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1
المؤلفون: Junichi Sakamoto, Kazue Tsuchimori, Yoshimasa Ishimura, Taiji Asami, Taisuke Mochida, Hideki Hirabayashi, Yoko Kanematsu-Yamaki, Tomoko Asakawa, Mariko Yoneyama-Hirozane, Yusuke Adachi, Naoki Nishizawa, Kouta Matsumiya, Hisashi Fujita, Hideo Fukui, Shiro Takekawa, Ayumu Niida
المصدر: Bioorganic & Medicinal Chemistry. 26:566-572
مصطلحات موضوعية: 0301 basic medicine, Agonist, Alkylation, Vomiting, medicine.drug_class, Clinical Biochemistry, Cmax, Mice, Obese, Pharmaceutical Science, Polyethylene glycol, Pharmacology, Infusions, Subcutaneous, Biochemistry, Polyethylene Glycols, Mice, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Pharmacokinetics, Drug Discovery, PEG ratio, medicine, Animals, Peptide YY, Amino Acid Sequence, Obesity, Molecular Biology, Organic Chemistry, Receptors, Neuropeptide Y, Mice, Inbred C57BL, 030104 developmental biology, chemistry, 030220 oncology & carcinogenesis, Anorectic, PEGylation, Molecular Medicine, Anti-Obesity Agents, Emetics, Half-Life
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::485a325364207c8d6fe45019dc4bf804Test
https://doi.org/10.1016/j.bmc.2017.12.014Test -
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المؤلفون: Nathalie Pop, Nikola Pluym, Shangjun Teng, Max Keller, Daniela Erdmann, Günther Bernhardt, Armin Buschauer
المصدر: Bioorganic & Medicinal Chemistry. 19:2859-2878
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Arginine, Biochemistry, Chemical synthesis, Flow cytometry, law.invention, chemistry.chemical_compound, Confocal microscopy, law, Cell Line, Tumor, Drug Discovery, medicine, Humans, Benzothiazoles, Cyanine, Guanidine, Molecular Biology, Fluorescent Dyes, medicine.diagnostic_test, Organic Chemistry, Antagonist, Flow Cytometry, Fluorescence, Combinatorial chemistry, Receptors, Neuropeptide Y, chemistry, Molecular Medicine, Linker, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::689988770eefafb4597a4847845bb315Test
https://doi.org/10.1016/j.bmc.2011.03.045Test -
3
المؤلفون: Tetsuya Kanno, Nagaaki Sato, Toshiyuki Takahashi, Akio Kanatani, Aya Sakuraba, Hisashi Iwaasa, Tomoko Hirohashi, Takehiro Fukami, Takunobu Shibata, Masaaki Hirose, Katsumasa Nonoshita, Yuji Haga, Junko Ito
المصدر: Bioorganic & Medicinal Chemistry. 14:7501-7511
مصطلحات موضوعية: Y5 Receptor, Molecular Structure, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Phenylpiperazine, Neuropeptide Y receptor, Biochemistry, Piperazines, Receptors, Neuropeptide Y, Structure-Activity Relationship, Piperazine, chemistry.chemical_compound, Drug Discovery, Humans, Molecular Medicine, Moiety, Urea derivatives, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::60db73a33b6a2ab5ea27175a791d4d90Test
https://doi.org/10.1016/j.bmc.2006.07.023Test -
4
المؤلفون: Marc Browning, John W. Russell, Astrid A. Ortiz, Gail K. Mattson, Sharon Flowers, Rachel T. McGovern, Mendi A. Higgins, Graham S. Poindexter, Wendy Clarke, Stefanie Rassnick, James E. Grace, John B. Hogan, Lawrence G. Iben, Ildiko Antal-Zimanyi, Kevin W. Gillman
المصدر: Bioorganic & Medicinal Chemistry. 14:5517-5526
مصطلحات موضوعية: medicine.medical_specialty, Time Factors, Clinical Biochemistry, Pharmaceutical Science, Neuropeptide, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Eating, Inhibitory Concentration 50, Radioligand Assay, Structure-Activity Relationship, Pharmacokinetics, In vivo, Internal medicine, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Chemistry, Organic Chemistry, Imidazoles, Antagonist, In vitro, Rats, Receptors, Neuropeptide Y, Bioavailability, Endocrinology, Anorectic, Molecular Medicine, Anti-Obesity Agents
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::82e01d7cffb040b3b57b8baf558bbd78Test
https://doi.org/10.1016/j.bmc.2006.04.042Test -
5
المؤلفون: Federica Balzano, Giuseppe Sicoli, Donatella Paolino, Salvatore Guccione, Ignacio Aldana, Carmen Frı́glola, Antonio Monge, Gloria Uccello-Barretta
المصدر: Bioorganic & Medicinal Chemistry. 12:447-458
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Molecular model, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Context (language use), Biochemistry, Inclusion compound, chemistry.chemical_compound, Cyclohexanes, Modelling methods, Drug Discovery, Humans, Molecular Biology, chemistry.chemical_classification, Cyclodextrins, Drug Carriers, Sulfonamides, Cyclodextrin, beta-Cyclodextrins, Organic Chemistry, Antagonist, Stereoisomerism, Receptors, Neuropeptide Y, chemistry, Drug delivery, Molecular Medicine, Drug carrier, Bromobenzenes
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4b65991c5b7cc0e71e8b7adcbab12926Test
https://doi.org/10.1016/j.bmc.2003.10.033Test -
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المؤلفون: Yves Pascal, Alain Calvet, Ingebrigt Sylte, C.R. Andrianjara, Svein G. Dahl
المصدر: Bioorganic & Medicinal Chemistry. 7:2737-2748
مصطلحات موضوعية: Models, Molecular, Molecular model, Protein Conformation, Stereochemistry, Static Electricity, Clinical Biochemistry, Pharmaceutical Science, In Vitro Techniques, Arginine, Ligands, Pancreatic Polypeptide, Biochemistry, mental disorders, Drug Discovery, Humans, Pancreatic polypeptide, Neuropeptide Y, Peptide YY, Receptor, Molecular Biology, chemistry.chemical_classification, BIBP-3226, Binding Sites, Chemistry, Organic Chemistry, Ligand (biochemistry), Neuropeptide Y receptor, Receptors, Neuropeptide Y, Amino acid, Thermodynamics, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ae6d2a92fffd38bb1cf5a7f737699c8aTest
https://doi.org/10.1016/s0968-0896Test(99)00229-1