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المؤلفون: Massimiliano Cuccioloni, Laura Bonfili, Mauro Angeletti, Riccardo Petrelli, Loredana Cappellacci, Anna Maria Eleuteri, Massimo Nabissi, Fabio Marchetti, Riccardo Pettinari, Valentina Cecarini
المصدر: ChemMedChem. 15:105-113
مصطلحات موضوعية: Cell Membrane Permeability, Stereochemistry, media_common.quotation_subject, Serum albumin, Hydrazone, chemistry.chemical_element, Antineoplastic Agents, Apoptosis, 01 natural sciences, Biochemistry, Ruthenium, Cell membrane, chemistry.chemical_compound, Coordination Complexes, Cell Line, Tumor, Drug Discovery, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Internalization, Cytotoxicity, media_common, Pharmacology, chemistry.chemical_classification, Binding Sites, biology, 010405 organic chemistry, Organic Chemistry, Hydrazones, Cell Cycle Checkpoints, DNA, In vitro, 0104 chemical sciences, Molecular Docking Simulation, Kinetics, 010404 medicinal & biomolecular chemistry, medicine.anatomical_structure, chemistry, biology.protein, Nucleic Acid Conformation, Molecular Medicine, Hydroxymethylglutaryl CoA Reductases, Cyclin-Dependent Kinase Inhibitor p27, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6998f8b0f4699db4e3fa2f6f17dbac7aTest
https://doi.org/10.1002/cmdc.201900551Test -
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المؤلفون: Massimiliano Cuccioloni, Matteo Mozzicafreddo, Valentina Cecarini, Mauro Angeletti, Laura Bonfili, Giacomo Rossi, Anna Maria Eleuteri, Jeffrey N. Keller
المصدر: Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease. 1842:127-134
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Cell Survival, Leupeptins, Proteolysis, Blotting, Western, Cysteine Proteinase Inhibitors, Protein degradation, Cathepsin B, Amyloid beta-Protein Precursor, Ubiquitin, Cell Line, Tumor, Autophagy, medicine, Amyloid precursor protein, Humans, Molecular Biology, biology, medicine.diagnostic_test, Adenine, Immunohistochemistry, Cell biology, Amino Acid Substitution, Proteasome, Biochemistry, Mutation, Ubiquitin–proteasome system, biology.protein, Proteasome inhibitor, Molecular Medicine, Mutant Proteins, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6069901796a75d1be793c0cd8b0c0e80Test
https://doi.org/10.1016/j.bbadis.2013.11.002Test -
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المؤلفون: Mauro Angeletti, Jeffrey N. Keller, Massimiliano Cuccioloni, Valentina Cecarini, Laura Bonfili, Matteo Mozzicafreddo, Anna Maria Eleuteri
المصدر: Cellular and molecular life sciences : CMLS. 73(18)
مصطلحات موضوعية: 0301 basic medicine, Proteasome Endopeptidase Complex, Cellular homeostasis, Disease, Biology, Protein aggregation, 03 medical and health sciences, Cellular and Molecular Neuroscience, Ubiquitin, Alzheimer Disease, Autophagy, Humans, Molecular Biology, Pharmacology, Neurons, Cell Biology, Cell biology, Crosstalk (biology), 030104 developmental biology, Proteasome, Chaperone (protein), Proteolysis, biology.protein, Molecular Medicine, Microtubule-Associated Proteins, Molecular Chaperones
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1039127cfc6bdf2107040196d7ed22e4Test
https://pubmed.ncbi.nlm.nih.gov/27120560Test -
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المؤلفون: Mauro Angeletti, Laura Bonfili, Matteo Mozzicafreddo, Anna Maria Eleuteri, Valentina Cecarini, Massimiliano Cuccioloni
المصدر: Chemical biologydrug design. 74(1)
مصطلحات موضوعية: Drug, Proteases, Serine Proteinase Inhibitors, media_common.quotation_subject, Endogeny, Biochemistry, Serine, Small Molecule Libraries, Structure-Activity Relationship, Phenols, Catalytic Domain, Drug Discovery, media_common, Pharmacology, chemistry.chemical_classification, Serine protease, Flavonoids, biology, Organic Chemistry, Serine Endopeptidases, Proteolytic enzymes, Polyphenols, Protein Structure, Tertiary, Enzyme, chemistry, Drug Design, biology.protein, Molecular Medicine, Pharmacophore
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a5b5361c81358b32cf902bb157723efdTest
https://pubmed.ncbi.nlm.nih.gov/19519739Test