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1دورية أكاديمية
المؤلفون: Shkedi, Arielle, Adkisson, Michael, Schroeder, Andrew, Eckalbar, Walter L, Kuo, Szu-Yu, Neckers, Leonard, Gestwicki, Jason E
المصدر: Journal of Medicinal Chemistry. 64(19)
مصطلحات موضوعية: Urologic Diseases, Cancer, Prostate Cancer, Antineoplastic Agents, Cell Line, Tumor, Cell Survival, HSP70 Heat-Shock Proteins, HSP90 Heat-Shock Proteins, Humans, Male, Prostatic Neoplasms, Proteasome Endopeptidase Complex, Proteostasis, Receptors, Androgen, Sequence Analysis, RNA, Stress, Physiological, Medicinal and Biomolecular Chemistry, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/0md990s0Test
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2دورية أكاديمية
المؤلفون: LaMonte, Gregory M, Almaliti, Jehad, Bibo-Verdugo, Betsaida, Keller, Lena, Zou, Bing Yu, Yang, Jennifer, Antonova-Koch, Yevgeniya, Orjuela-Sanchez, Pamela, Boyle, Colleen A, Vigil, Edgar, Wang, Lawrence, Goldgof, Gregory M, Gerwick, Lena, O’Donoghue, Anthony J, Winzeler, Elizabeth A, Gerwick, William H, Ottilie, Sabine
المصدر: Journal of Medicinal Chemistry. 60(15)
مصطلحات موضوعية: Biotechnology, Rare Diseases, Orphan Drug, Vector-Borne Diseases, Infectious Diseases, Malaria, Development of treatments and therapeutic interventions, 5.1 Pharmaceuticals, Infection, Good Health and Well Being, Antimalarials, Artemisinins, Dipeptides, Drug Design, Enzyme Assays, Hep G2 Cells, Humans, Molecular Docking Simulation, Oligopeptides, Plasmodium falciparum, Proteasome Endopeptidase Complex, Proteasome Inhibitors, Saccharomyces cerevisiae, Medicinal and Biomolecular Chemistry, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/0r57k1b0Test
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3
المؤلفون: Dipti Kanabar, Mimansa Goyal, Emma I. Kane, Tejashri Chavan, Abbas Kabir, Xuechun Wang, Snehal Shukla, Joseph Almasri, Sona Goswami, Gizem Osman, Marino Kokolis, Donald E. Spratt, Vivek Gupta, Aaron Muth
المصدر: Journal of medicinal chemistry. 65(13)
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Lung Neoplasms, Tumor Suppressor Proteins, Drug Discovery, Liver Neoplasms, Molecular Medicine, Humans
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::445014929000f13b6e2282c0fd170988Test
https://pubmed.ncbi.nlm.nih.gov/35758870Test -
4
المؤلفون: Xinyi Wu, Ping Sun, Xiuhui Chen, Lei Hua, Haowei Cai, Zhuorong Liu, Cheng Zhang, Shuli Liang, Yanhong Chen, Dan Wu, Yitao Ou, Wenhui Hu, Zhongjin Yang
المصدر: Journal of Medicinal Chemistry. 65:11985-12001
مصطلحات موضوعية: Mice, Inbred C57BL, Mice, Proteasome Endopeptidase Complex, Inflammasomes, Interleukin-1beta, NLR Family, Pyrin Domain-Containing 3 Protein, Drug Discovery, Anti-Inflammatory Agents, Animals, Molecular Medicine, Proteasome Inhibitors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aab8a2f7ce644c8aa45e667a1041b10fTest
https://doi.org/10.1021/acs.jmedchem.2c00523Test -
5
المؤلفون: Zhen Dai, Lu-yan An, Xiao-yi Chen, Fan Yang, Ni Zhao, Cui-cui Li, Ren Ren, Bing-yan Li, Wei-yan Tao, Pei Li, Cheng Jiang, Fang Yan, Zheng-yu Jiang, Qi-dong You, Bin Di, Li-li Xu
المصدر: Journal of Medicinal Chemistry. 65:5029-5043
مصطلحات موضوعية: Oxadiazoles, Oxidative Stress, Proteasome Endopeptidase Complex, NF-E2-Related Factor 2, Drug Discovery, Hunting, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f6a868bdc79e37c4cc3ee514246faec3Test
https://doi.org/10.1021/acs.jmedchem.1c02210Test -
6
المؤلفون: Xufen Yu, Jia Xu, Yudao Shen, Kaitlyn M. Cahuzac, Kwang-su Park, Brandon Dale, Jing Liu, Ramon E. Parsons, Jian Jin
المصدر: J Med Chem
مصطلحات موضوعية: Male, Proteasome Endopeptidase Complex, Dose-Response Relationship, Drug, Ubiquitin, Biological Availability, Mice, Nude, Antineoplastic Agents, Xenograft Model Antitumor Assays, Article, Mice, Structure-Activity Relationship, Pyrimidines, Cell Line, Tumor, PC-3 Cells, Proteolysis, Drug Discovery, Animals, Humans, Molecular Medicine, Pyrroles, Protein Kinase Inhibitors, Proto-Oncogene Proteins c-akt, Cell Division, Tumor Stem Cell Assay
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::339785175c1d33f70c781f6819c2f890Test
https://doi.org/10.1021/acs.jmedchem.1c02165Test -
7
المؤلفون: Jibu Lu, Yongjun Huang, Jing Huang, Rui He, Minhao Huang, Xiaoyun Lu, Yong Xu, Fengtao Zhou, Zhang Zhang, Ke Ding
المصدر: Journal of Medicinal Chemistry. 65:2313-2328
مصطلحات موضوعية: Male, Proteasome Endopeptidase Complex, Transplantation, Heterologous, Mice, SCID, Protein-Tyrosine Kinases, Ligands, Mice, Structure-Activity Relationship, Von Hippel-Lindau Tumor Suppressor Protein, Cell Line, Tumor, Drug Design, Neoplasms, Proteolysis, Drug Discovery, Animals, Humans, Molecular Medicine, Protein Kinase Inhibitors, Cell Proliferation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7ea1215ad315f59529f85ec1249b81aaTest
https://doi.org/10.1021/acs.jmedchem.1c01768Test -
8
المؤلفون: Xuechun Li, Ming Li, Chen Li, Guang Yang, Ning Liu, Ruonan Wang, Cheng Yang, Sheng Cao, Lan Ma, Yulin Liu, Zhiqiang Dong, Xiaoji Wang, Yuhong Yao, Mingming Wei
المصدر: Journal of Medicinal Chemistry. 64:16497-16511
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Antineoplastic Agents, Apoptosis, Drug resistance, Quinolones, medicine.disease_cause, Structure-Activity Relationship, In vivo, Cell Line, Tumor, hemic and lymphatic diseases, Drug Discovery, medicine, Humans, Cell Proliferation, Mutation, Ubiquitin, Chemistry, Proteolysis targeting chimera, Myeloid leukemia, hemic and immune systems, In vitro, body regions, Leukemia, Myeloid, Acute, fms-Like Tyrosine Kinase 3, Proteolysis, embryonic structures, Cancer research, Molecular Medicine, Benzimidazoles, Antiproliferative effect, Reactive Oxygen Species, psychological phenomena and processes, Signal Transduction, Flt3 itd
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::22bc3c0ff7344688035716e00fe57921Test
https://doi.org/10.1021/acs.jmedchem.1c00996Test -
9
المؤلفون: Cong, Li, Song, Liu, Baoyu, Dong, Chungen, Li, Lunan, Jian, Juan, He, Jumei, Zeng, Qiao, Zhou, Da, Jia, Youfu, Luo, Qingxiang, Sun
المصدر: Journal of medicinal chemistry. 65(16)
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Adenosine Triphosphate, Bacterial Proteins, Mycobacterium tuberculosis, Bithionol, Proteasome Inhibitors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::62870c8dc28f348f9fdcc44474cd2240Test
https://pubmed.ncbi.nlm.nih.gov/35926511Test -
10
المؤلفون: Felix Rohdich, Stefano Crosignani, Michael Busch, Christina Esdar, Manja Friese-Hamim, Markus Klein, Thomas Fuchss, Oliver Schadt, Djordje Musil, Ugo Zanelli, Michael P. Sanderson, Gina Walter-Bausch, Philip Hewitt, Jeyaprakashnarayanan Seenisamy
المصدر: Journal of Medicinal Chemistry. 64:10230-10245
مصطلحات موضوعية: Gene isoform, Proteasome Endopeptidase Complex, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Protein subunit, Protein degradation, medicine.disease, Protein Subunits, Structure-Activity Relationship, Haematopoiesis, Proteasome, Biochemistry, Drug Discovery, medicine, Humans, Molecular Medicine, Potency, Structure based, Proteasome Inhibitors, Multiple myeloma
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c1a3d051fc60306aef1b64a7ba1b3e7bTest
https://doi.org/10.1021/acs.jmedchem.1c00604Test