التفاصيل البيبلوغرافية
العنوان: |
Structure–Activity Relationship Studies and Discovery of a Potent Transient Receptor Potential Vanilloid (TRPV1) Antagonist 4-[3-Chloro-5-[(1 S)-1,2-dihydroxyethyl]-2-pyridyl]- N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2 H-pyridine-1-carboxamide (V116517) as a Clinical Candidate for Pain Management |
المؤلفون: |
Tafesse, Laykea, Kanemasa, Toshiyuki, Kurose, Noriyuki, Yu, Jianming, Asaki, Toshiyuki, Wu, Gang, Iwamoto, Yuka, Yamaguchi, Yoshitaka, Ni, Chiyou, Engel, John, Tsuno, Naoki, Patel, Aniket, Zhou, Xiaoming, Shintani, Takuya, Brown, Kevin, Hasegawa, Tsuyoshi, Shet, Manjunath, Iso, Yasuyoshi, Kato, Akira, Kyle, Donald J. |
المصدر: |
Journal of Medicinal Chemistry ; volume 57, issue 15, page 6781-6794 ; ISSN 0022-2623 1520-4804 |
بيانات النشر: |
American Chemical Society (ACS) |
سنة النشر: |
2014 |
مصطلحات موضوعية: |
Drug Discovery, Molecular Medicine |
نوع الوثيقة: |
article in journal/newspaper |
اللغة: |
English |
DOI: |
10.1021/jm500818a |
الإتاحة: |
https://doi.org/10.1021/jm500818aTest |
رقم الانضمام: |
edsbas.B3396A7D |
قاعدة البيانات: |
BASE |