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المصدر: Drug Discovery Today. 25:1793-1800
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Mechanism (biology), business.industry, Administration, Oral, Proteins, Computational biology, 03 medical and health sciences, Drug Delivery Systems, 030104 developmental biology, 0302 clinical medicine, Pharmaceutical Preparations, Pharmacokinetics, 030220 oncology & carcinogenesis, Proteolysis, Drug Discovery, Humans, Medicine, business, Oral retinoid, Drug metabolism
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::386b90be2147c5934da0dd545cc49b03Test
https://doi.org/10.1016/j.drudis.2020.07.013Test -
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المؤلفون: Beth Williamson, Patrick Barton, Paul Lancett, Robert J. Riley
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(8)
مصطلحات موضوعية: 0301 basic medicine, Metabolic Clearance Rate, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Cytochrome P-450 Enzyme System, In vivo, Drug Discovery, Potency, Distribution (pharmacology), Humans, RNA, Messenger, Glucuronosyltransferase, Cells, Cultured, biology, Chemistry, Drug discovery, Cytochrome P450, In vitro, Kinetics, 030104 developmental biology, Liver, Toxicity, biology.protein, Hepatocytes, Biological Assay
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f5077201af61743cce7568418f21778Test
https://pubmed.ncbi.nlm.nih.gov/29880630Test -
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المؤلفون: Beth Williamson, Robert J. Riley
المصدر: Expert opinion on drug metabolismtoxicology. 13(12)
مصطلحات موضوعية: 0301 basic medicine, Drug, Exploit, Computer science, media_common.quotation_subject, Toxicology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, 0302 clinical medicine, Humans, Drug Interactions, Risk management, media_common, ADME, Pharmacology, Risk Management, business.industry, Membrane Transport Proteins, Reproducibility of Results, Biological Transport, General Medicine, Disposition, Drug transporter, 030104 developmental biology, Drug development, Risk analysis (engineering), Liver, Drug Design, business, Absorption rate constant
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c5e9eab783ac77f6bdfe098087efb9c1Test
https://pubmed.ncbi.nlm.nih.gov/29121476Test -
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المؤلفون: Claire E. Wilson, Robert J. Riley, Gayle Dagnell, Beth Williamson
المصدر: Journal of pharmacological and toxicological methods. 84
مصطلحات موضوعية: 0301 basic medicine, Computational biology, Pharmacology, Toxicology, Rats, Sprague-Dawley, 03 medical and health sciences, Mice, Pharmacokinetics, Species Specificity, In vivo, High-Throughput Screening Assays, Animals, Humans, Rats, Wistar, ADME, Chemistry, Drug discovery, In vitro toxicology, In vitro, Rats, Mice, Inbred C57BL, 030104 developmental biology, Microsome, Microsomes, Liver
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f96ab9338e673b89673a450ff1fa4f5Test
https://pubmed.ncbi.nlm.nih.gov/27773845Test -
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المؤلفون: Timothy G. Brayman, Michael D. Mitchell, Mathias Lorbeer, Beth Williamson, Robert J. Riley
المصدر: Pharmacology Research & Perspectives
مصطلحات موضوعية: 0301 basic medicine, Agonist, CYP2B6, medicine.drug_class, knockout, Pharmacology, Biology, 030226 pharmacology & pharmacy, digestive system, 03 medical and health sciences, 0302 clinical medicine, Constitutive androstane receptor, medicine, General Pharmacology, Toxicology and Pharmaceutics, induction, Regulation of gene expression, Pregnane X receptor, DDIs, CYP3A4, Original Articles, digestive system diseases, Cell biology, 030104 developmental biology, Neurology, Nuclear receptor, Cell culture, Original Article, human PXR
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62f8602e6f25d24eb417cbf00ce0c558Test
http://europepmc.org/articles/PMC5045942Test