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المصدر: J Pharmacol Exp Ther
مصطلحات موضوعية: 0301 basic medicine, Agonist, Serotonin, Special Section on The Opioid Crisis, medicine.drug_class, Dopamine, Narcotic Antagonists, medicine.medical_treatment, media_common.quotation_subject, Drug Evaluation, Preclinical, Glutamic Acid, Bioinformatics, Partial agonist, 03 medical and health sciences, 0302 clinical medicine, medicine, Humans, media_common, Pharmacology, Clinical Trials as Topic, Neurotransmitter Agents, business.industry, Opioid use disorder, Abstinence, Opioid-Related Disorders, medicine.disease, Substance Withdrawal Syndrome, Orexin, Analgesics, Opioid, 030104 developmental biology, Opioid, Molecular Medicine, Cannabinoid, business, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0ca138ca665eef13c3906009c84cc728Test
https://doi.org/10.1124/jpet.119.258004Test -
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المؤلفون: Lebold Terry P, Diane Nepomuceno, Philip L. Johnson, Pascal Bonaventure, Michelle Wennerholm, Brian Lord, Jonathan Edward Shelton, Nicholas Carruthers, Shireman Brock T, Timothy W. Lovenberg, Anantha Shekhar, Christine Dugovic, Sujin Yun, Stephanie D. Fitz
المصدر: Journal of Pharmacology and Experimental Therapeutics. 352:590-601
مصطلحات موضوعية: Male, medicine.drug_class, Rapid eye movement sleep, Aminopyridines, CHO Cells, Pharmacology, Rats, Sprague-Dawley, Drug Discovery and Translational Medicine, Mice, Cricetulus, Piperidines, Orexin Receptors, Cricetinae, medicine, Animals, Humans, Hypnotics and Sedatives, Receptor, Mice, Knockout, Chemistry, Antagonist, Receptor antagonist, Rats, Orexin, Mice, Inbred C57BL, HEK293 Cells, Disinhibition, Anesthesia, Knockout mouse, Molecular Medicine, Orexin Receptor Antagonists, Sleep onset, medicine.symptom, Arousal, Stress, Psychological, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59a314c43002e84a551cda53e160fa9cTest
https://doi.org/10.1124/jpet.114.220392Test -
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المؤلفون: James R Shoblock, Sandra R. Chaplan, Anthony Ndifor, Steven W. Sutton, Nicholas I. Carruthers, Robin Halter, Michele C. Rizzolio, Ian Fraser, Tatiana Koudriakova, Pascal Bonaventure, Sujin Yun, Leah Aluisio, Christine Dugovic, Zuleima Aguilar, Jonathan Shelton, Brian Lord, Natalie Welty, Timothy W. Lovenberg, Michael A. Letavic, Diane Nepomuceno
المصدر: ResearcherID
مصطلحات موضوعية: Male, medicine.medical_specialty, Zolpidem, Pyridines, medicine.drug_class, Dopamine, Sleep, REM, CHO Cells, Pharmacology, Non-rapid eye movement sleep, Cell Line, Rats, Sprague-Dawley, Hypnotic, Mice, Cricetulus, Sleep Initiation and Maintenance Disorders, Internal medicine, medicine, Insomnia, Animals, Humans, Hypnotics and Sedatives, Mice, Knockout, Binding Sites, business.industry, Brain, Sleep in non-human animals, Rats, HEK293 Cells, Endocrinology, Sedative, Molecular Medicine, Orexin Receptor Antagonists, Sleep Stages, medicine.symptom, Sleep onset, Sleep, business, Somnolence, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58a22e350290152292370d7db2d63f57Test
https://doi.org/10.1124/jpet.115.225466Test -
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المؤلفون: Tommaso Miraval, Jasper Dingemanse, Gérard Hopfgartner, Kasra Shakeri-Nejad, Winfried Wagner-Redeker, Alexander Treiber, Matthias Hoch, Petra Hoever
المصدر: Drug Metabolism and Disposition. 41:1046-1059
مصطلحات موضوعية: Adult, Male, Receptors, Neuropeptide, Administration, Oral, Pharmaceutical Science, Pharmacology, Receptors, G-Protein-Coupled, Excretion, chemistry.chemical_compound, Orexin Receptors, Tandem Mass Spectrometry, Oral administration, Acetamides, medicine, Humans, Demethylation, Tetrahydroisoquinoline, Half-life, Metabolism, Isoquinolines, Orexin receptor, chemistry, Biochemistry, Almorexant, Chromatography, Liquid, Half-Life, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::350cc9c10a17e8666f21084f570fdea4Test
https://doi.org/10.1124/dmd.112.050120Test -
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المؤلفون: Sami Reijonen, Maria Jäntti, Johnny Näsman, Jaana Putula, Pauli M. Turunen, Christer Lindqvist, Jyrki P. Kukkonen
المصدر: Molecular Pharmacology. 83:621-632
مصطلحات موضوعية: Receptors, Neuropeptide, Cannabinoid receptor, Arachidonic Acids, CHO Cells, Immune receptor, Biology, Pharmacology, Glycerides, Receptors, G-Protein-Coupled, 03 medical and health sciences, 0302 clinical medicine, Receptor, Cannabinoid, CB1, Orexin Receptors, Cricetinae, Animals, Humans, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Receptor, Autocrine signalling, 030304 developmental biology, 0303 health sciences, Receptor, Muscarinic M1, Endocannabinoid system, Orexin receptor, Orexin, Cell biology, Autocrine Communication, Lipoprotein Lipase, Molecular Medicine, Signal transduction, 030217 neurology & neurosurgery, Endocannabinoids, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7d08875e8b29c440ade307bf8db5fd8eTest
https://doi.org/10.1124/mol.112.080523Test -
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المصدر: Molecular Pharmacology. 76:618-631
مصطلحات موضوعية: Receptors, Neuropeptide, medicine.medical_specialty, Pyrrolidines, Pharmacology, Receptors, G-Protein-Coupled, Orexin Receptors, Internal medicine, Acetamides, medicine, Animals, Humans, Receptor, Evoked Potentials, Neurons, Molecular Structure, Chemistry, Phenylurea Compounds, Dopaminergic, Antagonist, Isoquinolines, Orexin receptor, Rats, Orexin, Ventral tegmental area, Kinetics, Thiazoles, Endocrinology, medicine.anatomical_structure, Competitive antagonist, Molecular Medicine, Almorexant, Sleep, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::afe058889cf26991657995fd0d4c9584Test
https://doi.org/10.1124/mol.109.055152Test -
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المصدر: Pharmacological Reviews. 58:46-57
مصطلحات موضوعية: Receptors, Neuropeptide, Hypothalamo-Hypophyseal System, medicine.medical_specialty, Pituitary-Adrenal System, Receptors, G-Protein-Coupled, Orexin Receptors, Internal medicine, mental disorders, medicine, Animals, Humans, Pharmacology, Orexins, Chemistry, Adrenal cortex, Neuropeptides, digestive, oral, and skin physiology, Intracellular Signaling Peptides and Proteins, Orexin receptor, Orexin, medicine.anatomical_structure, Endocrinology, Glucocorticoid secretion, nervous system, Catecholamine, Molecular Medicine, Adrenal medulla, psychological phenomena and processes, hormones, hormone substitutes, and hormone antagonists, Glucocorticoid, Hypothalamic–pituitary–adrenal axis, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3d464269a73b84889eb1a344ce8a0103Test
https://doi.org/10.1124/pr.58.1.4Test -
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المؤلفون: Mark Wright, Stefano Zamuner, Paolo Bettica, Mario Pellegatti, Steven R. Thomas, Gary W. Boyle, Cecilia Renzulli, Mike Nash
المصدر: Drug Metabolism and Disposition. 39:215-227
مصطلحات موضوعية: Adult, Male, Receptors, Neuropeptide, Stereochemistry, Metabolite, Carboxylic acid, Administration, Oral, Pharmaceutical Science, Urine, Mass Spectrometry, Receptors, G-Protein-Coupled, Feces, chemistry.chemical_compound, Acetic acid, Orexin Receptors, medicine, Humans, Tissue Distribution, Carbon Radioisotopes, Benzofuran, Biotransformation, Chromatography, High Pressure Liquid, Benzofurans, Pharmacology, chemistry.chemical_classification, Molecular Structure, Chemistry, Metabolism, Middle Aged, Thiazoles, Hemiaminal, SB-649868, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::893492fb878b28111917fefe6e2dd81dTest
https://doi.org/10.1124/dmd.110.035386Test -
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المؤلفون: Takeshi Sakurai, Natsuko Tsujino
المصدر: Pharmacological Reviews. 61:162-176
مصطلحات موضوعية: Sleep Wake Disorders, medicine.medical_specialty, Molecular Sequence Data, Biology, Energy homeostasis, Reward system, Reward, Internal medicine, mental disorders, medicine, Animals, Homeostasis, Humans, Amino Acid Sequence, Wakefulness, Pharmacology, Orexins, Neuropeptides, digestive, oral, and skin physiology, Dopaminergic, Intracellular Signaling Peptides and Proteins, medicine.disease, Orexin, Endocrinology, nervous system, Hypothalamus, Molecular Medicine, Almorexant, Energy Metabolism, Sleep, Neuroscience, hormones, hormone substitutes, and hormone antagonists, psychological phenomena and processes, Signal Transduction, medicine.drug, Narcolepsy
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3bf12c4f0082a0759219f97f14bd0fb3Test
https://doi.org/10.1124/pr.109.001321Test