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المؤلفون: Yongbo Hu, Karen Collins, Edward J. Salaski, Nancy Torres, Eileen Frommer, Dennis Powell, Wang Xiaolun, Jeremy I. Levin, Donald Wojciechowicz, Dan Maarten Berger
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6571-6574
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Substrate Specificity, Structure-Activity Relationship, Pyrimidine analogue, Drug Discovery, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Kinase, Organic Chemistry, In vitro, Pyrimidines, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Pyrazoles, Molecular Medicine, Signal transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::981acddc510eaf8186f924c43131f046Test
https://doi.org/10.1016/j.bmcl.2009.10.030Test -
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المؤلفون: Nancy Torres, Eileen Frommer, Bloom Jonathan David, Karen Collins, Dunnick Alejandro Lee, George Diamantidis, Yongbo Hu, Minu Dutia, Christoph W. Zapf, Zhang Chunchun, Darrin William Hopper, Dan Maarten Berger, Donald Wojciechowicz, Dennis Powell, Martin Di Grandi, Jeremy I. Levin
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6957-6961
مصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Pyridines, Isostere, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Humans, Enzyme Inhibitors, Cytotoxicity, Molecular Biology, Cell Proliferation, chemistry.chemical_classification, Indazole, biology, Bicyclic molecule, Cell growth, Organic Chemistry, Pyrimidines, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Pyrazoles, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6346230a46b93ee107f73ab7d8869701Test
https://doi.org/10.1016/j.bmcl.2009.10.058Test -
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المؤلفون: Steven C. Kim, Frederick Lee, Eileen Frommer, Mengxiao Shi, Yongbo Hu, Donald Wojciechowicz, Robert Mallon, Greg Ciszewski, Dan Maarten Berger, Karen Collins, Ariamala Gopalsamy, Larry Feldberg
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6890-6892
مصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Pyrimidine, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Carboxamide, Biochemistry, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Kinase, Organic Chemistry, Hit to lead, Pyrimidines, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Pyrazoles, Molecular Medicine, Signal transduction, Lead compound
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9a6af29a6344c217dfecdc0daf235230Test
https://doi.org/10.1016/j.bmcl.2009.10.074Test