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1دورية أكاديمية
المؤلفون: Raubo, Piotr1 piotr.raubo@astrazeneca.com, Andrews, David M.1, McKelvie, Jennifer C.2, Robb, Graeme R.1, Smith, James M.1,3, Swarbrick, Martin E.3, Waring, Michael J.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Aug2015, Vol. 25 Issue 16, p3189-3193. 5p.
مصطلحات موضوعية: *SMALL molecules, *PHOSPHATIDYLINOSITOL 3-kinases, *PLATELET-derived growth factor, *STRUCTURAL optimization, *CELLULAR signal transduction, *BIOACCUMULATION
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2دورية أكاديمية
المؤلفون: Jones, Clifford D. cliff.jones@astrazeneca.com, Andrews, David M.1, Barker, Andrew J.1, Blades, Kevin1, Byth, Kate F.1, Finlay, M. Raymond V.1, Geh, Catherine1, Green, Clive P.1, Johannsen, Marie1, Walker, Mike1, Weir, Hazel M.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Dec2008, Vol. 18 Issue 24, p6486-6489. 4p.
مصطلحات موضوعية: *ENZYME inhibitors, *CYCLIN-dependent kinases, *IMIDAZOLES, *PYRIMIDINES, *CANCER cells, *DRUG lipophilicity, *ION channels, *PHARMACOKINETICS
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3دورية أكاديمية
المؤلفون: Jones, Clifford D.1 cliff.jones@astrazeneca.com, Andrews, David M.1, Barker, Andrew J.1, Blades, Kevin1, Daunt, Paula1, East, Simon1, Geh, Catherine1, Graham, Mark A.1, Johnson, Keith M.1, Loddick, Sarah A.1, McFarland, Heather M.1, McGregor, Alexandra1, Moss, Louise1, Rudge, David A.1, Simpson, Peter B.1, Swain, Michael L.1, Tam, Kin Y.1, Tucker, Julie A.2, Walker, Mike1
المصدر: Bioorganic & Medicinal Chemistry Letters. Dec2008, Vol. 18 Issue 24, p6369-6373. 5p.
مصطلحات موضوعية: *ENZYME inhibitors, *AMIDES, *PYRIMIDINES, *CYCLIN-dependent kinases, *CELL cycle, *CANCER cells, *XENOGRAFTS, *PHARMACEUTICAL chemistry
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4دورية أكاديمية
المؤلفون: Anderson, Malcolm1, Andrews, David M.1, Barker, Andy J.1, Brassington, Claire A.1, Breed, Jason1, Byth, Kate F., Culshaw, Janet D.1, Finlay, M. Raymond V.1, Fisher, Eric1, McMiken, Helen H.J.1, Green, Clive P. clive.green@astrazeneca.com, Heaton, Dave W.1, Nash, Ian A.1, Newcombe, Nicholas J.1, Oakes, Sandra E.1, Pauptit, Richard A.1, Roberts, Andrew1, Stanway, Judith J.1, Thomas, Andrew P.1, Tucker, Julie A.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Oct2008, Vol. 18 Issue 20, p5487-5492. 6p.
مصطلحات موضوعية: *IMIDAZOLES, *CYCLIN-dependent kinases, *CHEMICAL inhibitors, *DIMETHYL sulfone, *STRUCTURE-activity relationships, *CLINICAL medicine
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5دورية أكاديمية
المؤلفون: Andrews, David M. david.andrews@astrazeneca.com, Stokes, Elaine S.E. elaine.stokes@astrazeneca.com, Carr, Greg R.1, Matusiak, Zbigniew S.1, Roberts, Craig A.1, Waring, Michael J.1, Brady, Madeleine C.1, Chresta, Christine M.1, East, Simon J.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Apr2008, Vol. 18 Issue 8, p2580-2584. 5p.
مصطلحات موضوعية: *PIPERIDINE, *THIAZOLES, *HISTONE deacetylase, *PHARMACEUTICAL chemistry
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6دورية أكاديمية
المؤلفون: Andrews, David M. david.andrews@astrazeneca.com, Gibson, Keith M.1, Graham, Mark A.1, Matusiak, Zbigniew S.1, Roberts, Craig A.1, Stokes, Elaine S.E.1, Brady, Madeleine C.1, Chresta, Christine M.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Apr2008, Vol. 18 Issue 8, p2525-2529. 5p.
مصطلحات موضوعية: *BENZAMIDE, *MOIETIES (Chemistry), *MOLECULAR weights, *PHARMACEUTICAL chemistry
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7دورية أكاديمية
المؤلفون: Andrews, David M. da9978@gsk.com, Jones, Paul S.1, Mills, Gail1, Hind, S. Lucy1, Slater, Martin J.1, Trivedi, Naimisha1, Wareing, Katrina J.1
المصدر: Bioorganic & Medicinal Chemistry Letters. May2003, Vol. 13 Issue 10, p1657. 4p.
مصطلحات موضوعية: *PROTEOLYTIC enzymes, *HEPATITIS C, *LACTAMS
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8دورية أكاديمية
المؤلفون: Slater, Martin J. mjs40312@gsk.com, Andrews, David M.1, Baker, Graham1, Bethell, Susanne S.1, Carey, Seb1, Chaignot, Helene1, Clarke, Berwyn1, Coomber, Barry1, Ellis, Malcolm1, Good, Andrew1, Gray, Norman1, Hardy, George1, Jones, Paul1, Mills, Gail1, Robinson, Ed1
المصدر: Bioorganic & Medicinal Chemistry Letters. Dec2002, Vol. 12 Issue 23, p3359. 4p.
مصطلحات موضوعية: *PYRROLIDINE, *ENZYME inhibitors, *HEPATITIS C
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9دورية أكاديمية
المؤلفون: Finlay, M. Raymond V.1 ray.finlay@astrazeneca.com, Acton, David G.1, Andrews, David M.1, Barker, Andrew J.1, Dennis, Michael1, Fisher, Eric1, Graham, Mark A.1, Green, Clive P.1, Heaton, David W.1, Karoutchi, Galith1, Loddick, Sarah A.1, Morgentin, Rémy2, Roberts, Andrew1, Tucker, Julie A.3, Weir, Hazel M.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Aug2008, Vol. 18 Issue 15, p4442-4446. 5p.
مصطلحات موضوعية: *TUMORS, *PATHOLOGY, *CYSTS (Pathology), *ONCOLOGY
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10دورية أكاديمية
المؤلفون: Bradbury, Robert H. rob.bradbury@astrazeneca.com, Hales, Neil J., Rabow, Alfred A., Walker, Graeme E., Acton, David G.1, Andrews, David M.1, Ballard, Peter1, Brooks, Nigel A.N.1, Colclough, Nicola1, Girdwood, Alan1, Hancox, Urs J.1, Jones, Owen1, Jude, David1, Loddick, Sarah A.1, Mortlock, Andrew A.1
المصدر: Bioorganic & Medicinal Chemistry Letters. Sep2011, Vol. 21 Issue 18, p5442-5445. 4p.
مصطلحات موضوعية: *PROSTATE cancer treatment, *ANTIANDROGENS, *STEROID hormones, *DRUG administration, *ORAL drug administration, *PHARMACEUTICAL chemistry