المؤلفون: Alessia Lenoci, Maria E. Ourailidou, Clemens Zwergel, Dante Rotili, Antonello Mai, Frank J. Dekker

المساهمون: Chemical and Pharmaceutical Biology, Biopharmaceuticals, Discovery, Design and Delivery (BDDD), Medicinal Chemistry and Bioanalysis (MCB)

المصدر: Bioorganic & Medicinal Chemistry, 25(3), 847-856. PERGAMON-ELSEVIER SCIENCE LTD

مصطلحات موضوعية: 0301 basic medicine, Clinical Biochemistry, PROTEIN, Pharmaceutical Science, LSD1 HISTONE DEMETHYLASE, Biochemistry, law.invention, 0302 clinical medicine, THERAPEUTIC STRATEGY, law, Drug Discovery, Lysine demethylation, Enzyme Inhibitors, Histone Demethylases, chemistry.chemical_classification, Molecular Structure, DERIVATIVES, Chemistry, Irreversible inhibition, Biological activity, 030220 oncology & carcinogenesis, Biotinylation, Recombinant DNA, Molecular Medicine, HDAC INHIBITORS, LYSINE-SPECIFIC DEMETHYLASE 1, medicine.drug, STRUCTURAL BASIS, animal structures, Article, Structure-Activity Relationship, 03 medical and health sciences, OXIDATIVE HECK REACTION, lysine demethylation, tumorigenesis, tranylcypromine, irreversible inhibition, enzyme labeling, medicine, Humans, BREAST-CANCER, Molecular Biology, Dose-Response Relationship, Drug, Organic Chemistry, Tranylcypromine, Enzyme labeling, Protein profiling, 030104 developmental biology, Enzyme, Molecular Probes, Tumorigenesis, CELLS, BIOLOGICAL-ACTIVITY, Function (biology), HeLa Cells

وصف الملف: application/pdf

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9bc6385cc4af7e29bcb34a432f57c504Test
https://doi.org/10.1016/j.bmc.2016.11.043Test

المؤلفون: Di Pietro, Ornella, Alencar, Nelson, Esteban, Gerard, Viayna, Elisabet, Szałaj, Natalia, Vázquez, Javier, Juárez-Jiménez, Jordi, Sola, Irene, Pérez, Belén, Solé Piñol, Montserrat, Unzeta López, Mercedes, Muñoz-Torrero López-Ibarra, Diego, Luque Garriga, F. Xavier, Universitat Autònoma de Barcelona. Departament de Bioquímica i de Biologia Molecular

المصدر: Dipòsit Digital de Documents de la UAB
Universitat Autònoma de Barcelona

مصطلحات موضوعية: 0301 basic medicine, Monoamine Oxidase Inhibitors, Molecular model, Stereochemistry, Clinical Biochemistry, Triazole, Pharmaceutical Science, 01 natural sciences, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, Humans, Structure–activity relationship, Monoamine oxidase B, Monoamine Oxidase, Molecular Biology, Alkyl, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Irreversible inhibition, Alzheimer's disease, Cycloaddition, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, Pargyline, chemistry, Click-chemistry, Drug Design, Click chemistry, Molecular Medicine, Selectivity

وصف الملف: application/pdf

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4df53678fd7026e019de1edc4e4dabc4Test
https://doi.org/10.1016/j.bmc.2016.06.045Test

المؤلفون: Rose, Ngw, Blaskovich, MA, Wong, A, Lajoie, GA

مصطلحات موضوعية: vinylglycines, olefination, alpha-amino acid, Alpha-Amino-Acids, Stereoselective Synthesis, Enantioselective Synthesis, Asymmetric Syntheses, L-Vinylglycine, L-2-Amino-4-Methoxy-Trans-3-Butenoic Acid, Aspartate-Aminotransferase, Irreversible Inhibition, Practical Synthesis, Methyl-Esters

العلاقة: orcid:0000-0001-9447-2292

الإتاحة: https://doi.org/10.1016/S0040-4020Test(00)01146-7
https://espace.library.uq.edu.au/view/UQ:255844Test