-
1
المؤلفون: Mark Smith, Justin P. Annes, Paul Allegretti, Benjamin Yeh, Matthew Caffet, Yassan Abdolazimi, Timothy M. Horton, Hannah P. Moeller, Guillermina Michel
المصدر: Bioorg Med Chem
مصطلحات موضوعية: DYRK1A, Clinical Biochemistry, Pharmaceutical Science, Protein Serine-Threonine Kinases, 01 natural sciences, Biochemistry, Article, Small Molecule Libraries, Structure-Activity Relationship, In vivo, Insulin-Secreting Cells, Drug Discovery, Humans, Insulin, Inducer, Naphthyridines, Cytotoxicity, Molecular Biology, Protein Kinase Inhibitors, Cell Proliferation, Binding Sites, 010405 organic chemistry, Kinase, Chemistry, Regeneration (biology), Organic Chemistry, Cell cycle, Protein-Tyrosine Kinases, Small molecule, 0104 chemical sciences, Cell biology, Protein Structure, Tertiary, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Kinetics, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::02c14bde7a6a312e8cc57343ff6fb1caTest
https://pubmed.ncbi.nlm.nih.gov/31757680Test -
2
المؤلفون: Paul Allegretti, Mark Smith, Justin P. Annes, Hannah P. Moeller, Sooyeon Lee, Timothy M. Horton
المصدر: Cell Chemical Biology. 26:213-222.e6
مصطلحات موضوعية: Male, Clinical Biochemistry, chemistry.chemical_element, Zinc, Protein Serine-Threonine Kinases, Biology, 01 natural sciences, Biochemistry, Article, Tosyl Compounds, Mice, Tandem Mass Spectrometry, Insulin-Secreting Cells, Drug Discovery, Animals, Humans, Moiety, Chelation, Protein Kinase Inhibitors, Molecular Biology, Chromatography, High Pressure Liquid, Chelating Agents, Pharmacology, geography, geography.geographical_feature_category, 010405 organic chemistry, Protein-Tyrosine Kinases, Ethylenediamines, Islet, Small molecule, 0104 chemical sciences, Cell biology, Mice, Inbred C57BL, chemistry, Dithizone, Drug delivery, Aminoquinolines, Molecular Medicine, Intracellular, Function (biology)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8521e602d26d282307860eb83cdf6556Test
https://doi.org/10.1016/j.chembiol.2018.10.019Test