-
1دورية أكاديمية
المؤلفون: Jian Wang (5901), Nikolay V. Dokholyan (84409)
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Genetics, Pharmacology, Infectious Diseases, Virology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Information Systems not elsewhere classified, various data sets, computational drug screening, predict binding affinities, drug target identification, upon comprehensive tests, learning approaches surveyed, unknown small molecules, small molecules, protein target, predict interactions, unknown proteins, unknown compounds, existing methods, deep learning, best ability, based approaches
-
2دورية أكاديمية
المؤلفون: Summers, Robert, Pasaje, Charisse, Pisco, Joao, Striepen, Josefine, Luth, Madeline, Kumpornsin, Krittikorn, Carpenter, Emma, Munro, Justin, Lin, De, Plater, Andrew, Punekar, Avinash, Shepherd, Andrew, Shepherd, Sharon, Vanaerschot, Manu, Murithi, James, Rubiano, Kelly, Akidil, Aslı, Ottilie, Sabine, Mittal, Nimisha, Dilmore, A, Won, Madalyn, Mandt, Rebecca, McGowen, Kerry, Owen, Edward, Walpole, Chris, Llinás, Manuel, Lee, Marcus, Fidock, David, Gilbert, Ian, Wirth, Dyann, Niles, Jacquin, Baragaña, Beatriz, Lukens, Amanda, Winzeler, Elizabeth
المصدر: Cell Chemical Biology, vol 29, iss 2
مصطلحات موضوعية: Plasmodium falciparum, acetyl-CoA synthetase, antimalarial, drug development, drug target identification, histone acetylation, malaria, mechanism of action, Acetate-CoA Ligase, Antimalarials, Enzyme Inhibitors, Humans, Models, Molecular, Molecular Structure, Parasitic Sensitivity Tests
وصف الملف: application/pdf
العلاقة: qt2t51p0mx; https://escholarship.org/uc/item/2t51p0mxTest
-
3
المؤلفون: Maria Gordillo-Maranon
مصطلحات موضوعية: Genomics, Pharmacogenomics, genome-wide association studies, GWAS, drug target identification and validation
الإتاحة: https://doi.org/10.5522/04/25541392.v1Test
https://figshare.com/articles/dataset/Disease_coverage_overlap_and_divergence_of_human_genome-wide_association_studies_and_pharmaceutical_research_and_development/25541392Test -
4دورية أكاديمية
المؤلفون: Yingrong Xu (1778419), Graham M. West (624715), Mario Abdelmessih (11254994), Matthew D. Troutman (2291176), Robert A. Everley (811578)
مصطلحات موضوعية: Biophysics, Biochemistry, Genetics, Molecular Biology, Physiology, Pharmacology, Biotechnology, Inorganic Chemistry, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, chemical-denaturation-based SPROX, Stability Proteomics Methods, MS time, affinity purification methods, thermal-denaturation-based TPP, 2 D setup, OnePot 2 D formats, Drug Target Identification, kinase hits, protein domain-level information, K 562 lysate, higher-molecular-weight proteins, drug target engagement studies, data analysis, peptide-level quantification, OnePot 2 D format, OnePot 2 D Format Stability proteom., Unique SPROX hits, protein targets, resource efficiency
-
5
المؤلفون: Matthew J. Winter, Yosuke Ono, Jonathan S. Ball, Anna Walentinsson, Erik Michaelsson, Anna Tochwin, Steffen Scholpp, Charles R. Tyler, Steve Rees, Malcolm J Hetheridge, Mohammad Bohlooly-Y
مصطلحات موضوعية: Pharmacology, Basic Pharmacology, Clinical Pharmacology and Therapeutics, Clinical Pharmacy and Pharmacy Practice, Pharmaceutical Sciences, Pharmacogenomics, Toxicology (incl. Clinical Toxicology), Pharmacology and Pharmaceutical Sciences not elsewhere classified, CRISPR/Cas9, zebrafish, heart failure, drug target identification and validation, human whole exome sequencing
الإتاحة: https://doi.org/10.3389/fphar.2022.827686.s001Test
https://figshare.com/articles/dataset/DataSheet1_A_Combined_Human_in_Silico_and_CRISPR_Cas9-Mediated_in_Vivo_Zebrafish_Based_Approach_to_Provide_Phenotypic_Data_for_Supporting_Early_Target_Validation_zip/19645320Test -
6
المؤلفون: Ophélie Lo-Thong-Viramoutou, Philippe Charton, Xavier F. Cadet, Brigitte Grondin-Perez, Emma Saavedra, Cédric Damour, Frédéric Cadet
مصطلحات موضوعية: Artificial Intelligence and Image Processing, Knowledge Representation and Machine Learning, Applied Statistics, Computational Linguistics, artificial intelligence, machine learning, non-linear modeling, drug target identification, Trypanosoma cruzi detoxification pathway, Entamoeba histolytica glycolysis pathway, penicillin production
الإتاحة: https://doi.org/10.3389/frai.2022.744755.s004Test
https://figshare.com/articles/dataset/Table_3_Non-linearity_of_Metabolic_Pathways_Critically_Influences_the_Choice_of_Machine_Learning_Model_XLSX/20046320Test -
7
المؤلفون: Ophélie Lo-Thong-Viramoutou, Philippe Charton, Xavier F. Cadet, Brigitte Grondin-Perez, Emma Saavedra, Cédric Damour, Frédéric Cadet
مصطلحات موضوعية: Artificial Intelligence and Image Processing, Knowledge Representation and Machine Learning, Applied Statistics, Computational Linguistics, artificial intelligence, machine learning, non-linear modeling, drug target identification, Trypanosoma cruzi detoxification pathway, Entamoeba histolytica glycolysis pathway, penicillin production
الإتاحة: https://doi.org/10.3389/frai.2022.744755.s001Test
https://figshare.com/articles/dataset/Data_Sheet_1_Non-linearity_of_Metabolic_Pathways_Critically_Influences_the_Choice_of_Machine_Learning_Model_pdf/20046311Test -
8
المؤلفون: Ophélie Lo-Thong-Viramoutou, Philippe Charton, Xavier F. Cadet, Brigitte Grondin-Perez, Emma Saavedra, Cédric Damour, Frédéric Cadet
مصطلحات موضوعية: Artificial Intelligence and Image Processing, Knowledge Representation and Machine Learning, Applied Statistics, Computational Linguistics, artificial intelligence, machine learning, non-linear modeling, drug target identification, Trypanosoma cruzi detoxification pathway, Entamoeba histolytica glycolysis pathway, penicillin production
الإتاحة: https://doi.org/10.3389/frai.2022.744755.s005Test
https://figshare.com/articles/dataset/Table_4_Non-linearity_of_Metabolic_Pathways_Critically_Influences_the_Choice_of_Machine_Learning_Model_XLSX/20046323Test -
9
المؤلفون: Ophélie Lo-Thong-Viramoutou, Philippe Charton, Xavier F. Cadet, Brigitte Grondin-Perez, Emma Saavedra, Cédric Damour, Frédéric Cadet
مصطلحات موضوعية: Artificial Intelligence and Image Processing, Knowledge Representation and Machine Learning, Applied Statistics, Computational Linguistics, artificial intelligence, machine learning, non-linear modeling, drug target identification, Trypanosoma cruzi detoxification pathway, Entamoeba histolytica glycolysis pathway, penicillin production
الإتاحة: https://doi.org/10.3389/frai.2022.744755.s002Test
https://figshare.com/articles/dataset/Table_1_Non-linearity_of_Metabolic_Pathways_Critically_Influences_the_Choice_of_Machine_Learning_Model_XLSX/20046314Test -
10
المؤلفون: Ophélie Lo-Thong-Viramoutou, Philippe Charton, Xavier F. Cadet, Brigitte Grondin-Perez, Emma Saavedra, Cédric Damour, Frédéric Cadet
مصطلحات موضوعية: Artificial Intelligence and Image Processing, Knowledge Representation and Machine Learning, Applied Statistics, Computational Linguistics, artificial intelligence, machine learning, non-linear modeling, drug target identification, Trypanosoma cruzi detoxification pathway, Entamoeba histolytica glycolysis pathway, penicillin production
الإتاحة: https://doi.org/10.3389/frai.2022.744755.s003Test
https://figshare.com/articles/dataset/Table_2_Non-linearity_of_Metabolic_Pathways_Critically_Influences_the_Choice_of_Machine_Learning_Model_XLSX/20046317Test