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1دورية أكاديمية
المؤلفون: Fish, Inbar, Stößel, Anne, Eitel, Katrin, Valant, Celine, Albold, Sabine, Huebner, Harald, Möller, Dorothee, Clark, Mary J, Sunahara, Roger K, Christopoulos, Arthur, Shoichet, Brian K, Gmeiner, Peter
المصدر: Journal of medicinal chemistry. 60(22)
مصطلحات موضوعية: CHO Cells, Animals, Humans, Cricetulus, Tritium, Carbachol, Acetylcholine, N-Methylscopolamine, Isoxazoles, Benzofurans, Arrestin, Receptor, Muscarinic M1, Receptor, Muscarinic M2, Receptor, Muscarinic M3, Receptors, Nicotinic, Muscarinic Agonists, Ligands, Drug Design, Quaternary Ammonium Compounds, HEK293 Cells, Molecular Docking Simulation, Brain Disorders, Medicinal and Biomolecular Chemistry, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/7fq8g9h3Test
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المؤلفون: Regan Ashby, Kate Thomson, Cindy Karouta, Ian G. Morgan, Tamsin Kelly
المصدر: British Journal of Pharmacology. 178:4501-4517
مصطلحات موضوعية: Atropine, Pharmacology, Muscarine, Carbachol, business.industry, Dopamine, Muscarinic Antagonists, Retina, eye diseases, chemistry.chemical_compound, Nicotinic agonist, chemistry, Muscarinic acetylcholine receptor, Myopia, medicine, Oxotremorine, Animals, Humans, Cholinergic, business, Chickens, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0608bf04ae7997074fe34b0eebfe111cTest
https://doi.org/10.1111/bph.15629Test -
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المؤلفون: Barbara Rinaldi, Clive P. Page, Luigino Calzetta, Mario Cazzola, Maria Gabriella Matera, Paola Rogliani
المساهمون: Calzetta, L, Rogliani, P, Page, C, Rinaldi, B, Cazzola, M, Matera, Mg.
المصدر: Pulmonary Pharmacology & Therapeutics. 56:39-50
مصطلحات موضوعية: Male, Pulmonary and Respiratory Medicine, Carbachol, Human airways, Settore MED/10 - Malattie dell'Apparato Respiratorio, Bronchi, Muscarinic Antagonists, Pharmacology, Contractility, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Muscarinic acetylcholine receptor, medicine, Humans, Pharmacology (medical), 030212 general & internal medicine, Adrenergic beta-2 Receptor Agonists, Aged, Papaverine, Chemistry, Biochemistry (medical), Olodaterol, Muscarinic antagonist, Drug Synergism, Muscle, Smooth, Tiotropium bromide, Middle Aged, respiratory system, Synergy, Benzoxazines, Bronchodilator Agents, respiratory tract diseases, Drug Combinations, 030228 respiratory system, Female, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ae195d11e32e592f59799d7c1b1ae388Test
https://doi.org/10.1016/j.pupt.2019.03.004Test -
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المؤلفون: Subhash Kulkarni, Jianyi Yin, Chung Ming Tse, Pankaj J. Pasricha, Julie G. In, Mark Donowitz, Kelli Johnson
المصدر: Am J Physiol Cell Physiol
مصطلحات موضوعية: 0301 basic medicine, Anions, Atropine, Carbachol, Physiology, Bethanechol, Cholinergic Agonists, Muscarinic Agonists, Receptors, Nicotinic, Muscarinic agonist, Hexamethonium, 03 medical and health sciences, chemistry.chemical_compound, Mice, 0302 clinical medicine, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Nicotinic Antagonist, Intestinal Mucosa, Non-Neuronal Cholinergic System, Cell Biology, Receptors, Muscarinic, Acetylcholine, Cell biology, Intestines, 030104 developmental biology, Nicotinic agonist, Enterocytes, chemistry, 030220 oncology & carcinogenesis, medicine.drug, Research Article
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b93a8a7357d83e58f4513a8870962fbeTest
https://pubmed.ncbi.nlm.nih.gov/32551856Test -
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المؤلفون: María Elena Sales, Francisco Sánchez, P. Martínez Pulido, Y. Sanchez, A.R. Salem, Alejandro J. Español
المصدر: International immunopharmacology. 84
مصطلحات موضوعية: 0301 basic medicine, Carbachol, Paclitaxel, Angiogenesis, Cell Survival, Immunology, Mice, Nude, Cholinergic Agonists, Muscarinic agonist, Cell Line, 03 medical and health sciences, 0302 clinical medicine, Mammary Glands, Animal, Cancer stem cell, Muscarinic acetylcholine receptor, medicine, Immunology and Allergy, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Humans, Drug Interactions, Cell Proliferation, Pharmacology, Neovascularization, Pathologic, Chemistry, Mammary Neoplasms, Experimental, Antineoplastic Agents, Phytogenic, Receptors, Muscarinic, 030104 developmental biology, Nicotinic agonist, 030220 oncology & carcinogenesis, Administration, Metronomic, Cancer research, Cholinergic, Female, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ddfc55e090dd2ebb3c1535dff61dcd2dTest
https://pubmed.ncbi.nlm.nih.gov/32591266Test -
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المؤلفون: Asheebo Rojas, Alec Walker, Thota Ganesh, Raymond Dingledine
المصدر: ACS Chemical Neuroscience. 8:712-717
مصطلحات موضوعية: Male, 0301 basic medicine, Patch-Clamp Techniques, Carbachol, Physiology, Cost effectiveness, Cognitive Neuroscience, Muscarinic Antagonists, Muscarinic Agonists, Pharmacology, Biochemistry, Article, Methylatropine, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Bromide, medicine, Animals, Humans, Atropine Derivatives, Pilocarpine, Muscarinic antagonist, Cell Biology, General Medicine, Mice, Inbred C57BL, Disease Models, Animal, Atropine, 030104 developmental biology, chemistry, 030217 neurology & neurosurgery, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::77a4b08c501a8c4cda69e84c81c19d85Test
https://doi.org/10.1021/acschemneuro.6b00334Test -
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المؤلفون: Hongwei Li, Philipp Risel, Shoji Maeda, Harald Hübner, Brian K. Kobilka, Jonas Kaindl, Changwen Jin, Xiaogang Niu, Yunfei Hu, Peter Gmeiner, Jun Xu
المصدر: Molecular cell. 75(1)
مصطلحات موضوعية: Protein Conformation, alpha-Helical, Magnetic Resonance Spectroscopy, Pyridines, Allosteric regulation, Genetic Vectors, Gene Expression, Biology, Molecular Dynamics Simulation, Spodoptera, Ligands, 03 medical and health sciences, 0302 clinical medicine, Muscarinic acetylcholine receptor, Thiadiazoles, Arrestin, Sf9 Cells, Animals, Humans, Protein Interaction Domains and Motifs, Cloning, Molecular, Receptor, Molecular Biology, 030304 developmental biology, G protein-coupled receptor, 0303 health sciences, Receptor, Muscarinic M2, Binding Sites, Pilocarpine, Cell Biology, Nuclear magnetic resonance spectroscopy, Isoxazoles, Ligand (biochemistry), Transmembrane protein, Acetylcholine, Recombinant Proteins, Quaternary Ammonium Compounds, Kinetics, Biophysics, Thermodynamics, Carbachol, Protein Conformation, beta-Strand, Baculoviridae, 030217 neurology & neurosurgery, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::01fc3cac70fdf8f2cac7dce55b1d8dd0Test
https://pubmed.ncbi.nlm.nih.gov/31103421Test -
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المؤلفون: Hülya Cabadak, Banu Aydın
المصدر: Journal of receptor and signal transduction research. 40(1)
مصطلحات موضوعية: 0301 basic medicine, Cell physiology, Carbachol, Cholinergic Agents, Cholinergic Agonists, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Erythroid Cells, Muscarinic acetylcholine receptor, medicine, Humans, Receptors, Cholinergic, Molecular Biology, Caspase, Cell Proliferation, biology, Cell Differentiation, Cell Biology, Cell biology, Enzyme Activation, 030104 developmental biology, chemistry, Apoptosis, 030220 oncology & carcinogenesis, Caspases, biology.protein, Cholinergic, Hemin, K562 Cells, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8232d311a7906b59d531326cfbb46738Test
https://pubmed.ncbi.nlm.nih.gov/31910706Test -
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المؤلفون: Martin Diener, O. S. Ilyaskina, Moritz Bünemann, F. Machka, Ervice Pouokam, Mathias S. Wickleder, A. Mattern
المصدر: Organic & Biomolecular Chemistry. 16:6680-6687
مصطلحات موضوعية: Agonist, medicine.drug_class, Metal Nanoparticles, 02 engineering and technology, Ligands, 010402 general chemistry, 01 natural sciences, Biochemistry, chemistry.chemical_compound, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Receptors, Cholinergic, Physical and Theoretical Chemistry, Receptor, Chemistry, Ligand, Organic Chemistry, Long-term potentiation, 021001 nanoscience & nanotechnology, Rats, 0104 chemical sciences, HEK293 Cells, Biophysics, Cholinergic, Carbachol, Hexamethonium, Gold, 0210 nano-technology, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2f869155de6454e7fc90f316ebb78ad7Test
https://doi.org/10.1039/c8ob01686kTest -
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المؤلفون: Deborah L. Smith, Sarah J. Neal, Lei Zhang, Jeremy R. Edgerton, Jennifer E. Davoren, Sarah Grimwood, John T. Lazzaro, Chewah Lee
المصدر: Molecular Pharmacology. 90:177-187
مصطلحات موضوعية: Male, 0301 basic medicine, Carbachol, Allosteric modulator, Pyridines, Stereochemistry, Allosteric regulation, CHO Cells, Isoindoles, Hippocampus, Rats, Sprague-Dawley, Radioligand Assay, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Allosteric Regulation, Cricetinae, Muscarinic acetylcholine receptor, medicine, Radioligand, Animals, Humans, Fluorometry, Pharmacology, Membranes, Chemistry, Ligand binding assay, Receptor, Muscarinic M1, N-Methylscopolamine, Acetylcholine, Electrophysiological Phenomena, Kinetics, HEK293 Cells, 030104 developmental biology, Positron-Emission Tomography, Autoradiography, Molecular Medicine, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59a4cbb153c3abcd01cb4427f9543370Test
https://doi.org/10.1124/mol.116.104737Test