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المؤلفون: Peter Orth, Bandarpalle B. Shankar, Daniel Lundell, Corey O. Strickland, Vinay Girijavallabhan, Chaoyang Dai, Joseph A. Kozlowski, Janeta Popovici-Muller, Brian J. Lavey, Jing Sun, Shiying Chen, Dansu Li, John J. Piwinski, Razia Rizvi, M. Arshad Siddiqui, Kristin E. Rosner, Lianyun Zhao, Zhuyan Guo, Wong Michael K C, Neng-Yang Shih, Xiaoda Niu
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3172-3176
مصطلحات موضوعية: Pyrrolidines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Carboxamide, ADAM17 Protein, Tartrate, Biochemistry, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Oral administration, Amide, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Tartrates, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, Amides, Rats, Enzyme Activation, ADAM Proteins, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5ffe3fdf02a5dba0580b311b55f7fe2Test
https://doi.org/10.1016/j.bmcl.2011.01.002Test -
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المؤلفون: Liping Yang, Shelby Umland, Peter Orth, Daniel Lundell, Luke Firmansjah, Feltz Robert, Chaoyang Dai, Joseph A. Kozlowski, Wensheng Yu, Janeta Popovici-Muller, Seong Heon Kim, Vincent S. Madison, John J. Piwinski, De-Yi Yang, M. Arshad Siddiqui, Ling Tong, Xiaoda Niu, Brian J. Lavey, Guowei Zhou, Banderpalle B. Shankar, Razia Rizvi, Kristin E. Rosner, Neng-Yang Shih, Aneta Kosinski, Hong Bian, Dansu Li, Vinay Girijavallabhan, Lei Chen, Himanshu Shah, Zhuyan Guo, Jing Sun, Wong Michael K C
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:7283-7287
مصطلحات موضوعية: medicine.medical_treatment, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Hydantoin, ADAM17 Protein, Pharmacology, Biochemistry, Arthritis, Rheumatoid, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Humans, Protease Inhibitors, Molecular Biology, Whole blood, chemistry.chemical_classification, biology, Acetylene, Organic Chemistry, Biological activity, Haplorhini, In vitro, Rats, ADAM Proteins, Cytokine, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Tumor necrosis factor alpha
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1f13e3eb17b7abab77da7bd68ad794d7Test
https://doi.org/10.1016/j.bmcl.2010.10.081Test -
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المؤلفون: Gopinadhan N. Anilkumar, Qingbei Zeng, Brian F. Mcguinness, Chung-Her Jenh, Guizhen Dong, Lisa Guise Zawacki, Inna Schulman, Yueheng Jiang, Seong Heon Kim, Yuefei Shao, Youheng Shu, Wong Michael K C, Doug W. Hobbs, Stuart B. Rosenblum, Neng-Yang Shih, James W. Hall, Carolyn DiIanni Carroll, Wensheng Yu, Joseph A. Kozlowski
المصدر: Bioorganicmedicinal chemistry letters. 21(5)
مصطلحات موضوعية: Receptors, CXCR3, Stereochemistry, medicine.drug_class, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CXCR3, Biochemistry, Piperazines, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, stomatognathic system, Piperidines, immune system diseases, Drug Discovery, medicine, Moiety, Humans, skin and connective tissue diseases, Receptor, Molecular Biology, IC50, Piperazine, Molecular Structure, Organic Chemistry, Antagonist, hemic and immune systems, In vitro, stomatognathic diseases, chemistry, Molecular Medicine, Piperidine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9894b320a60ce2053010ea1122688132Test
https://pubmed.ncbi.nlm.nih.gov/21277198Test