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المؤلفون: Kristin Beirow, Julia Jedamzik, Lukas Schulig, Konrad W. Wurm, Christian J. Lemmerhirt, Robert K. Hofstetter, Andreas Link, Patrick J. Bednarski
المصدر: ChemMedChem.
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Biochemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::0e8a268eaeb445ef757b1d01a0fea24aTest
https://doi.org/10.1002/cmdc.202300145Test -
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المؤلفون: Konrad W. Wurm, Frieda‐Marie Bartz, Lukas Schulig, Anja Bodtke, Patrick J. Bednarski, Andreas Link
المصدر: ChemMedChem. 17(16)
مصطلحات موضوعية: Pharmacology, KCNQ Potassium Channels, Organic Chemistry, Drug Discovery, Molecular Medicine, Aminopyridines, Carbamates, General Pharmacology, Toxicology and Pharmaceutics, Phenylenediamines, Biochemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::698ae1acec4bb254149c5ab8a71b8bc9Test
https://pubmed.ncbi.nlm.nih.gov/35687532Test -
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المؤلفون: Anja Bodtke, Markus K. Kindermann, Kristin Beirow, Andreas Link, Christian Bock, Patrick J. Bednarski, Abdrrahman Shemsu Surur, Lukas Schulig
المصدر: ChemMedChem. 14:952-964
مصطلحات موضوعية: Pharmacology, Liver injury, chemistry.chemical_classification, Sulfide, 010405 organic chemistry, Retigabine, Organic Chemistry, medicine.disease, 01 natural sciences, Biochemistry, Propanamide, Potassium channel, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, chemistry, Drug Discovery, Toxicity, medicine, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Flupirtine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::22343d7220e977504c96263ec6d95cabTest
https://doi.org/10.1002/cmdc.201900112Test -
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المؤلفون: Martin Napierkowski, Lisa Wolff, Siva Sankar Murthy Bandaru, Claudia Urbainsky, Steven Behnisch‐Cornwell, Carola Schulzke, Christopher Horst Lillig, Muhammad Zubair, Patrick J. Bednarski
المصدر: Chemmedchem
مصطلحات موضوعية: GPX1, Thioredoxin reductase, Glutathione reductase, DNA fragmentation, Apoptosis, medicine.disease_cause, 01 natural sciences, Biochemistry, chemistry.chemical_compound, Glutathione Peroxidase GPX1, Heterocyclic Compounds, Drug Discovery, Tumor Cells, Cultured, General Pharmacology, Toxicology and Pharmaceutics, Enzyme Inhibitors, chemistry.chemical_classification, Membrane Potential, Mitochondrial, biology, Full Paper, Molecular Structure, Chemistry, Glutathione peroxidase, Full Papers, Molecular Medicine, cytotoxicity, Cell Survival, Antineoplastic Agents, Sulfides, Superoxide dismutase, Structure-Activity Relationship, Very Important Paper, medicine, Humans, Cell Proliferation, Pharmacology, Reactive oxygen species, Glutathione Peroxidase, pentathiepin, Dose-Response Relationship, Drug, 010405 organic chemistry, Organic Chemistry, Glutathione, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Oxidative Stress, biology.protein, cancer cells, Drug Screening Assays, Antitumor, Oxidative stress
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0ccc766db533f3ed3c5850477407fbc9Test
https://pubmed.ncbi.nlm.nih.gov/32311219Test -
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المؤلفون: Christian, Bock, Abdrrahman S, Surur, Kristin, Beirow, Markus K, Kindermann, Lukas, Schulig, Anja, Bodtke, Patrick J, Bednarski, Andreas, Link
المصدر: ChemMedChem. 14(9)
مصطلحات موضوعية: HEK293 Cells, Potassium Channels, Aminopyridines, Humans, Carbamates, Phenylenediamines, Oxidation-Reduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::f8510d3efc6493c659a5686de87e8851Test
https://pubmed.ncbi.nlm.nih.gov/30861620Test -
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المؤلفون: Siva Sankar Murthy Bandaru, Christopher Horst Lillig, Patrick J. Bednarski, Muhammad Zubair, Steven Behnisch‐Cornwell, Carola Schulzke, Claudia Urbainsky, Martin Napierkowski, Lisa Wolff
المصدر: ChemMedChem. 15:1497-1497
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Membrane potential, GPX1, Glutathione peroxidase, Organic Chemistry, medicine.disease_cause, Biochemistry, Cell biology, chemistry, Apoptosis, Drug Discovery, Cancer cell, medicine, Molecular Medicine, DNA fragmentation, General Pharmacology, Toxicology and Pharmaceutics, Cytotoxicity, Oxidative stress
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::25a192debb204c604460d447d10687d3Test
https://doi.org/10.1002/cmdc.202000577Test -
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المصدر: ChemMedChem. 10:368-379
مصطلحات موضوعية: Cell Survival, Nitrogen, Potassium, Analgesic, Aminopyridines, chemistry.chemical_element, Mice, Transgenic, Pharmacology, Biochemistry, Cell Line, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, General Pharmacology, Toxicology and Pharmaceutics, Cytotoxicity, Analgesics, KCNQ Potassium Channels, Retigabine, Organic Chemistry, Electrochemical Techniques, Transforming Growth Factor alpha, Potassium channel, Acetaminophen, HEK293 Cells, Mechanism of action, chemistry, Hepatocytes, Molecular Medicine, medicine.symptom, Flupirtine, Oxidation-Reduction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d5a1db43422724f869881e1c59a45bc7Test
https://doi.org/10.1002/cmdc.201402442Test -
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المصدر: ChemMedChem. 5:103-117
مصطلحات موضوعية: Molecular model, Stereochemistry, Caspase 3, Cysteine Proteinase Inhibitors, Molecular Dynamics Simulation, Crystallography, X-Ray, Caspase 8, Biochemistry, Catalytic Domain, Drug Discovery, Humans, Amino Acid Sequence, General Pharmacology, Toxicology and Pharmaceutics, Pechmann condensation, Caspase, Fluorescent Dyes, Pharmacology, Binding Sites, Tetrapeptide, biology, Chemistry, Organic Chemistry, Hydrogen Bonding, AutoDock, Recombinant Proteins, Kinetics, Docking (molecular), biology.protein, Molecular Medicine, Oligopeptides
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dcd1292366d53758d7725a47d15a8caTest
https://doi.org/10.1002/cmdc.200900356Test -
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المؤلفون: Renate Grünert, Ralph Holl, Hans-Ulrich Humpf, Dirk Schepmann, Bettina Jung, Patrick J. Bednarski, Bernhard Wünsch, Werner Englberger
المصدر: ChemMedChem. 4:2111-2122
مصطلحات موضوعية: Intrinsic activity, Stereochemistry, Ligands, Ring (chemistry), Biochemistry, Piperazines, Cell Line, Stereocenter, δ-opioid receptor, chemistry.chemical_compound, Cell Line, Tumor, Receptors, Opioid, delta, Drug Discovery, Humans, Moiety, General Pharmacology, Toxicology and Pharmaceutics, Piperazine, Cell Proliferation, Pharmacology, Molecular Structure, Bicyclic molecule, Organic Chemistry, Affinities, chemistry, Benzamides, Molecular Medicine, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7d35da34f3392bfd3f0f94fdc1272a27Test
https://doi.org/10.1002/cmdc.200900358Test -
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المؤلفون: Renate Grünert, Janice R. Aldrich-Wright, Dianne M. Fisher, Ronald R. Fenton, Peter Turner, Patrick J. Bednarski
المصدر: ChemMedChem. 2:488-495
مصطلحات موضوعية: Models, Molecular, Stereochemistry, chemistry.chemical_element, Antineoplastic Agents, Platinum Compounds, Crystal structure, Biochemistry, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Humans, Cytotoxic T cell, General Pharmacology, Toxicology and Pharmaceutics, Pharmacology, Cisplatin, Molecular Structure, Organic Chemistry, Leukemia L1210, Intercalating Agents, In vitro, chemistry, Molecular Medicine, Orthorhombic crystal system, Platinum, Chirality (chemistry), medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::13d7a007eb807942d2b658bacd482567Test
https://doi.org/10.1002/cmdc.200600211Test