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المؤلفون: Mirunalini Ravichandran, Subhiksha Subramanian
المصدر: Fundamental & Clinical Pharmacology. 36:72-80
مصطلحات موضوعية: Pharmacology, Nervous system, Orexins, Drug discovery, Neuropeptides, digestive, oral, and skin physiology, Optogenetics, Biology, Orexin receptor, Receptors, G-Protein-Coupled, medicine.anatomical_structure, nervous system, Orexin Receptors, Sleep Initiation and Maintenance Disorders, mental disorders, medicine, Drug approval, Humans, Pharmacology (medical), Receptor, Neuroscience, hormones, hormone substitutes, and hormone antagonists, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3940a00d6a047f0695b9a1c4ed9a95caTest
https://doi.org/10.1111/fcp.12723Test -
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المؤلفون: Jalal Zaringhalam, Shahrbanoo Oryan, Kobra Askari, Akram Eidi, Abbas Haghparast
المصدر: European Journal of Pain. 25:2266-2277
مصطلحات موضوعية: medicine.drug_class, Pain, Pharmacology, mental disorders, medicine, Noxious stimulus, Animals, Rats, Wistar, Receptor, Orexins, business.industry, musculoskeletal, neural, and ocular physiology, Ventral Tegmental Area, TCS-OX2-29, Receptor antagonist, Rats, Orexin, Ventral tegmental area, Anesthesiology and Pain Medicine, medicine.anatomical_structure, Nociception, nervous system, Analgesia, business, psychological phenomena and processes, Tail flick test, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0d7ddb066c1978153eef3578c4bde04fTest
https://doi.org/10.1002/ejp.1840Test -
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المؤلفون: Jagadeesh Aluri, Margaret Moline, Ziad Hussein, Oneeb Majid, Bojan Lalovic, Ishani Landry
المصدر: Journal of Clinical Pharmacology
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Adolescent, exposure‐response analysis, Pyridines, insomnia, Lemborexant, Administration, Oral, Drug Elimination Routes, Placebo, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, 0302 clinical medicine, Pharmacometrics, Pharmacokinetics, population pharmacokinetics, Sleep Initiation and Maintenance Disorders, Internal medicine, medicine, Humans, Pharmacology (medical), Adverse effect, Aged, Aged, 80 and over, Pharmacology, Clinical Trials as Topic, business.industry, Middle Aged, medicine.disease, Orexin receptor, Pyrimidines, Upper respiratory tract infection, orexin antagonist, Area Under Curve, 030220 oncology & carcinogenesis, Female, Orexin Receptor Antagonists, medicine.symptom, business, Body mass index, Somnolence
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b19a5d8098fca84dc00ffa96a77f0381Test
https://doi.org/10.1002/jcph.1683Test -
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المؤلفون: Junji Furukawa, Chika Higashi, Shunsuke Maehara, Takashi Takeuchi, Takumi Ota, Natsuko Yuge
المصدر: Neuropsychopharmacology Reports
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Administration, Oral, CHO Cells, Pharmacology, OX1 receptor, Rats, Sprague-Dawley, Cricetulus, Orexin Receptors, In vivo, Cricetinae, medicine, Animals, Humans, Pharmacology (medical), sleep, Receptor, Orexins, Chemistry, Antagonist, Electroencephalography, Original Articles, OX2 receptor, Receptor antagonist, In vitro, Rats, Bioavailability, Orexin, Psychiatry and Mental health, Clinical Psychology, orexin, Original Article, Orexin Receptor Antagonists
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::feb587ea061a73b9b03f49de9c18959cTest
https://doi.org/10.1002/npr2.12105Test -
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المؤلفون: Benjamin Berger, Jasper Dingemanse, Priska Kaufmann, Annelize Koch
المصدر: The Journal of Clinical Pharmacology. 60:931-941
مصطلحات موضوعية: Adult, Male, Hydrocortisone, CYP3A, medicine.drug_class, Midazolam, Urinary system, Pharmacology, 030226 pharmacology & pharmacy, Drug Administration Schedule, Young Adult, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Orexin Receptors, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, Pharmacology (medical), Adverse effect, business.industry, Middle Aged, Receptor antagonist, Healthy Volunteers, Orexin, Area Under Curve, 030220 oncology & carcinogenesis, Concomitant, Cytochrome P-450 CYP3A Inhibitors, Orexin Receptor Antagonists, business, Biomarkers, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::64a45b1401d368d57cd1f5de0f8b1f73Test
https://doi.org/10.1002/jcph.1588Test -
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المؤلفون: Tadashi Saigusa, Masami Yamaguchi, Manabu Ishikawa, Yuri Aono
المصدر: Neuropsychopharmacology Reports. 40:30-38
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, medicine.drug_class, Chemistry, Inhibitory postsynaptic potential, Receptor antagonist, Orexin receptor, Psychiatry and Mental health, Clinical Psychology, Orexin-A, Endocrinology, Nociception, medicine.anatomical_structure, nervous system, Dorsal root ganglion, Internal medicine, Hyperalgesia, medicine, Pharmacology (medical), Sciatic nerve, medicine.symptom
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::5eac72e3908bb928f3992efda4eea0b2Test
https://doi.org/10.1002/npr2.12094Test -
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المؤلفون: Larisa Reyderman, Jagadeesh Aluri, Kenya Nakai, Bojan Lalovic, Margaret Moline, Ishani Landry, Takashi Ueno, Satish Dayal, Yukiko Miyajima, Nancy Hall, Gleb Filippov
المصدر: Clinical Pharmacology in Drug Development
مصطلحات موضوعية: Adult, Male, CYP2B6, Pyridines, Itraconazole, CYP3A, orexin receptor antagonists, Cmax, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, 0302 clinical medicine, drug‐drug interaction, Pharmacokinetics, Cytochrome P-450 CYP3A, Humans, Medicine, Drug Interactions, Pharmacology (medical), Cytochrome P-450 Enzyme Inducers, Bupropion, business.industry, Brief Report, Middle Aged, Cytochrome P-450 CYP2B6, Pyrimidines, Area Under Curve, 030220 oncology & carcinogenesis, Cytochrome P-450 CYP3A Inhibitors, Midazolam, Female, Brief Reports, business, pharmacokinetics, Fluconazole, lemborexant, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bcf08514e8d52bbf289e88aa00268bcTest
https://doi.org/10.1002/cpdd.915Test -
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المؤلفون: John Gatfield, Catherine Roch, Thierry Sifferlen, Jodi T. Williams, Alexander Treiber, Christoph Boss, Martin Bolli, Christine Brotschi, Bibia Heidmann, Francois Jenck
المصدر: ChemMedChem. 14:1257-1270
مصطلحات موضوعية: Oxadiazole, Pharmacology, 01 natural sciences, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Orexin Receptors, Drug Discovery, Animals, Cytochrome P-450 CYP3A, Humans, General Pharmacology, Toxicology and Pharmaceutics, Receptor, Oxadiazoles, CYP3A4, 010405 organic chemistry, Organic Chemistry, Suvorexant, Antagonist, Azepines, Triazoles, Orexin receptor, Rats, 0104 chemical sciences, Orexin, 010404 medicinal & biomolecular chemistry, chemistry, Molecular Medicine, Orexin Receptor Antagonists, Wakefulness, Sleep, Half-Life
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b115f7c0f955cf770604ab0fdaa3d44Test
https://doi.org/10.1002/cmdc.201900242Test -
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المؤلفون: Henri Xhaard, Erik A.A. Wallén, Jari Yli-Kauhaluoma, Jyrki P. Kukkonen, Teppo O. Leino, Lasse Karhu, Ainoleena Turku
المصدر: ChemMedChem. 14:965-981
مصطلحات موضوعية: Pharmacology, Indole test, Agonist, Bicyclic molecule, 010405 organic chemistry, Stereochemistry, Chemistry, medicine.drug_class, Organic Chemistry, Biological activity, Potentiator, 01 natural sciences, Biochemistry, Orexin receptor, 0104 chemical sciences, 3. Good health, Orexin, 010404 medicinal & biomolecular chemistry, mental disorders, Drug Discovery, medicine, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Binding site, psychological phenomena and processes
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::61323be3ae0c6af0b57567aabae3d334Test
https://doi.org/10.1002/cmdc.201900074Test -
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المؤلفون: Clemens Muehlan, Ivan Ulč, Isabelle Zenklusen, Jasper Dingemanse, Jiří Liška
المصدر: Clinical and Experimental Pharmacology and Physiology. 47:1843-1849
مصطلحات موضوعية: Adult, 0301 basic medicine, Pyrrolidines, Physiology, Cmax, Pharmacology, Young Adult, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Physiology (medical), medicine, Humans, Distribution (pharmacology), Drug Interactions, Rosuvastatin, Rosuvastatin Calcium, IC50, Chemistry, Imidazoles, Antagonist, nutritional and metabolic diseases, Middle Aged, Orexin receptor, 030104 developmental biology, Tolerability, 030220 oncology & carcinogenesis, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::63d8165bab096fb86eba0bf6e9b7a33cTest
https://doi.org/10.1111/1440-1681.13370Test