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1دورية أكاديمية
المؤلفون: Liddle, John1 john.2.liddle@gsk.com, Bamborough, Paul1, Barker, Michael D.1, Campos, Sebastien1, Chung, Chun-Wa1, Cousins, Rick P.C.1, Faulder, Paul1, Heathcote, Michelle L.1, Hobbs, Heather1, Holmes, Duncan S.1, Ioannou, Chris1, Ramirez-Molina, Cesar1, Morse, Mary A.1, Osborn, Ruth2, Payne, Jeremy J.1, Pritchard, John M.1, Rumsey, William L.2, Tape, Daniel T.1, Vicentini, Giorgia1, Whitworth, Caroline1
المصدر: Bioorganic & Medicinal Chemistry Letters. Aug2012, Vol. 22 Issue 16, p5222-5226. 5p.
مصطلحات موضوعية: *PHENYL compounds, *AZAINDOLE derivatives, *BIOAVAILABILITY, *CHEMICAL inhibitors, *MATHEMATICAL optimization, *AZAINDOLES
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2دورية أكاديمية
المؤلفون: Swarbrick, Martin E., Beswick, Paul J., Gleave, Robert J. robert.j.gleave@gsk.com, Green, Richard H.1, Bingham, Sharon1, Bountra, Chas, Carter, Malcolm C., Chambers, Laura J.1, Chessell, Iain P., Clayton, Nick M.1, Collins, Sue D.1, Corfield, John A.1, Hartley, C. David, Kleanthous, Savvas1, Lambeth, Paul F.1, Lucas, Fiona S.1, Mathews, Neil, Naylor, Alan1, Page, Lee W.1, Payne, Jeremy J.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Aug2009, Vol. 19 Issue 15, p4504-4508. 5p.
مصطلحات موضوعية: *CYCLOOXYGENASE 2 inhibitors, *ETHER (Anesthetic), *PHARMACOKINETICS, *ALLERGIES, *PYRIMIDINES, *ANIMAL models in research
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3دورية أكاديمية
المؤلفون: Liddle, John1 john.2.liddle@gsk.com, Bamborough, Paul1, Barker, Michael D.1, Campos, Sebastien1, Cousins, Rick P.C.1, Cutler, Geoffrey J.2, Hobbs, Heather1, Holmes, Duncan S.1, Ioannou, Chris1, Mellor, Geoff W.2, Morse, Mary A.1, Payne, Jeremy J.1, Pritchard, John M.1, Smith, Kathryn J.1, Tape, Daniel T.1, Whitworth, Caroline1, Williamson, Richard A.1
المصدر: Bioorganic & Medicinal Chemistry Letters. May2009, Vol. 19 Issue 9, p2504-2508. 5p.
مصطلحات موضوعية: *INDOLE, *PROTEIN kinases, *ENZYME inhibitors, *ORGANIC synthesis, *STRUCTURE-activity relationships, *BINDING sites