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المؤلفون: Dennis V. Nazareno, Guowei Zhou, Herbert Binch, William J. Greenlee, Mary Cohen-Williams, Jayaram R. Tagat, Diane E. Grotz, Jean E. Lachowicz, James J. Kaminski, Joseph A. Kozlowski, Gordon Crosby, Stuart W. McCombie, Vicki L. Coffin, Kathleen Cox, Vilma Ruperto, Craig D. Boyle, Samuel Chackalamannil, Ruth A. Duffy, Hubert B. Josien, Yuguang Wang, John W. Clader, William Billard
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2311-2314
مصطلحات موضوعية: Stereochemistry, Microdialysis, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Dioxoles, Muscarinic Antagonists, Benzylidene Compounds, Biochemistry, Structure-Activity Relationship, Cytochrome P-450 Enzyme System, Drug Stability, Pharmacokinetics, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Moiety, Sulfones, Molecular Biology, Receptor, Muscarinic M2, Oxidative metabolism, Chemistry, Organic Chemistry, Muscarinic antagonist, Receptors, Muscarinic, Acetylcholine, Rats, Bioavailability, Macaca fascicularis, Area Under Curve, Drug Design, Microsomes, Liver, Microsome, Molecular Medicine, Selectivity, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4596ee0f6758218aaf4305ca38b8523fTest
https://doi.org/10.1016/s0960-894xTest(01)00435-8 -
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المؤلفون: Guowei Zhou, Ruth A. Duffy, Herbert Binch, Jean E. Lachowicz, Lisa A. Taylor, William Billard, Derek B. Lowe, Joseph A. Kozlowski, Robert D. McQuade, Gordon Crosby, Vilma Ruperto, Henry Guzik
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2255-2257
مصطلحات موضوعية: Pyridines, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Muscarinic Antagonists, Naphthalenes, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Alkaloids, Piperidines, Dibenzazepines, Drug Discovery, Muscarinic acetylcholine receptor, Benzene Derivatives, medicine, Animals, Humans, Structure–activity relationship, Furans, Receptor, Molecular Biology, Receptor, Muscarinic M2, Organic Chemistry, Antagonist, Muscarinic antagonist, Muscarinic acetylcholine receptor M2, Sulfoxide, Receptors, Muscarinic, Acetylcholine, Corpus Striatum, Recombinant Proteins, Rats, chemistry, Drug Design, Molecular Medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4687a6dfde6b8966420c582c2ce3bbebTest
https://doi.org/10.1016/s0960-894xTest(00)00438-8