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المؤلفون: Katherine Fenner, Abhishek Srivastava, Beth Williamson, Andrew Pike
المصدر: Journal of Pharmaceutical Sciences. 110:1412-1417
مصطلحات موضوعية: Pharmaceutical Science, Excipient, 02 engineering and technology, 030226 pharmacology & pharmacy, Dialysis tubing, 03 medical and health sciences, 0302 clinical medicine, Renal Dialysis, medicine, Humans, Drug Interactions, Equilibrium dialysis, Solubility, ADME, Chromatography, Chemistry, Blood Proteins, 021001 nanoscience & nanotechnology, Pharmaceutical Preparations, Free fraction, Lipophilicity, Lipinski's rule of five, 0210 nano-technology, Dialysis, Protein Binding, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::74ce67d843a0379d03045dc1f7d6ae4bTest
https://doi.org/10.1016/j.xphs.2020.11.018Test -
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المؤلفون: Dermot F. McGinnity, Beth Williamson, Stephanie Harlfinger
المصدر: Drug Metabolism and Disposition. 48:1137-1146
مصطلحات موضوعية: Male, Drug Evaluation, Preclinical, Extrapolation, Datasets as Topic, Pharmaceutical Science, Pharmacology, Models, Biological, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, medicine, Cytochrome P-450 CYP3A, Humans, In vitro in vivo, Human liver, Chemistry, Target engagement, Recombinant Proteins, Hepatobiliary Elimination, medicine.anatomical_structure, Liver, 030220 oncology & carcinogenesis, Hepatocyte, Hepatocytes, Microsomes, Liver, Microsome, Female, Drug metabolism, Oral retinoid
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::77ee63503e9e698986d5025960432a99Test
https://doi.org/10.1124/dmd.120.000131Test -
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المؤلفون: S A Foley, Robert J. Riley, Matthew G. Soars, Beth Williamson, P Barton
المصدر: Expert Opinion on Drug Metabolism & Toxicology. 12:201-216
مصطلحات موضوعية: Drug, media_common.quotation_subject, Pharmacology, Toxicology, Bioinformatics, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, Animals, Humans, Medicine, Drug Interactions, Pharmacokinetics, media_common, business.industry, Drug discovery, Membrane Transport Proteins, Biological Transport, Transporter, General Medicine, Liver, Pharmaceutical Preparations, Drug Design, 030220 oncology & carcinogenesis, business
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5adede26936155a26e5bd682b90e295eTest
https://doi.org/10.1517/17425255.2016.1132308Test -
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المؤلفون: Beth Williamson, Patrick Barton, Paul Lancett, Robert J. Riley
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(8)
مصطلحات موضوعية: 0301 basic medicine, Metabolic Clearance Rate, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Cytochrome P-450 Enzyme System, In vivo, Drug Discovery, Potency, Distribution (pharmacology), Humans, RNA, Messenger, Glucuronosyltransferase, Cells, Cultured, biology, Chemistry, Drug discovery, Cytochrome P450, In vitro, Kinetics, 030104 developmental biology, Liver, Toxicity, biology.protein, Hepatocytes, Biological Assay
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f5077201af61743cce7568418f21778Test
https://pubmed.ncbi.nlm.nih.gov/29880630Test -
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المؤلفون: Beth Williamson, Robert J. Riley
المصدر: Expert opinion on drug metabolismtoxicology. 13(12)
مصطلحات موضوعية: 0301 basic medicine, Drug, Exploit, Computer science, media_common.quotation_subject, Toxicology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, 0302 clinical medicine, Humans, Drug Interactions, Risk management, media_common, ADME, Pharmacology, Risk Management, business.industry, Membrane Transport Proteins, Reproducibility of Results, Biological Transport, General Medicine, Disposition, Drug transporter, 030104 developmental biology, Drug development, Risk analysis (engineering), Liver, Drug Design, business, Absorption rate constant
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c5e9eab783ac77f6bdfe098087efb9c1Test
https://pubmed.ncbi.nlm.nih.gov/29121476Test -
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المؤلفون: Timothy G. Brayman, Michael D. Mitchell, Mathias Lorbeer, Beth Williamson, Robert J. Riley
المصدر: Pharmacology Research & Perspectives
مصطلحات موضوعية: 0301 basic medicine, Agonist, CYP2B6, medicine.drug_class, knockout, Pharmacology, Biology, 030226 pharmacology & pharmacy, digestive system, 03 medical and health sciences, 0302 clinical medicine, Constitutive androstane receptor, medicine, General Pharmacology, Toxicology and Pharmaceutics, induction, Regulation of gene expression, Pregnane X receptor, DDIs, CYP3A4, Original Articles, digestive system diseases, Cell biology, 030104 developmental biology, Neurology, Nuclear receptor, Cell culture, Original Article, human PXR
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62f8602e6f25d24eb417cbf00ce0c558Test
http://europepmc.org/articles/PMC5045942Test