-
1
المؤلفون: James R. Gosset, Zhiwu Lin, Jeffrey R. Chabot, Odette A. Fahmi, Albert M. Kim, Vu Le, Parya Nouri, Amit S. Kalgutkar, Steven G. Terra, Leonard Buckbinder, Jennifer Q. Dong, Kristin Chidsey
المصدر: Drug Metabolism and Disposition. 45:501-511
مصطلحات موضوعية: Adult, Male, 0301 basic medicine, Population, Cmax, Pharmaceutical Science, Pyrimidinones, Pharmacology, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Statistical significance, Acetamides, medicine, Cytochrome P-450 CYP3A, Humans, heterocyclic compounds, RNA, Messenger, Enzyme Inhibitors, education, Cells, Cultured, Peroxidase, education.field_of_study, CYP3A4, Cholesterol, Area under the curve, Middle Aged, 030104 developmental biology, chemistry, Enzyme Induction, Hepatocytes, Midazolam, Female, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d5f66b7e444e3d1890b02b39832bfc45Test
https://doi.org/10.1124/dmd.116.074476Test -
2
المؤلفون: Li Di, Bo Feng, Jennifer Q. Dong, Kazuko Sagawa, Tim F. Ryder, Manthena V.S. Varma, Steven G. Terra, Amit S. Kalgutkar, Angela Wolford
المصدر: Drug Metabolism and Disposition. 44:209-219
مصطلحات موضوعية: Male, 0301 basic medicine, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Pharmaceutical Science, Pyrimidinones, Pharmacology, 030226 pharmacology & pharmacy, Thiouracil, Mice, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Pharmacokinetics, Acetamides, Animals, Cytochrome P-450 Enzyme Inhibitors, Humans, Rats, Wistar, Peroxidase, biology, Chemistry, Cytochrome P450, Haplorhini, In vitro, Rats, Bioavailability, HEK293 Cells, 030104 developmental biology, Intestinal Absorption, Myeloperoxidase, Renal physiology, Hepatocytes, Microsomes, Liver, biology.protein, Microsome, Female, Caco-2 Cells, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cfca1f808303a6721d41a7358f78ad02Test
https://doi.org/10.1124/dmd.115.067868Test