نتائج البحث - "ALLOSTERIC MODULATION"

1

Identification of Koumine as a Translocator Protein 18 kDa Positive Allosteric Modulator for the Treatment of Inflammatory and Neuropathic Pain

المؤلفون: Bojun Xiong, Guilin Jin, Ying Xu, Wenbing You, Yufei Luo, Menghan Fang, Bing Chen, Huihui Huang, Jian Yang, Xu Lin, Changxi Yu

المصدر: Frontiers in Pharmacology
Frontiers in Pharmacology, Vol 12 (2021)

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a3746e11607f3cd837400de72fd841c8Test
http://europepmc.org/articles/PMC8264504Test

2

It takes two—or more—to tango: Revisiting the role of dopamine transporter oligomerization

المؤلفون: Harald H. Sitte, Ulrik Gether

المصدر: The Journal of Biological Chemistry
Gether, U & Sitte, H H 2021, ' It takes two-or more-to tango : Revisiting the role of dopamine transporter oligomerization ', Journal of Biological Chemistry, vol. 296, 100629 . https://doi.org/10.1016/j.jbc.2021.100629Test

مصطلحات موضوعية: 0301 basic medicine, monoamine transporters, Allosteric regulation, AL, AIM-100-like compound, Endocytosis, Biochemistry, Reuptake, oligomerization, 03 medical and health sciences, Editors' Pick Highlight, Dopamine, DAT, dopamine transporter, medicine, Animals, Humans, endocytosis, Neurotransmitter sodium symporter, Molecular Biology, dopamine transporter, Dopamine transporter, Dopamine Plasma Membrane Transport Proteins, dimerization, allosteric modulation, 030102 biochemistry & molecular biology, biology, Chemistry, Transporter, Cell Biology, SERT, serotonin, Transmembrane protein, 030104 developmental biology, NET, norepinephrine, biology.protein, Biophysics, NSS, neurotransmitter:sodium symporter, Protein Multimerization, medicine.drug, TM, transmembrane

وصف الملف: application/pdf

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::02dbc05ec5cee35576bc25e4aa4af8cdTest
http://europepmc.org/articles/PMC8100069Test

3

Allosteric Modulation of GPCRs of Class A by Cholesterol

المؤلفون: Jan Jakubík, Esam E. El-Fakahany

المصدر: International Journal of Molecular Sciences
International Journal of Molecular Sciences, Vol 22, Iss 1953, p 1953 (2021)

مصطلحات موضوعية: 0301 basic medicine, Allosteric regulation, Review, Ligands, Catalysis, GPCRs, Receptors, G-Protein-Coupled, Inorganic Chemistry, lcsh:Chemistry, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Allosteric Regulation, Animals, Humans, Molecular Targeted Therapy, Physical and Theoretical Chemistry, Binding site, Receptor, Molecular Biology, lcsh:QH301-705.5, Spectroscopy, G protein-coupled receptor, Binding Sites, allosteric modulation, Cholesterol, allergology, Anticholesteremic Agents, Organic Chemistry, Cholesterol binding, Cell Membrane, cholesterol, General Medicine, Computer Science Applications, Cell biology, 030104 developmental biology, Membrane protein, chemistry, lcsh:Biology (General), lcsh:QD1-999, lipids (amino acids, peptides, and proteins), 030217 neurology & neurosurgery, Function (biology), hormones, hormone substitutes, and hormone antagonists, Protein Binding

وصف الملف: application/pdf

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8b03ce097b7a92892fd9a5c3a6c343e8Test
http://europepmc.org/articles/PMC7920425Test

4

Menthol acts as a positive allosteric modulator on nematode levamisole sensitive nicotinic acetylcholine receptors

المؤلفون: Sasa M. Trailovic, Shivani Choudhary, Xiaoyu Zhang, Djordje S. Marjianović, Joel R. Coats, Alan P. Robertson, Richard J. Martin, Colin R. Wong, Melanie Abongwa

المصدر: International Journal for Parasitology: Drugs and Drug Resistance, Vol 9, Iss, Pp 44-53 (2019)
International Journal for Parasitology-Drugs and Drug Resistance
International Journal for Parasitology: Drugs and Drug Resistance

مصطلحات موضوعية: 0301 basic medicine, Allosteric modulator, 030231 tropical medicine, Cholinergic Agents, Receptors, Nicotinic, nAChR, Pharmacology, Article, lcsh:Infectious and parasitic diseases, Nicotine, Xenopus laevis, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Allosteric Regulation, medicine, Animals, lcsh:RC109-216, Pharmacology (medical), Receptor, Allosteric modulation, Ascaris suum, Nematode, Acetylcholine receptor, Anthelmintics, Monoterpenoid, 3. Good health, Oesophagostomum, Menthol, 030104 developmental biology, Infectious Diseases, Nicotinic agonist, Levamisole, chemistry, Monoterpenes, Cholinergic, Female, Parasitology, Acetylcholine, medicine.drug

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5f5f48a04db1e4b2cbd37f24e72e41b4Test
https://doi.org/10.1016/j.ijpddr.2018.12.005Test

5

The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase

المؤلفون: Marchesani, Gianquinto, Autiero, Michielon, Campanini, Faggiano, Bettati, Mozzarelli, Spyrakis, Bruno

المصدر: European journal of biochemistry 288 (2021): 3034–3054. doi:10.1111/febs.15645
info:cnr-pdr/source/autori:Marchesani, F. and Gianquinto, E. and Autiero, I. and Michielon, A. and Campanini, B. and Faggiano, S. and Bettati, S. and Mozzarelli, A. and Spyrakis, F. and Bruno, S./titolo:The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase/doi:10.1111%2Ffebs.15645/rivista:European journal of biochemistry/anno:2021/pagina_da:3034/pagina_a:3054/intervallo_pagine:3034–3054/volume:288