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1
المؤلفون: Massimiliano Cuccioloni, Laura Bonfili, Mauro Angeletti, Riccardo Petrelli, Loredana Cappellacci, Anna Maria Eleuteri, Massimo Nabissi, Fabio Marchetti, Riccardo Pettinari, Valentina Cecarini
المصدر: ChemMedChem. 15:105-113
مصطلحات موضوعية: Cell Membrane Permeability, Stereochemistry, media_common.quotation_subject, Serum albumin, Hydrazone, chemistry.chemical_element, Antineoplastic Agents, Apoptosis, 01 natural sciences, Biochemistry, Ruthenium, Cell membrane, chemistry.chemical_compound, Coordination Complexes, Cell Line, Tumor, Drug Discovery, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Internalization, Cytotoxicity, media_common, Pharmacology, chemistry.chemical_classification, Binding Sites, biology, 010405 organic chemistry, Organic Chemistry, Hydrazones, Cell Cycle Checkpoints, DNA, In vitro, 0104 chemical sciences, Molecular Docking Simulation, Kinetics, 010404 medicinal & biomolecular chemistry, medicine.anatomical_structure, chemistry, biology.protein, Nucleic Acid Conformation, Molecular Medicine, Hydroxymethylglutaryl CoA Reductases, Cyclin-Dependent Kinase Inhibitor p27, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6998f8b0f4699db4e3fa2f6f17dbac7aTest
https://doi.org/10.1002/cmdc.201900551Test -
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المؤلفون: Francesco Alessandro Palermo, Laura Bonfili, Aida Capone, Irene Ricci, Matteo Mozzicafreddo, Mauro Angeletti, Massimiliano Cuccioloni, Paolo Cocci, Anna Maria Eleuteri, Valentina Cecarini, Gilberto Mosconi
المصدر: The Journal of Steroid Biochemistry and Molecular Biology. 152:1-7
مصطلحات موضوعية: Receptors, Steroid, medicine.drug_class, Endocrinology, Diabetes and Metabolism, In silico, Clinical Biochemistry, Phthalic Acids, Biology, Biochemistry, Endocrinology, Cell Line, Tumor, Gene expression, medicine, Humans, RNA, Messenger, Liver X receptor, Receptor, Molecular Biology, Transcription factor, Liver X Receptors, Binding Sites, Bile acid, Fibric Acids, Liver X receptor alpha, Hep G2 Cells, Cell Biology, Metabolism, Orphan Nuclear Receptors, Organophosphates, Molecular Docking Simulation, Molecular Medicine, Environmental Pollutants, Sterol Regulatory Element Binding Protein 1, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::86c189d0f0273dae68e0b3136cf19ef5Test
https://doi.org/10.1016/j.jsbmb.2015.04.011Test -
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المؤلفون: Massimiliano Cuccioloni, Matteo Mozzicafreddo, Valentina Cecarini, Mauro Angeletti, Laura Bonfili, Giacomo Rossi, Anna Maria Eleuteri, Jeffrey N. Keller
المصدر: Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease. 1842:127-134
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Cell Survival, Leupeptins, Proteolysis, Blotting, Western, Cysteine Proteinase Inhibitors, Protein degradation, Cathepsin B, Amyloid beta-Protein Precursor, Ubiquitin, Cell Line, Tumor, Autophagy, medicine, Amyloid precursor protein, Humans, Molecular Biology, biology, medicine.diagnostic_test, Adenine, Immunohistochemistry, Cell biology, Amino Acid Substitution, Proteasome, Biochemistry, Mutation, Ubiquitin–proteasome system, biology.protein, Proteasome inhibitor, Molecular Medicine, Mutant Proteins, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6069901796a75d1be793c0cd8b0c0e80Test
https://doi.org/10.1016/j.bbadis.2013.11.002Test -
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المؤلفون: Mauro Angeletti, Laura Bonfili, Matteo Mozzicafreddo, Anna Maria Eleuteri, Valentina Cecarini, Massimiliano Cuccioloni
المصدر: Chemical biologydrug design. 74(1)
مصطلحات موضوعية: Drug, Proteases, Serine Proteinase Inhibitors, media_common.quotation_subject, Endogeny, Biochemistry, Serine, Small Molecule Libraries, Structure-Activity Relationship, Phenols, Catalytic Domain, Drug Discovery, media_common, Pharmacology, chemistry.chemical_classification, Serine protease, Flavonoids, biology, Organic Chemistry, Serine Endopeptidases, Proteolytic enzymes, Polyphenols, Protein Structure, Tertiary, Enzyme, chemistry, Drug Design, biology.protein, Molecular Medicine, Pharmacophore
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a5b5361c81358b32cf902bb157723efdTest
https://pubmed.ncbi.nlm.nih.gov/19519739Test