دورية أكاديمية

Structure–Activity Relationship Studies and Discovery of a Potent Transient Receptor Potential Vanilloid (TRPV1) Antagonist 4-[3-Chloro-5-[(1 S)-1,2-dihydroxyethyl]-2-pyridyl]- N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2 H-pyridine-1-carboxamide (V116517) as a Clinical Candidate for Pain Management

التفاصيل البيبلوغرافية
العنوان: Structure–Activity Relationship Studies and Discovery of a Potent Transient Receptor Potential Vanilloid (TRPV1) Antagonist 4-[3-Chloro-5-[(1 S)-1,2-dihydroxyethyl]-2-pyridyl]- N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2 H-pyridine-1-carboxamide (V116517) as a Clinical Candidate for Pain Management
المؤلفون: Tafesse, Laykea, Kanemasa, Toshiyuki, Kurose, Noriyuki, Yu, Jianming, Asaki, Toshiyuki, Wu, Gang, Iwamoto, Yuka, Yamaguchi, Yoshitaka, Ni, Chiyou, Engel, John, Tsuno, Naoki, Patel, Aniket, Zhou, Xiaoming, Shintani, Takuya, Brown, Kevin, Hasegawa, Tsuyoshi, Shet, Manjunath, Iso, Yasuyoshi, Kato, Akira, Kyle, Donald J.
المصدر: Journal of Medicinal Chemistry ; volume 57, issue 15, page 6781-6794 ; ISSN 0022-2623 1520-4804
بيانات النشر: American Chemical Society (ACS)
سنة النشر: 2014
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
نوع الوثيقة: article in journal/newspaper
اللغة: English
DOI: 10.1021/jm500818a
الإتاحة: https://doi.org/10.1021/jm500818aTest
رقم الانضمام: edsbas.B3396A7D
قاعدة البيانات: BASE