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المؤلفون: Andrea Brancale, Claire Simons, Chris Pepper, Salvatore Ferla, Justin T. Ochalek, Jinge Zhu, Ahmed S. Aboraia, Hector F. DeLuca
المصدر: Journal of Medicinal Chemistry. 57:7702-7715
مصطلحات موضوعية: Models, Molecular, RM, Stereochemistry, Antineoplastic Agents, Chemistry Techniques, Synthetic, Heme, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Catalytic Domain, Cell Line, Tumor, Drug Discovery, medicine, Cytochrome P-450 Enzyme Inhibitors, Humans, Imidazole, Structure–activity relationship, QD, Vitamin D3 24-Hydroxylase, Cell Proliferation, chemistry.chemical_classification, Sequence Homology, Amino Acid, biology, Imidazoles, Active site, R1, Leukemia, Lymphocytic, Chronic, B-Cell, Small molecule, Amino acid, chemistry, Docking (molecular), biology.protein, Molecular Medicine, Ketoconazole, medicine.drug
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6126ade9051c95c2959dd02a8d274fbeTest
https://doi.org/10.1021/jm5009314Test -
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المؤلفون: Grazia Chiellini, Hector F. DeLuca, Rafal Barycki, Jinge Zhu
المصدر: Biochemistry. 49:10403-10411
مصطلحات موضوعية: Drug Evaluation, Preclinical, HL-60 Cells, Biology, medicine.disease_cause, Biochemistry, Gene Expression Regulation, Enzymologic, law.invention, Mice, Maltose-binding protein, Affinity chromatography, CYP24A1, law, Escherichia coli, medicine, Animals, Humans, Enzyme kinetics, Enzyme Inhibitors, Vitamin D3 24-Hydroxylase, Cells, Cultured, chemistry.chemical_classification, Molecular biology, Recombinant Proteins, Enzyme, chemistry, Steroid Hydroxylases, biology.protein, Recombinant DNA, Receptors, Calcitriol, Heterologous expression, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6db8793d978e5694a3af88d390543d02Test
https://doi.org/10.1021/bi101488pTest -
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المصدر: Journal of Medicinal Chemistry. 50:5824-5832
مصطلحات موضوعية: Keratinocytes, Transcription, Genetic, Calcitriol, Duodenum, Stereochemistry, medicine.medical_treatment, TRPV Cation Channels, Vitamin D3 24-Hydroxylase, Ether, Binding, Competitive, Chemical synthesis, Calcitriol receptor, Cell Line, Steroid, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Benzyl Compounds, Drug Discovery, polycyclic compounds, medicine, Animals, Humans, Structure–activity relationship, Cell Proliferation, Chemistry, Stereoisomerism, Biological activity, Rats, Allyl Compounds, Mice, Inbred C57BL, Biochemistry, Alkynes, Steroid Hydroxylases, Receptors, Calcitriol, Molecular Medicine, Calcium, Female, lipids (amino acids, peptides, and proteins), Calcium Channels, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e1ff4456af3144b14abb4f478555aac4Test
https://doi.org/10.1021/jm070882dTest -
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المؤلفون: Miyuki Anzai, Kazuya Takenouchi, Akihiro Yoshida, Hiroshi Saito, Hiroaki Takayama, Daishiro Miura, Toshie Fujishima, Seiichi Ishizuka, Nozomi Saito, Atsushi Kittaka
المصدر: Organic Letters. 5:4859-4862
مصطلحات موضوعية: Vitamin, chemistry.chemical_classification, Osteosarcoma, Molecular Structure, Stereochemistry, Organic Chemistry, Cell Differentiation, HL-60 Cells, Biochemistry, Calcitriol receptor, Lactones, chemistry.chemical_compound, Calcitriol, Cytochrome P-450 Enzyme System, chemistry, Steroid Hydroxylases, Cytochrome P-450 Enzyme Inhibitors, Humans, Receptors, Calcitriol, Surface modification, Physical and Theoretical Chemistry, Vitamin D3 24-Hydroxylase, Lactone
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::654bc7dc9d003c268201b34e770965f9Test
https://doi.org/10.1021/ol035922wTest