinc, ADAM17 Protein, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, X-Ray Diffraction, Drug Discovery, Structure–activity relationship, Moiety, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Ligand, Hydantoins, Organic Chemistry, Hydrogen Bonding, ADAM Proteins, Enzyme, chemistry, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f39d5f4051d8a87a9707d21fbe52849Test
https://pubmed.ncbi.nlm.nih.gov/20172725Test -
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المؤلفون: Len Favreau, Chunli Huang, Guowei Zhou, Neng-Yang Shih, Waldemar Gonsiorek, R. William Hipkin, Charles A. Lunn, Ling Tong, Joseph A. Kozlowski, Joseph Kelly, Lei Chen, Brian J. Lavey, Asra Malikzay, Razia Rizvi, Eric J. Gilbert, Bandarpalle B. Shankar, Daniel Lundell, Wong Michael K C, Stuart W. McCombie, Youhao Dong, Youheng Shu
المصدر: Bioorganicmedicinal chemistry letters. 20(2)
مصطلحات موضوعية: Drug Inverse Agonism, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ring (chemistry), Biochemistry, Chemical synthesis, Sulfone, Receptor, Cannabinoid, CB2, chemistry.chemical_compound, Structure-Activity Relationship, Cytochrome P-450 Enzyme System, Piperidines, Drug Discovery, Moiety, Structure–activity relationship, Animals, Humans, Sulfones, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Aryl, Organic Chemistry, Sulfonamide, Rats, chemistry, Molecular Medicine, Piperidine, Calcium Channels
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dbdfe23991c9196dd275858b3d1c234Test
https://pubmed.ncbi.nlm.nih.gov/20005710Test