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المؤلفون: Eleonora Spinozzi, Marta Ferrati, Cecilia Baldassarri, Filippo Maggi, Roman Pavela, Giovanni Benelli, Cristina Aguzzi, Laura Zeppa, Loredana Cappellacci, Alessandro Palmieri, Riccardo Petrelli
المصدر: Journal of Natural Products. 86:1307-1316
مصطلحات موضوعية: Pharmacology, Complementary and alternative medicine, Organic Chemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Analytical Chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::1a057bc4e19b3d8bb5f2960c42135e30Test
https://doi.org/10.1021/acs.jnatprod.3c00137Test -
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المؤلفون: Fabio Marchetti, Alessia Tombesi, Corrado Di Nicola, Riccardo Pettinari, Federico Verdicchio, Alessandra Crispini, Francesca Scarpelli, Cecilia Baldassarri, Elisa Marangoni, Anders Hofer, Agustín Galindo, Riccardo Petrelli
المصدر: Inorganic Chemistry. 61:13561-13575
مصطلحات موضوعية: Inorganic Chemistry, Oorganisk kemi, Physical and Theoretical Chemistry
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f99089aa605a3e0863003e90e651d5f5Test
https://doi.org/10.1021/acs.inorgchem.2c02201Test -
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المؤلفون: Fabio Marchetti, Armando J. L. Pombeiro, Riccardo Pettinari, Agustín Galindo, Loredana Cappellacci, Claudio Pettinari, Laura Bonfili, Massimiliano Cuccioloni, M. Fátima C. Guedes da Silva, Riccardo Petrelli, Anna Maria Eleuteri, Corrado Di Nicola
المصدر: Inorganic Chemistry. 57:14123-14133
مصطلحات موضوعية: Double bond, Pyrazolone, chemistry.chemical_element, Antineoplastic Agents, Crystallography, X-Ray, Ligands, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, Ruthenium, Inorganic Chemistry, chemistry.chemical_compound, Coordination Complexes, Cell Line, Tumor, medicine, Humans, Hexamethylbenzene, Pyrazolones, Physical and Theoretical Chemistry, Methylene, chemistry.chemical_classification, Molecular Structure, 010405 organic chemistry, Ligand, Hydrazones, Nuclear magnetic resonance spectroscopy, Tautomer, 0104 chemical sciences, Models, Chemical, chemistry, Drug Design, Quantum Theory, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7d5325af47e7a2eae4fdcf754627dba3Test
https://doi.org/10.1021/acs.inorgchem.8b01935Test -
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المؤلفون: Massimo Nabissi, Maura Pellei, Wilma Quaglia, Cristina Cimarelli, Alessandro Bonifazi, Dirk Schepmann, Riccardo Petrelli, Alessandro Piergentili, Consuelo Amantini, Valerio Mammoli, Giulio Vistoli, Fabio Del Bello, Bernhard Wünsch, Elisabetta Barocelli, Giorgio Santoni, Lisa Flammini, Simona Bertoni
المصدر: Journal of Medicinal Chemistry. 58:8601-8615
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Pain, Phencyclidine, Ligands, Receptors, N-Methyl-D-Aspartate, Dioxanes, Mice, Drug Discovery, medicine, Animals, Receptors, sigma, Moiety, Binding site, Receptor, Analgesics, Binding Sites, Chemistry, Antagonist, Affinities, Rats, Drug Design, Molecular Medicine, NMDA receptor, Pharmacophore, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33c7677a77ebe0542d0780d716a34aacTest
https://doi.org/10.1021/acs.jmedchem.5b01214Test -
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المؤلفون: Alessandro Paiardini, Loredana Cappellacci, Livia Leoni, Fabio Del Bello, Marco Messina, Francesca Cutruzzolà, Riccardo Petrelli, Ilaria Torquati, Silvia Fernicola, Giorgio Giardina, Serena Rinaldo, Giordano Rampioni
المساهمون: Fernicola, Silvia, Torquati, Ilaria, Paiardini, Alessandro, Giardina, Giorgio, Rampioni, Giordano, Messina, Marco, Leoni, Livia, Del Bello, Fabio, Petrelli, Riccardo, Rinaldo, Serena, Cappellacci, Loredana, Cutruzzolà, Francesca
المصدر: Journal of Medicinal Chemistry. 58:8269-8284
مصطلحات موضوعية: Models, Molecular, Guanine, Phosphodiesterase Inhibitors, Stereochemistry, Allosteric regulation, pharmaceutical science, Substrate Specificity, Structure-Activity Relationship, Drug Discovery, c-di-GMP, biofilm, Pseudomonas aeruginosa, Caulobacter crescentus, WspR, PleD, RocR, inhibitors, copper(I)-catalyzed 1,3-dipolar cycloaddition, click chemistry, Huisgen cycloaddition, alkynes, azides, dinucleoside, heterodinucleoside, 1,2,3-triazole, purine, Structure–activity relationship, Moiety, Cyclic GMP, biology, Chemistry, Escherichia coli Proteins, Active site, Triazoles, Small molecule, Anti-Bacterial Agents, Biofilms, Drug Design, Pseudomonas aeruginosa, Phosphodiester bond, Second messenger system, biology.protein, Molecular Medicine, Indicators and Reagents, Diguanylate cyclase, Phosphorus-Oxygen Lyases, molecular medicine, drug discovery
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::246111e3c149a657b36c79f2f870cc89Test
https://doi.org/10.1021/acs.jmedchem.5b01184Test -
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المؤلفون: Palmarisa Franchetti, Flavio Cimadamore, Leonardo Sorci, Stefania Scotti, Riccardo Petrelli, Loredana Cappellacci, Giulio Magni, G. Orsomando
المصدر: Biochemistry. 46:4912-4922
مصطلحات موضوعية: Niacinamide, Stereochemistry, Magnesium Chloride, Pyridinium Compounds, Biochemistry, Isozyme, Cell Line, Substrate Specificity, chemistry.chemical_compound, Chlorides, Cell Line, Tumor, NMNAT1, Ribavirin, medicine, Humans, Nicotinamide-Nucleotide Adenylyltransferase, Ternary complex, Nicotinamide mononucleotide, Nicotinamide, Nicotinamide-nucleotide adenylyltransferase, NAD, Isoenzymes, Kinetics, chemistry, Zinc Compounds, Product inhibition, Tiazofurin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e91060701cbce16d4c28b5023c0ec7e3Test
https://doi.org/10.1021/bi6023379Test -
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المؤلفون: Mario Grifantini, Karl-Norbert Klotz, Patrizia Vita, Palmarisa Franchetti, Claudia Martini, Antonio Lavecchia, Loredana Cappellacci, Barbara Costa, Ettore Novellino, M. Pasqualini, Riccardo Petrelli
المساهمون: L., Cappellacci, P., Franchetti, M., Pasqualini, R., Petrelli, P., Vita, Lavecchia, Antonio, Novellino, Ettore, B., Costa, C., Martini, K. N., Klotz, M., Grifantini
المصدر: Journal of Medicinal Chemistry. 48:1550-1562
مصطلحات موضوعية: Models, Molecular, Agonist, Adenosine, drug design, Stereochemistry, medicine.drug_class, Ribose, homology modeling, Carboxamide, CHO Cells, In Vitro Techniques, Binding, Competitive, Radioligand Assay, chemistry.chemical_compound, Adenosine A1 receptor, Cricetulus, GPCR, Cricetinae, Drug Discovery, Purinergic P1 Receptor Agonists, medicine, Animals, Humans, Receptor, molecular dynamic, Receptors, Purinergic P1, Brain, molecular docking, Adenosine receptor, Rats, Biochemistry, chemistry, Adenylyl Cyclase Inhibitors, CCPA, Molecular Medicine, Cattle, A1 adenosine receptor agonist, medicine.drug
وصف الملف: ELETTRONICO
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::93f2a13e636613050de836e3bd342781Test
https://doi.org/10.1021/jm049408nTest