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1
المؤلفون: Shoji Asakura, Michiyuki Suzuki, Kazutomi Kusano, Takashi Ueno, Tomomi Ishida, Carsten T. Beuckmann, Jagadeesh Aluri, Takaaki Kameyama
المصدر: Drug Metabolism and Disposition. 49:31-38
مصطلحات موضوعية: Pharmacology, business.industry, Metabolite, Glucuronidation, Pharmaceutical Science, Urine, 030226 pharmacology & pharmacy, Orexin receptor, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, chemistry, Oral administration, 030220 oncology & carcinogenesis, Medicine, business, Drug metabolism, ADME
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::310105c91488bc39459672158f368b02Test
https://doi.org/10.1124/dmd.120.000229Test -
2
المصدر: J Pharmacol Exp Ther
مصطلحات موضوعية: 0301 basic medicine, Agonist, Serotonin, Special Section on The Opioid Crisis, medicine.drug_class, Dopamine, Narcotic Antagonists, medicine.medical_treatment, media_common.quotation_subject, Drug Evaluation, Preclinical, Glutamic Acid, Bioinformatics, Partial agonist, 03 medical and health sciences, 0302 clinical medicine, medicine, Humans, media_common, Pharmacology, Clinical Trials as Topic, Neurotransmitter Agents, business.industry, Opioid use disorder, Abstinence, Opioid-Related Disorders, medicine.disease, Substance Withdrawal Syndrome, Orexin, Analgesics, Opioid, 030104 developmental biology, Opioid, Molecular Medicine, Cannabinoid, business, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0ca138ca665eef13c3906009c84cc728Test
https://doi.org/10.1124/jpet.119.258004Test -
3
المؤلفون: Friedbert Weiss, Alessandra Matzeu, Rémi Martin-Fardon, Tony M. Kerr
المصدر: Journal of Pharmacology and Experimental Therapeutics. 359:273-279
مصطلحات موضوعية: Male, 0301 basic medicine, medicine.medical_specialty, Lateral hypothalamus, Pyridines, Drug-Seeking Behavior, Thalamus, Extinction, Psychological, Cocaine dependence, 03 medical and health sciences, 0302 clinical medicine, Cocaine, Orexin Receptors, Internal medicine, medicine, Animals, Urea, Drug Interactions, Naphthyridines, Rats, Wistar, Receptor, Pharmacology, Benzoxazoles, Orexins, Antagonist, Extinction (psychology), Isoquinolines, medicine.disease, Orexin receptor, Rats, Orexin, 030104 developmental biology, Endocrinology, Behavioral Pharmacology, Molecular Medicine, Psychology, 030217 neurology & neurosurgery, Paraventricular Hypothalamic Nucleus
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5be26fd0f80f31097ee12f2261515075Test
https://doi.org/10.1124/jpet.116.235945Test -
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المؤلفون: Lebold Terry P, Diane Nepomuceno, Philip L. Johnson, Pascal Bonaventure, Michelle Wennerholm, Brian Lord, Jonathan Edward Shelton, Nicholas Carruthers, Shireman Brock T, Timothy W. Lovenberg, Anantha Shekhar, Christine Dugovic, Sujin Yun, Stephanie D. Fitz
المصدر: Journal of Pharmacology and Experimental Therapeutics. 352:590-601
مصطلحات موضوعية: Male, medicine.drug_class, Rapid eye movement sleep, Aminopyridines, CHO Cells, Pharmacology, Rats, Sprague-Dawley, Drug Discovery and Translational Medicine, Mice, Cricetulus, Piperidines, Orexin Receptors, Cricetinae, medicine, Animals, Humans, Hypnotics and Sedatives, Receptor, Mice, Knockout, Chemistry, Antagonist, Receptor antagonist, Rats, Orexin, Mice, Inbred C57BL, HEK293 Cells, Disinhibition, Anesthesia, Knockout mouse, Molecular Medicine, Orexin Receptor Antagonists, Sleep onset, medicine.symptom, Arousal, Stress, Psychological, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59a314c43002e84a551cda53e160fa9cTest
https://doi.org/10.1124/jpet.114.220392Test -
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المؤلفون: James R Shoblock, Sandra R. Chaplan, Anthony Ndifor, Steven W. Sutton, Nicholas I. Carruthers, Robin Halter, Michele C. Rizzolio, Ian Fraser, Tatiana Koudriakova, Pascal Bonaventure, Sujin Yun, Leah Aluisio, Christine Dugovic, Zuleima Aguilar, Jonathan Shelton, Brian Lord, Natalie Welty, Timothy W. Lovenberg, Michael A. Letavic, Diane Nepomuceno
المصدر: ResearcherID
مصطلحات موضوعية: Male, medicine.medical_specialty, Zolpidem, Pyridines, medicine.drug_class, Dopamine, Sleep, REM, CHO Cells, Pharmacology, Non-rapid eye movement sleep, Cell Line, Rats, Sprague-Dawley, Hypnotic, Mice, Cricetulus, Sleep Initiation and Maintenance Disorders, Internal medicine, medicine, Insomnia, Animals, Humans, Hypnotics and Sedatives, Mice, Knockout, Binding Sites, business.industry, Brain, Sleep in non-human animals, Rats, HEK293 Cells, Endocrinology, Sedative, Molecular Medicine, Orexin Receptor Antagonists, Sleep Stages, medicine.symptom, Sleep onset, Sleep, business, Somnolence, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58a22e350290152292370d7db2d63f57Test
https://doi.org/10.1124/jpet.115.225466Test -
6
المؤلفون: Tommaso Miraval, Jasper Dingemanse, Gérard Hopfgartner, Kasra Shakeri-Nejad, Winfried Wagner-Redeker, Alexander Treiber, Matthias Hoch, Petra Hoever
المصدر: Drug Metabolism and Disposition. 41:1046-1059
مصطلحات موضوعية: Adult, Male, Receptors, Neuropeptide, Administration, Oral, Pharmaceutical Science, Pharmacology, Receptors, G-Protein-Coupled, Excretion, chemistry.chemical_compound, Orexin Receptors, Tandem Mass Spectrometry, Oral administration, Acetamides, medicine, Humans, Demethylation, Tetrahydroisoquinoline, Half-life, Metabolism, Isoquinolines, Orexin receptor, chemistry, Biochemistry, Almorexant, Chromatography, Liquid, Half-Life, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::350cc9c10a17e8666f21084f570fdea4Test
https://doi.org/10.1124/dmd.112.050120Test -
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المؤلفون: Sami Reijonen, Maria Jäntti, Johnny Näsman, Jaana Putula, Pauli M. Turunen, Christer Lindqvist, Jyrki P. Kukkonen
المصدر: Molecular Pharmacology. 83:621-632
مصطلحات موضوعية: Receptors, Neuropeptide, Cannabinoid receptor, Arachidonic Acids, CHO Cells, Immune receptor, Biology, Pharmacology, Glycerides, Receptors, G-Protein-Coupled, 03 medical and health sciences, 0302 clinical medicine, Receptor, Cannabinoid, CB1, Orexin Receptors, Cricetinae, Animals, Humans, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Receptor, Autocrine signalling, 030304 developmental biology, 0303 health sciences, Receptor, Muscarinic M1, Endocannabinoid system, Orexin receptor, Orexin, Cell biology, Autocrine Communication, Lipoprotein Lipase, Molecular Medicine, Signal transduction, 030217 neurology & neurosurgery, Endocannabinoids, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7d08875e8b29c440ade307bf8db5fd8eTest
https://doi.org/10.1124/mol.112.080523Test -
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المؤلفون: Shang Cheng Huang, Ling Ling Hwang, Yu Wen E Dai, Yen Hsien Lee, Lih-Chu Chiou
المصدر: Journal of Pharmacology and Experimental Therapeutics. 334:522-529
مصطلحات موضوعية: Male, Receptors, Neuropeptide, medicine.medical_specialty, Patch-Clamp Techniques, Pyridines, Action Potentials, Blood Pressure, Receptors, G-Protein-Coupled, Orexin-A, Heart Rate, Orexin Receptors, Internal medicine, mental disorders, medicine, Animals, Premovement neuronal activity, Patch clamp, Neurons, Pharmacology, Medulla Oblongata, Orexins, Chemistry, Neuropeptides, digestive, oral, and skin physiology, Intracellular Signaling Peptides and Proteins, Rostral ventrolateral medulla, Isoquinolines, TCS-OX2-29, Immunohistochemistry, Orexin receptor, Rats, Orexin, Endocrinology, nervous system, Hypertension, Medulla oblongata, Molecular Medicine, Female, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3dc3990a5c1ab5d4ac0d1cc274f75d02Test
https://doi.org/10.1124/jpet.110.167791Test -
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المؤلفون: Anne Marcuz, Pari Malherbe, Olivier Roche, Claudia Kratzeisen, Joseph G. Wettstein, Caterina Bissantz
المصدر: Molecular Pharmacology. 78:81-93
مصطلحات موضوعية: Pharmacology, Stereochemistry, Antagonist, Biology, Orexin receptor, Orexin, chemistry.chemical_compound, Transmembrane domain, chemistry, medicine, Molecular Medicine, Almorexant, Binding site, Receptor, medicine.drug, EMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::195e5c9b026ae9d3fbafdc0bc260a541Test
https://doi.org/10.1124/mol.110.064584Test -
10
المصدر: Molecular Pharmacology. 76:618-631
مصطلحات موضوعية: Receptors, Neuropeptide, medicine.medical_specialty, Pyrrolidines, Pharmacology, Receptors, G-Protein-Coupled, Orexin Receptors, Internal medicine, Acetamides, medicine, Animals, Humans, Receptor, Evoked Potentials, Neurons, Molecular Structure, Chemistry, Phenylurea Compounds, Dopaminergic, Antagonist, Isoquinolines, Orexin receptor, Rats, Orexin, Ventral tegmental area, Kinetics, Thiazoles, Endocrinology, medicine.anatomical_structure, Competitive antagonist, Molecular Medicine, Almorexant, Sleep, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::afe058889cf26991657995fd0d4c9584Test
https://doi.org/10.1124/mol.109.055152Test