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المؤلفون: Valentina Cecarini, Salima Selmi, Massimiliano Cuccioloni, Chunmei Gong, Laura Bonfili, Yadong Zheng, Manuela Cortese, Mauro Angeletti, Soumaya Kilani, Anna Maria Eleuteri
المصدر: Molecules; Volume 27; Issue 21; Pages: 7591
مصطلحات موضوعية: Prunus armeniaca, Amygdalin, Organic Chemistry, Pharmaceutical Science, Breast Neoplasms, Apoptosis, Analytical Chemistry, Chemistry (miscellaneous), Proteolysis, Drug Discovery, amygdalin, proteasome, autophagy, apoptosis, cancer, apricot kernel extract, Humans, Molecular Medicine, Female, Physical and Theoretical Chemistry
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a03d686e08101ffb374731f8787cd755Test
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المؤلفون: Massimiliano Cuccioloni, Laura Bonfili, Mauro Angeletti, Riccardo Petrelli, Loredana Cappellacci, Anna Maria Eleuteri, Massimo Nabissi, Fabio Marchetti, Riccardo Pettinari, Valentina Cecarini
المصدر: ChemMedChem. 15:105-113
مصطلحات موضوعية: Cell Membrane Permeability, Stereochemistry, media_common.quotation_subject, Serum albumin, Hydrazone, chemistry.chemical_element, Antineoplastic Agents, Apoptosis, 01 natural sciences, Biochemistry, Ruthenium, Cell membrane, chemistry.chemical_compound, Coordination Complexes, Cell Line, Tumor, Drug Discovery, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Internalization, Cytotoxicity, media_common, Pharmacology, chemistry.chemical_classification, Binding Sites, biology, 010405 organic chemistry, Organic Chemistry, Hydrazones, Cell Cycle Checkpoints, DNA, In vitro, 0104 chemical sciences, Molecular Docking Simulation, Kinetics, 010404 medicinal & biomolecular chemistry, medicine.anatomical_structure, chemistry, biology.protein, Nucleic Acid Conformation, Molecular Medicine, Hydroxymethylglutaryl CoA Reductases, Cyclin-Dependent Kinase Inhibitor p27, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6998f8b0f4699db4e3fa2f6f17dbac7aTest
https://doi.org/10.1002/cmdc.201900551Test -
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المؤلفون: Anna Maria Eleuteri, Valentina Cecarini, Allan H. White, Claudio Pettinari, Laura Bonfili, Mauro Angeletti, Riccardo Pettinari, Massimo Nabissi, Massimiliano Cuccioloni, Matteo Mozzicafreddo, Brian W. Skelton, Fabio Marchetti
المصدر: Journal of medicinal chemistry. 57(11)
مصطلحات موضوعية: Chemistry, Stereochemistry, Ligand, Poly ADP ribose polymerase, Biphenyl Compounds, Cell Cycle, chemistry.chemical_element, Antineoplastic Agents, Apoptosis, DNA, Ruthenium, Structure-Activity Relationship, Cell culture, Coordination Complexes, Cell Line, Tumor, Drug Discovery, Cancer cell, Molecular Medicine, DNA fragmentation, Humans, MTT assay, Drug Screening Assays, Antitumor, Pyrazolones
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c66e7a264a29983a9509aab18e6dfeb4Test
https://pubmed.ncbi.nlm.nih.gov/24793593Test -
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المؤلفون: Valentina Cecarini, Matteo Mozzicafreddo, Anna Maria Eleuteri, Fabio Marchetti, Mauro Angeletti, Riccardo Pettinari, Claudio Pettinari, Giulio Lupidi, Laura Bonfili, Massimiliano Cuccioloni
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Proteasome Inhibition, Curcumin, Stereochemistry, chemistry.chemical_element, Antineoplastic Agents, Apoptosis, Oxidative phosphorylation, Biochemistry, Ruthenium, chemistry.chemical_compound, Neoplasms, Drug Discovery, Humans, General Pharmacology, Toxicology and Pharmaceutics, Pharmacology, Organic Chemistry, Biological activity, DNA, HCT116 Cells, Oxidative Stress, chemistry, Proteasome, Molecular Medicine, Drug Screening Assays, Antitumor, Proteasome Inhibitors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::df49f5527322df47321193f3027a81ccTest
http://hdl.handle.net/11581/249367Test -
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المؤلفون: Mauro Angeletti, Laura Bonfili, Matteo Mozzicafreddo, Anna Maria Eleuteri, Valentina Cecarini, Massimiliano Cuccioloni
المصدر: Chemical biologydrug design. 74(1)
مصطلحات موضوعية: Drug, Proteases, Serine Proteinase Inhibitors, media_common.quotation_subject, Endogeny, Biochemistry, Serine, Small Molecule Libraries, Structure-Activity Relationship, Phenols, Catalytic Domain, Drug Discovery, media_common, Pharmacology, chemistry.chemical_classification, Serine protease, Flavonoids, biology, Organic Chemistry, Serine Endopeptidases, Proteolytic enzymes, Polyphenols, Protein Structure, Tertiary, Enzyme, chemistry, Drug Design, biology.protein, Molecular Medicine, Pharmacophore
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a5b5361c81358b32cf902bb157723efdTest
https://pubmed.ncbi.nlm.nih.gov/19519739Test